Synthesis and SAR of aminoalkoxy-biaryl-4-carboxamides: Novel and selective histamine H3 receptor antagonists von FAGHIH, Ramin, DWIGHT, Wesley, JIA BAO PAN, FOX, Gerard B, KRUEGER, Kathy M, ESBENSHADE, Timothy A, MCVEY, Jill M, MARSH, Kennan, BENNANI, Youssef L, HANCOCK, Arthur A

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Structure-activity relationships of non-imidazole H3 receptor ligands. Part 2: Binding preference for D-amino acids motifs von FAGHIH, Ramin, DWIGHT, Wesley, KRUEGER, Kathy M, FOX, Gerard B, HANCOCK, Arthur A, BENNANI, Youssef L, BLACK, Larry, HUAQING LIU, GENTLES, Robert, PHELAN, Kathleen, ESBENSHADE, Timothy A, IRELAND, Lynne, MILLER, Thomas R, KANG, Chae-Hee

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Structure-activity relationships of non-imidazole H3 receptor ligands. Part 3: 5-Substituted 3-phenyl-1,2,4-oxadiazoles as potent antagonists von GFESSER, Gregory A, ZHANG, Henry, KRUEGER, Kathy M, BENNANI, Youssef L, HANCOCK, Arthur A, FAGHIH, Ramin, DINGES, Jurgen, FOX, Gerard B, PAN, Jia Bao, ESBENSHADE, Timothy A, YAO, Betty B, WITTE, David, MILLER, Thomas R, KANG, Chae-Hee

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D-Amino Acid Homopiperazine Amides: Discovery of A-320436, a Potent and Selective Non-Imidazole Histamine H3-Receptor Antagonist von Curtis, Michael P., Dwight, Wesley, Pratt, John, Cowart, Marlon, Esbenshade, Timothy A., Krueger, Kathy M., Fox, Gerard B., Pan, Jia Bao, Pagano, Thomas G., Hancock, Arthur A., Faghih, Ramin, Bennani, Youssef L.

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Synthesis and SAR of aminoalkoxy-biaryl-4-carboxamides: novel and selective histamine H 3 receptor antagonists von Faghih, Ramin, Dwight, Wesley, Pan, Jia Bao, Fox, Gerard B., Krueger, Kathy M., A. Esbenshade, Timothy, McVey, Jill M., Marsh, Kennan, Bennani, Youssef L., Hancock, Arthur A.

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Structure–Activity relationships of non-imidazole H 3 Receptor ligands. Part 2: binding preference for d-Amino acids motifs von Faghih, Ramin, Dwight, Wesley, Black, Larry, Liu, Huaqing, Gentles, Robert, Phelan, Kathleen, Esbenshade, Timothy A, Ireland, Lynne, Miller, Thomas R, Kang, Chae-Hee, Krueger, Kathy M, Fox, Gerard B, Hancock, Arthur A, Bennani, Youssef L

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Structure–activity relationships of non-imidazole H 3 receptor ligands. Part 3: 5-Substituted 3-phenyl-1,2,4-oxadiazoles as potent antagonists von Gfesser, Gregory A., Zhang, Henry, Dinges, Jurgen, Fox, Gerard B., Pan, Jia Bao, Esbenshade, Timothy A., Yao, Betty B., Witte, David, Miller, Thomas R., Kang, Chae-Hee, Krueger, Kathy M., Bennani, Youssef L., Hancock, Arthur A., Faghih, Ramin

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D‐Amino Acid Homopiperazine Amides: Discovery of A‐320436, a Potent and Selective Non‐Imidazole Histamine H 3 ‐Receptor Antagonist von Curtis, Michael P., Dwight, Wesley, Pratt, John, Cowart, Marlon, Esbenshade, Timothy A., Krueger, Kathy M., Fox, Gerard B., Pan, Jia Bao, Pagano, Thomas G., Hancock, Arthur A., Faghih, Ramin, Bennani, Youssef L.

