The specificity of JAK3 kinase inhibitors von Changelian, Paul S., Moshinsky, Deborah, Kuhn, Cyrille F., Flanagan, Mark E., Munchhof, Michael J., Harris, Thomas M., Whipple, David A., Doty, Jonathan L., Sun, Jianmin, Kent, Craig R., Magnuson, Kelly S., Perregaux, David G., Sawyer, Perry S., Kudlacz, Elizabeth M.

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Structure of the Catalytic Domain of Human Polo-like Kinase 1 von Kothe, Michael, Kohls, Darcy, Low, Simon, Coli, Rocco, Cheng, Alan C, Jacques, Suzanne L, Johnson, Theresa L, Lewis, Cristina, Loh, Christine, Nonomiya, Jim, Sheils, Alissa L, Verdries, Kimberly A, Wynn, Thomas A, Kuhn, Cyrille, Ding, Yuan-Hua

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Investigation of the binding pocket of human hematopoietic prostaglandin (PG) D2 synthase (hH-PGDS): A tale of two waters von Trujillo, John I., Kiefer, James R., Huang, Wei, Day, Jacqueline E., Moon, Joseph, Jerome, Gina M., Bono, Christine P., Kornmeier, Christine M., Williams, Melanie L., Kuhn, Cyrille, Rennie, Glen R., Wynn, Thomas A., Carron, Christopher P., Thorarensen, Atli

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Bipiperidinyl Carboxylic Acid Amides as Potent, Selective, and Functionally Active CCR4 Antagonists von Kuhn, Cyrille F., Bazin, Marc, Philippe, Laurence, Zhang, Jiansu, Tylaska, Laurie, Miret, Juan, Bauer, Paul H.

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Research Article: Selectivity-determining Residues in Plk1 von Kothe, Michael, Kohls, Darcy, Low, Simon, Coli, Rocco, Rennie, Glen R., Feru, Frederic, Kuhn, Cyrille, Ding, Yuan-Hua

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Selectivity-determining Residues in Plk1 von Kothe, Michael, Kohls, Darcy, Low, Simon, Coli, Rocco, Rennie, Glen R, Feru, Frederic, Kuhn, Cyrille, Ding, Yuan-Hua

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Design, synthesis and biological evaluation of novel aminothiazoles as antiviral compounds acting against human rhinovirus von Décor, Anne, Grand-Maître, Chantal, Hucke, Oliver, O’Meara, Jeff, Kuhn, Cyrille, -Forget, Léa Constantineau, Brochu, Christian, Malenfant, Eric, Bertrand-Laperle, Mégan, Bordeleau, Josée, Ghiro, Elise, Pesant, Marc, Fazal, Gulrez, Gorys, Vida, Little, Michael, Boucher, Colette, Bordeleau, Sylvain, Turcotte, Pascal, Guo, Tim, Garneau, Michel, Spickler, Catherine, Gauthier, Annick

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Potent and selective thiophene urea-templated inhibitors of S6K von Ye, Ping, Kuhn, Cyrille, Juan, Miret, Sharma, Rahul, Connolly, Brendan, Alton, Gordon, Liu, Hu, Stanton, Robert, Kablaoui, Natasha M.

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Identification of benzofurano[3,2-d]pyrimidin-2-ones, a new series of HIV-1 nucleotide-competing reverse transcriptase inhibitors von Tremblay, Martin, Bethell, Richard C., Cordingley, Michael G., DeRoy, Patrick, Duan, Jianmin, Duplessis, Martin, Edwards, Paul J., Faucher, Anne-Marie, Halmos, Ted, James, Clint A., Kuhn, Cyrille, Lacoste, Jean-Éric, Lamorte, Louie, LaPlante, Steven R., Malenfant, Éric, Minville, Joannie, Morency, Louis, Morin, Sébastien, Rajotte, Daniel, Salois, Patrick, Simoneau, Bruno, Tremblay, Sonia, Sturino, Claudio F.

