Aminodifluorosulfinium Tetrafluoroborate Salts as Stable and Crystalline Deoxofluorinating Reagents von Beaulieu, Francis, Beauregard, Louis-Philippe, Courchesne, Gabriel, Couturier, Michel, LaFlamme, François, L’Heureux, Alexandre

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Conformationally Constrained ortho-Anilino Diaryl Ureas: Discovery of 1‑(2-(1′-Neopentylspiro[indoline-3,4′-piperidine]-1-yl)phenyl)-3-(4-(trifluoromethoxy)phenyl)urea, a Potent, S... von Qiao, Jennifer X, Wang, Tammy C, Ruel, Réjean, Thibeault, Carl, L’Heureux, Alexandre, Schumacher, William A, Spronk, Steven A, Hiebert, Sheldon, Bouthillier, Gilles, Lloyd, John, Pi, Zulan, Schnur, Dora M, Abell, Lynn M, Hua, Ji, Price, Laura A, Liu, Eddie, Wu, Qimin, Steinbacher, Thomas E, Bostwick, Jeffrey S, Chang, Ming, Zheng, Joanna, Gao, Qi, Ma, Baoqing, McDonnell, Patricia A, Huang, Christine S, Rehfuss, Robert, Wexler, Ruth R, Lam, Patrick Y. S

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Aminodifluorosulfinium Salts: Selective Fluorination Reagents with Enhanced Thermal Stability and Ease of Handling von L’Heureux, Alexandre, Beaulieu, Francis, Bennett, Christopher, Bill, David R, Clayton, Simon, LaFlamme, François, Mirmehrabi, Mahmoud, Tadayon, Sam, Tovell, David, Couturier, Michel

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Synthesis of functionalized 7-azaindoles via directed ortho-metalations von L’Heureux, Alexandre, Thibault, Carl, Ruel, Réjean

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Concise and Efficient Synthesis of 4-Fluoro-1H-pyrrolo[2,3-b]pyridine von Thibault, Carl, L'Heureux, Alexandre, Bhide, Rajeev S, Ruel, Réjean

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Deoxofluorination Reactions Using N,N-Disubstituted Aminodifluorosulfinium Tetrafluoroborate Salts von Mahé, Olivier, L’Heureux, Alexandre, Couturier, Michel, Bennett, Christopher, Clayton, Simon, Tovell, David, Beaulieu, Francis, Paquin, Jean-François

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New azole antagonists with high affinity for the P2Y1 receptor von Ruel, Réjean, L’Heureux, Alexandre, Thibeault, Carl, Daris, Jean-Paul, Martel, Alain, Price, Laura A., Wu, Qimin, Hua, Ji, Wexler, Ruth R., Rehfuss, Robert, Lam, Patrick Y.S.

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Potent P2Y1 urea antagonists bearing various cyclic amine scaffolds von Ruel, Réjean, L’Heureux, Alexandre, Thibeault, Carl, Lapointe, Philippe, Martel, Alain, Qiao, Jennifer X., Hua, Ji, Price, Laura A., Wu, Qimin, Chang, Ming, Zheng, Joanna, Huang, Christine S., Wexler, Ruth R., Rehfuss, Robert, Lam, Patrick Y.S.

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New azole antagonists with high affinity for the P2Y(1) receptor von Ruel, Réjean, L'Heureux, Alexandre, Thibeault, Carl, Daris, Jean-Paul, Martel, Alain, Price, Laura A, Wu, Qimin, Hua, Ji, Wexler, Ruth R, Rehfuss, Robert, Lam, Patrick Y S

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Discovery and preclinical studies of 5-isopropyl-6-(5-methyl-1,3,4-oxadiazol-2-yl)- N-(2-methyl-1 H-pyrrolo[2,3- b]pyridin-5-yl)pyrrolo[2,1- f][1,2,4]triazin-4-amine (BMS-645737),... von Ruel, Réjean, Thibeault, Carl, L’Heureux, Alexandre, Martel, Alain, Cai, Zhen-Wei, Wei, Donna, Qian, Ligang, Barrish, Joel C., Mathur, Arvind, D’Arienzo, Celia, Hunt, John T., Kamath, Amrita, Marathe, Punit, Zhang, Yueping, Derbin, George, Wautlet, Barri, Mortillo, Steven, Jeyaseelan, Robert, Henley, Benjamin, Tejwani, Ravindra, Bhide, Rajeev S., Trainor, George L., Fargnoli, Joseph, Lombardo, Louis J.