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Structure-activity relationships of non-imidazole H(3) receptor ligands. Part 3: 5-Substituted 3-phenyl-1,2,4-oxadiazoles as potent antagonists von Gfesser, Gregory A, Zhang, Henry, Dinges, Jurgen, Fox, Gerard B, Pan, Jia Bao, Esbenshade, Timothy A, Yao, Betty B, Witte, David, Miller, Thomas R, Kang, Chae-Hee, Krueger, Kathy M, Bennani, Youssef L, Hancock, Arthur A, Faghih, Ramin

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Structure-activity relationships of non-imidazole H(3) receptor ligands. Part 2: binding preference for D-amino acids motifs von Faghih, Ramin, Dwight, Wesley, Black, Larry, Liu, Huaqing, Gentles, Robert, Phelan, Kathleen, Esbenshade, Timothy A, Ireland, Lynne, Miller, Thomas R, Kang, Chae-Hee, Krueger, Kathy M, Fox, Gerard B, Hancock, Arthur A, Bennani, Youssef L

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D-amino acid homopiperazine amides: discovery of A-320436, a potent and selective non-imidazole histamine H(3)-receptor antagonist von Curtis, Michael P, Dwight, Wesley, Pratt, John, Cowart, Marlon, Esbenshade, Timothy A, Krueger, Kathy M, Fox, Gerard B, Pan, Jia Bao, Pagano, Thomas G, Hancock, Arthur A, Faghih, Ramin, Bennani, Youssef L

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Fecal Microbiota Composition Drives Immune Activation in HIV-infected Individuals von Neff, Charles Preston, Krueger, Owen, Xiong, Kathy, Arif, Sabrina, Nusbacher, Nichole, Schneider, Jennifer M., Cunningham, Annie W., Armstrong, Abigail, Li, Sam, McCarter, Martin D., Campbell, Thomas B., Lozupone, Catherine A., Palmer, Brent E.

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Development of Orally Efficacious Allosteric Inhibitors of TNFα via Fragment-Based Drug Design von Dietrich, Justin D, Longenecker, Kenton L, Wilson, Noel S, Goess, Christian, Panchal, Sanjay C, Swann, Steven L, Petros, Andrew M, Hobson, Adrian D, Ihle, David, Song, Danying, Richardson, Paul, Comess, Kenneth M, Cox, Philip B, Dombrowski, Amanda, Sarris, Kathy, Donnelly-Roberts, Diana L, Duignan, David B, Gomtsyan, Arthur, Jung, Paul, Krueger, A Chris, Mathieu, Suzanne, McClure, Andrea, Stoll, Vincent S, Wetter, Jill, Mankovich, John A, Hajduk, Philip J, Vasudevan, Anil, Stoffel, Robert H, Sun, Chaohong

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Genome-wide analysis identifies 12 loci influencing human reproductive behavior von Barban, Nicola, de Vlaming, Ronald, Vaez, Ahmad, Tropf, Felix C, Shen, Xia, Chasman, Daniel I, Nolte, Ilja M, van der Laan, Sander W, Perry, John R B, Ahluwalia, Tarunveer S, Bakshi, Andrew, Ben-Avraham, Danny, Bjornsdottir, Gyda, Bonder, Marc Jan, Bui, Minh, Cavadino, Alana, Chavarro, Jorge E, Turman, Constance, Esko, Tõnu, Falahi, Fahimeh, Fontana, Mark Alan, Franke, Lude, Gandin, Ilaria, Gieger, Christian, Guo, Xiuqing, Hofer, Edith, Huang, Hongyan, Joshi, Peter K, Karlsson, Robert, Kifley, Annette, Lagou, Vasiliki, Liu, Tian, Makalic, Enes, Meddens, S Fleur W, Miller, Mike, van der Most, Peter J, Myhre, Ronny, Kalafati, Ioanna Panagiota, Porcu, Eleonora, Rietveld, Cornelius A, Ryan, Kathleen A, Saba, Yasaman, Schmidt, Daniel, Tönjes, Anke, Wellmann, Juergen, Willeit, Peter, Zhao, Wei, Zhernakova, Daria V, Balkau, Beverley, Barzilai, Nir, Bisgaard, Hans, Boomsma, Dorret I, Cappellani, Stefania, Ciullo, Marina, Cox, Simon R, Davey-Smith, George, Deary, Ian J, Deloukas, Panos, Eriksson, Johan G, Faul, Jessica D, Greiser, Karin Halina, de Haan, Hugoline G, Harris, Tamara B, Homuth, Georg, Holliday, Elizabeth G, Jugessur, Astanand, Kardia, Sharon L R, Lachance, Genevieve, Liu, Yongmei, Lucht, Michael, Luoto, Riitta, Mellström, Dan, Milani, Lili, Ohlsson, Claes, Olsen, Jørn, Ong, Ken K, Perola, Markus, Peyser, Patricia A, Pirastu, Mario, Raitakari, Olli, Rudan, Igor, Schmidt, Helena, Schmidt, Reinhold, Schupf, Nicole, Smit, Johannes, Stumvoll, Michael, Swertz, Morris A, Thurik, A Roy, Uitterlinden, André G, Vaccargiu, Simona, Vitart, Veronique, Vuckovic, Dragana, Wang, Jie Jin, Wareham, Nicholas J, Willemsen, Gonneke, Willeit, Johann, Krueger, Robert F, Cesarini, David, Koellinger, Philipp D, Mills, Melinda C