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Discovery of Potent, Orally Bioavailable Inhibitors of Human Cytomegalovirus von Fader, Lee, Brault, Martine, Desjardins, Jessica, Dansereau, Nathalie, Lamorte, Louie, Tremblay, Sonia, Bilodeau, François, Bordeleau, Josée, Duplessis, Martin, Gorys, Vida, Gillard, James, Gleason, James L, James, Clint, Joly, Marc-André, Kuhn, Cyrille, Llinas-Brunet, Montse, Luo, Laibin, Morency, Louis, Morin, Sébastien, Parisien, Mathieu, Poirier, Maude, Thibeault, Carl, Trinh, Thao, Sturino, Claudio, Srivastava, Sanjay, Yoakim, Christiane, Franti, Michael

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Selective cell adhesion inhibitors: Barbituric acid based α4β7—MAdCAM inhibitors von Harriman, Geraldine C., Brewer, Matthias, Bennett, Robert, Kuhn, Cyrille, Bazin, Marc, Larosa, Greg, Skerker, Paul, Cochran, Nancy, Gallant, Debra, Baxter, Deborah, Picarella, Dominic, Jaffee, Bruce, Luly, Jay R., Briskin, Michael J.

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Selective cell adhesion inhibitors: Barbituric acid based alpha 4 beta 7 - MAdCAM inhibitors von Harriman, Geraldine C, Brewer, Matthias, Bennett, Robert, Kuhn, Cyrille, Bazin, Marc, Larosa, Greg, Skerker, Paul, Cochran, Nancy, Gallant, Debra, Baxter, Deborah, Picarella, Dominic, Jaffee, Bruce, Luly, Jay R, Briskin, Michael J

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SPRK1 INHIBITORS AND METHODS OF USE von KUHN, Cyrille, LI, Lianhai

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Enhanced selectivity profile of pyrazole-urea based DFG-out p38α inhibitors von Liu, Hu, Kuhn, Cyrille, Feru, Frederic, Jacques, Suzanne L., Deshmukh, Gayatri D., Ye, Ping, Rennie, Glen R., Johnson, Theresa, Kazmirski, Steven, Low, Simon, Coli, Rocco, Ding, Yuan-hua, Cheng, Alan C., Tecle, Haile, English, Jessie M., Stanton, Robert, Wu, Joe C.

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Enhanced selectivity profile of pyrazole-urea based DFG-out p38a inhibitors von Liu, Hu, Kuhn, Cyrille, Feru, Frederic, Jacques, Suzanne L, Deshmukh, Gayatri D, Ye, Ping, Rennie, Glen R, Johnson, Theresa, Kazmirski, Steven, Low, Simon, Coli, Rocco, Ding, Yuan-Hua, Cheng, Alan C, Tecle, Haile, English, Jessie M, Stanton, Robert, Wu, Joe C

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Design, Synthesis and Potential Utility of Fluorescence Probes that Target DFG-out Conformation of p38α for High Throughput Screening Binding Assay von Tecle, Haile, Feru, Frederic, Liu, Hu, Kuhn, Cyrille, Rennie, Glen, Morris, Mark, Shao, Jiangxing, Cheng, Alan C, Gikunju, Diana, Miret, Juan, Coli, Rocco, Xi, Simon (Hualin), Clugston, Susan L, Low, Simon, Kazmirski, Steven, Ding, Yuan-Hua, Cao, Qing, Johnson, Theresa L, Deshmukh, Gayatri D, DiNitto, Jonathan P, Wu, Joe C, English, Jessie M

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Domino Aza-Claisen/Mannich Cyclization Reaction from a Chiral α-Alkoxy Enamine or Sequential Alkylation of an α-Alkoxy Ester Enolate or Nitrile Anion, Followed by an Intramolecular... von Kuhn, Cyrille, Skaltsounis, Leandros, Monneret, Claude, Florent, Jean-Claude

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Synthesis and biological evaluation of new cross-conjugated dienone marine prostanoid analogues von Kuhn, Cyrille, Roulland, Emmanuel, Madelmont, Jean-Claude, Monneret, Claude, Florent, Jean-Claude

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Solid-Phase Enolate Chemistry Investigated Using HR-MAS NMR Spectroscopy von Fruchart, Jean-Sébastien, Lippens, Guy, Kuhn, Cyrille, Gras-Masse, Hélène, Melnyk, Oleg

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Efficient Use of the Iron Ortho-Nitrophenylporphyrin Chloride to Mimic Biological Oxidations of Dimethylaminoantipyrine von Bazin, Marc J., Shi, Helen, Delaney, Jeannine, Kline, Billie, Zhu, Zhendong, Kuhn, Cyrille, Berlioz, Francoise, Farley, Kathleen A., Fate, Gwen, Lam, Wing, Walker, Gregory S., Yu, Linning, Pollastri, Michael P.

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