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Copper-catalyzed coupling of ( S)-1-(3-bromophenyl)-ethylamine and N–H containing heteroarenes using microwave heating von Wu, Yong-Jin, He, Huan, L'Heureux, Alexandre

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Pyranophane Transannular Diels−Alder Approach to (+)-Chatancin:  A Biomimetic Asymmetric Total Synthesis von Soucy, Pierre, L'Heureux, Alexandre, Toró, András, Deslongchamps, Pierre

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( S, E)- N-[1-(3-Heteroarylphenyl)ethyl]-3-(2-fluorophenyl)acrylamides: synthesis and KCNQ2 potassium channel opener activity von L’Heureux, Alexandre, Martel, Alain, He, Huan, Chen, Jie, Sun, Li-Qiang, Starrett, John E., Natale, Joanne, Dworetzky, Steven I., Knox, Ronald J., Harden, David G., Weaver, David, Thompson, Mark W., Wu, Yong-Jin

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Transannular Diels−Alder Studies on the Asymmetric Total Synthesis of Chatancin:  The Pyranophane Approach von Toró, András, L'Heureu, Alexandre, Deslongchamps, Pierre

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(S)-N-[1-(3-Morpholin-4-ylphenyl)ethyl]- 3-phenylacrylamide:  An Orally Bioavailable KCNQ2 Opener with Significant Activity in a Cortical Spreading Depression Model of Migraine von Wu, Yong-Jin, Boissard, Christopher G, Greco, Corinne, Gribkoff, Valentin K, Harden, David G, He, Huan, L'Heureux, Alexandre, Kang, Shing Hong, Kinney, Gene G, Knox, Ronald J, Natale, Joanne, Newton, Amy E, Lehtinen-Oboma, Sanna, Sinz, Michael W, Sivarao, Digavalli V, Starrett, John E, Sun, Li-Qiang, Tertyshnikova, Svetlana, Thompson, Mark W, Weaver, David, Wong, Henry S, Zhang, Lei, Dworetzky, Steven I

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Synthesis and Structure−Activity Relationship of Acrylamides as KCNQ2 Potassium Channel Openers von Wu, Yong-Jin, He, Huan, Sun, Li-Qiang, L'Heureux, Alexandre, Chen, Jie, Dextraze, Pierre, Starrett, John E, Boissard, Christopher G, Gribkoff, Valentin K, Natale, Joanne, Dworetzky, Steven I

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Concise and Efficient Synthesis of 4-Fluoro-1 H -pyrrolo[2,3- b ]pyridine von Thibault, Carl, L'Heureux, Alexandre, Bhide, Rajeev S., Ruel, Réjean

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DISUBSTITUTED-AMINODIFLUOROSULFINIUM SALTS, PROCESS FOR PREPARING SAME AND METHOD OF USE AS DEOXOFLUORINATION REAGENTS von L'HEUREUX, ALEXANDRE, COUTURIER, MICHEL

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Conformationally Constrained ortho- Anilino Diaryl Ureas: Discovery of 1-(2-(1′-Neopentylspiro[indoline-3,4′-piperidine]-1-yl)phenyl)-3-(4-(trifluoromethoxy)phenyl)urea, a Potent,... von Qiao, Jennifer X., Wang, Tammy C., Ruel, Réjean, Thibeault, Carl, L’Heureux, Alexandre, Schumacher, William A., Spronk, Steven A., Hiebert, Sheldon, Bouthillier, Gilles, Lloyd, John, Pi, Zulan, Schnur, Dora M., Abell, Lynn M., Hua, Ji, Price, Laura A., Liu, Eddie, Wu, Qimin, Steinbacher, Thomas E., Bostwick, Jeffrey S., Chang, Ming, Zheng, Joanna, Gao, Qi, Ma, Baoqing, McDonnell, Patricia A., Huang, Christine S., Rehfuss, Robert, Wexler, Ruth R., Lam, Patrick Y. S.

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Disubstituted-aminodifluorosulfinium salts, process for preparing same and method of use as deoxofluorination reagents von L'HEUREUX ALEXANDRE, COUTURIER MICHEL A

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