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Early-Life Outcomes in Relation to Social Determinants of Health for Children Born Extremely Preterm von Bell, Edward F., Alksninis, Barbara, Hoffman, Laurie, Leach, Teresa M., Ventura, Suzy, Hibbs, Anna Maria, Walsh, Michele C., Yalcinkaya, Gulgun, Holmes, Anne, Johnson, Kathy, Beiersdorfer, Traci, Fischer, Estelle E., Hessling, Jody, Malcolm, William F., Grimes, Sandra, Gustafson, Kathryn E., Bose, Gennie, Rhodes-Ryan, Ginger, Patel, Ravi M., Carlton, David P., Bottcher, Diane I., Higgins, Rosemary D., Smiley, Lucy, Duncan, Andrea, Stephens, Emily K., Allain, Elizabeth, Green, Charles, Jones, Patrick M., Morris, Brenda H., Wright, Sharon L., Nelin, Leif D., Slaughter, Jonathan L., Fortney, Christine A., Levengood, Katelyn, Batterson, Nancy, Sullivan, Rox Ann, Fowler, Aubrey, Tonneman, Jill, Chao, Michelle, Beckford, Demi R., Baugher, Hallie, Hanlon, Cory, McCool, Jacqueline, Bann, Carla M., Crawford, Margaret M., Bentley, Barbara, Bruno, Elizabeth, Palmquist, Andrew W., Proud, Melinda S., John, Nicholas H. St, Wager, Natalie, Church, Paige T., Sibley, Cecelia E., Nelson, Kathleen G., Preskitt, Julie, Purdy, Isabell B., Vaucher, Yvonne E., Bell, Edward F., Colaizy, Tarah T., Widness, John A., Goeke, Claire A., Walker, Jacky R., Henning, Megan M., Ellsbury, Dan L., Bauer, Charles R., Calejo, Maria, Berkowits, Michelle Harwood, Watterberg, Kristi L., Catts, Christine, Vangala, Saritha, Boylin, Elizabeth, Maffett, Deanna, Sabaratnam, Premini, Scorsone, Ann Marie, Wadkins, Holly I.M., Yost, Kelley, Li, Emily, Brion, Luc P., Heyne, Roy J., Adams, Sally S., Guzman, Alicia, Heyne, Elizabeth T., McDougald, E. Rebecca, Morgan, Janet S., Minton, Stephen D., Sheffield, Mark J., Rau, Carrie A., Jordan, Jamie, Steffen, Michael, Weaver-Lewis, Kimberlee, Zanetti, Karen, Jackson, Barbara G., Halfond, Raquel, Waldrep, Ellen L., Shankaran, Seetha, Panaitescu, Bogdan, Wiggins, Stephanie A., Jacobs, Harris, Butler, Christine G., Romano, Elaine

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Efalizumab (anti-CD11a)-induced increase in peripheral blood leukocytes in psoriasis patients is preferentially mediated by altered trafficking of memory CD8+ T cells into lesional... von Vugmeyster, Yulia, Kikuchi, Toyoko, Lowes, Michelle A., Chamian, Francesca, Kagen, Mark, Gilleaudeau, Patricia, Lee, Edmund, Howell, Kathy, Bodary, Sarah, Dummer, Wolfgang, Krueger, James G.

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Rapid Development of an Integrated Network Infrastructure to Conduct Phase 3 COVID-19 Vaccine Trials von Mena Lora, Alfredo J, Long, Jessica E, Huang, Yunda, Baden, Lindsey R, El Sahly, Hana M, Follmann, Dean, Goepfert, Paul, Gray, Glenda, Grinsztejn, Beatriz, Kotloff, Karen, Rouphael, Nadine, Sobieszczyk, Magdelena, Walsh, Stephen R, Andriesen, Jessica, Shah, Karan A, Zhang, Yuanyuan, Gilbert, Peter, Janes, Holly, Gay, Cynthia L, Falsey, Ann R, Tripp, Rebecca L, Gorman, Richard L, Tong, Tina, Marovich, Mary, Neuzil, Kathleen, Corey, Lawrence, Kublin, James G

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Cyclopropylamino Acid Amide as a Pharmacophoric Replacement for 2,3-Diaminopyridine. Application to the Design of Novel Bradykinin B1 Receptor Antagonists von Wood, Michael R, Schirripa, Kathy M, Kim, June J, Wan, Bang-Lin, Murphy, Kathy L, Ransom, Richard W, Chang, Raymond S. L, Tang, Cuyue, Prueksaritanont, Thomayant, Detwiler, Theodore J, Hettrick, Lisa A, Landis, Elizabeth R, Leonard, Yvonne M, Krueger, Julie A, Lewis, Sidney D, Pettibone, Douglas J, Freidinger, Roger M, Bock, Mark G

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Baseline Features and Reasons for Nonparticipation in the Colonoscopy Versus Fecal Immunochemical Test in Reducing Mortality From Colorectal Cancer (CONFIRM) Study, a Colorectal Ca... von Robertson, Douglas J, Dominitz, Jason A, Beed, Alexander, Boardman, Kathy D, Del Curto, Barbara J, Guarino, Peter D, Imperiale, Thomas F, LaCasse, Andrew, Larson, Meaghan F, Gupta, Samir, Lieberman, David, Planeta, Beata, Shaukat, Aasma, Sultan, Shanaz, Menees, Stacy B, Saini, Sameer D, Schoenfeld, Philip, Goebel, Stephan, von Rosenvinge, Erik C, Baffy, Gyorgy, Halasz, Ildiko, Pedrosa, Marcos C, Kahng, Lyn Sue, Cassim, Riaz, Greer, Katarina B, Kinnard, Margaret F, Bhatt, Divya B, Dunbar, Kerry B, Harford, Jr, William V, Mengshol, John A, Olson, Jed E, Patel, Swati G, Antaki, Fadi, Fisher, Deborah A, Sullivan, Brian A, Lenza, Christopher, Prajapati, Devang N, Wong, Helen, Beyth, Rebecca, Lieb, 2nd, John G, Manlolo, Joseph, Ona, Fernando V, Cole, Rhonda A, Khalaf, Natalia, Kahi, Charles J, Kohli, Divyanshoo Rai, Rai, Tarun, Sharma, Prateek, Anastasiou, Jiannis, Hagedorn, Curt, Fernando, Ronald S, Jackson, Christian S, Jamal, M Mazen, Lee, Robert H, Merchant, Farrukh, May, Folasade P, Pisegna, Joseph R, Omer, Endashaw, Parajuli, Dipendra, Said, Adnan, Nguyen, Toan D, Tombazzi, Claudio Ruben, Feldman, Paul A, Jacob, Leslie, Koppelman, Rachel N, Lehenbauer, Kyle P, Desai, Deepak S, Madhoun, Mohammad F, Tierney, William M, Ho, Minh Q, Hockman, Heather J, Lopez, Christopher, Carter Paulson, Emily, Tobi, Martin, Pinillos, Hugo L, Young, Michele, Ho, Nancy C, Mascarenhas, Ranjan, Promrat, Kirrichai, Mutha, Pritesh R, Pandak, Jr, William M, Shah, Tilak, Schubert, Mitchell, Pancotto, Frank S, Gawron, Andrew J, Underwood, Amelia E, Ho, Samuel B, Magno-Pagatzaurtundua, Priscilla, Toro, Doris H, Beymer, Charles H, Kaz, Andrew M, Elwing, Jill, Gill, Jeffrey A, Goldsmith, Susan F, Yao, Michael D, Protiva, Petr, Pohl, Heiko, Kyriakides, Tassos

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Cyclopropylamino Acid Amide as a Pharmacophoric Replacement for 2,3-Diaminopyridine. Application to the Design of Novel Bradykinin B 1 Receptor Antagonists von Wood, Michael R., Schirripa, Kathy M., Kim, June J., Wan, Bang-Lin, Murphy, Kathy L., Ransom, Richard W., Chang, Raymond S. L., Tang, Cuyue, Prueksaritanont, Thomayant, Detwiler, Theodore J., Hettrick, Lisa A., Landis, Elizabeth R., Leonard, Yvonne M., Krueger, Julie A., Lewis, Sidney D., Pettibone, Douglas J., Freidinger, Roger M., Bock, Mark G.

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