Diastereoselective One-Pot Knoevenagel Condensation/Corey–Chaykovsky Cyclopropanation von Clemens, Jeremy J, Asgian, Juliana L, Busch, Brett B, Coon, Timothy, Ernst, Justin, Kaljevic, Leonard, Krenitsky, Paul J, Neubert, Timothy D, Schweiger, Edwin J, Termin, Andreas, Stamos, Dean

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Synthesis of the ( S, S, S)-diastereomer of the 15-membered biaryl ring system of RP 66453 von Krenitsky, Paul J., Boger, Dale L.

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Preparation of the 14-membered l, l-cycloisodityrosine subunit of RP 66453 von Krenitsky, Paul J., Boger, Dale L.

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CYCLIN-DEPENDENT KINASE DEGRADING COMPOUNDS von MENDY, Derek, MERCURIO, Frank, KRENITSKY, Paul J, XIE, Weilin, HAUGHEY, Michael P, ELSNER, Jan, PLANTEVIN-KRENITSKY, Veronique

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CK1 alpha AND DUAL CK1 alpha / GSPT1 DEGRADING COMPOUNDS von Sapienza, John, Haughey, Michael P, Elsner, Jan, Plantevin-Krenitsky, Veronique, Xie, Weilin, Mendy, Derek, Mercurio, Frank, Krenitsky, Paul J, Papa, Patrick W

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MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR von ZHOU, Jinglan, MILLER, Mark, Thomas, KHATUYA, Haripada, FRIEMAN, Bryan, A, CLEVELAND, Thomas, HADIDA RUAH, Sara S, BEAR, Brian, GROOTENHUIS, Peter, Diederik Jan, SILINA, Alina, COON, Timothy, Richard, UY, Johnny, KRENITSKY, Paul, J, CLEMENS, Jeremy

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MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR von ZHOU, Jinglan, MILLER, Mark, Thomas, KHATUYA, Haripada, FRIEMAN, Bryan, A, CLEVELAND, Thomas, HADIDA RUAH, Sara S, BEAR, Brian, GROOTENHUIS, Peter, Diederik Jan, SILINA, Alina, COON, Timothy, Richard, UY, Johnny, KRENITSKY, Paul, J, CLEMENS, Jeremy

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Divergent mechanisms for the dealkoxycarbonylation of a 2-(3-azetidinyl)malonate by chloride and cyanide von Gilligan, Paul J., Krenitsky, Paul J.

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MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR von ZHOU, Jinglan, MILLER, Mark, Thomas, KHATUYA, Haripada, FRIEMAN, Bryan, A, CLEVELAND, Thomas, HADIDA RUAH, Sara S, BEAR, Brian, GROOTENHUIS, Peter, Diederik Jan, SILINA, Alina, COON, Timothy, Richard, UY, Johnny, KRENITSKY, Paul, J, CLEMENS, Jeremy

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Modulators of cystic fibrosis transmembrane conductance regulator von Hadida Ruah, Sara S, Khatuya, Haripada, Cleveland, Thomas, Silina, Alina, Uy, Johnny, Frieman, Bryan A, Clemens, Jeremy, Coon, Timothy Richard, Grootenhuis, Peter Diederik Jan, Zhou, Jinglan, Miller, Mark Thomas, Bear, Brian, Krenitsky, Paul J

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MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR von ZHOU, Jinglan, MILLER, Mark, Thomas, KHATUYA, Haripada, FRIEMAN, Bryan, A, CLEVELAND, Thomas, HADIDA RUAH, Sara S, BEAR, Brian, GROOTENHUIS, Peter, Diederik Jan, SILINA, Alina, COON, Timothy, Richard, UY, Johnny, KRENITSKY, Paul, J, CLEMENS, Jeremy

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Synthesis of the (S,S,S)-Diastereomer (I) of the 15-Membered Biaryl Ring System of RP 66453 von Krenitsky, Paul J., Boger, Dale L.

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ChemInform Abstract: Preparation of the 14-Membered L,L-Cycloisodityrosine Subunit of RP 66453 von Krenitsky, Paul J., Boger, Dale L.

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Automated multi-scale computational pathotyping (AMSCP) of inflamed synovial tissue von Bell, Richard D., Brendel, Matthew, Konnaris, Maxwell A., Xiang, Justin, Otero, Miguel, Fontana, Mark A., Bai, Zilong, Krenitsky, Daria M., Meednu, Nida, Rangel-Moreno, Javier, Scheel-Toellner, Dagmar, Carr, Hayley, Nayar, Saba, McMurray, Jack, DiCarlo, Edward, Anolik, Jennifer H., Donlin, Laura T., Orange, Dana E., Kenney, H. Mark, Schwarz, Edward M., Filer, Andrew, Ivashkiv, Lionel B., Wang, Fei

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When structure–affinity relationships meet structure–kinetics relationships: 3-((Inden-1-yl)amino)-1-isopropyl-cyclopentane-1-carboxamides as CCR2 antagonists von Vilums, Maris, Zweemer, Annelien J.M., Barmare, Farhana, van der Gracht, Anouk M.F., Bleeker, Dave C.T., Yu, Zhiyi, de Vries, Henk, Gross, Raymond, Clemens, Jeremy, Krenitsky, Paul, Brussee, Johannes, Stamos, Dean, Saunders, John, Heitman, Laura H., IJzerman, Adriaan P.

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Structure–Kinetic RelationshipsAn Overlooked Parameter in Hit-to-Lead Optimization: A Case of Cyclopentylamines as Chemokine Receptor 2 Antagonists von Vilums, Maris, Zweemer, Annelien J. M, Yu, Zhiyi, de Vries, Henk, Hillger, Julia M, Wapenaar, Hannah, Bollen, Ilse A. E, Barmare, Farhana, Gross, Raymond, Clemens, Jeremy, Krenitsky, Paul, Brussee, Johannes, Stamos, Dean, Saunders, John, Heitman, Laura H, IJzerman, Adriaan P

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Synthesis, Corticotropin-Releasing Factor Receptor Binding Affinity, and Pharmacokinetic Properties of Triazolo-, Imidazo-, and Pyrrolopyrimidines and -pyridines von Chorvat, Robert J, Bakthavatchalam, Rajagopal, Beck, James P, Gilligan, Paul J, Wilde, Richard G, Cocuzza, Anthony J, Hobbs, Frank W, Cheeseman, Robert S, Curry, Matthew, Rescinito, Joseph P, Krenitsky, Paul, Chidester, Dennis, Yarem, Jerry A, Klaczkiewicz, John D, Hodge, C. Nicholas, Aldrich, Paul E, Wasserman, Zelda R, Fernandez, Christine H, Zaczek, Robert, Fitzgerald, Lawrence W, Huang, Shiew-Mei, Shen, Helen L, Wong, Y. Nancy, Chien, Ben M, Quon, Check Y, Arvanitis, Argyrios

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MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR von Gross, Raymond Stanley, Clemens, Jeremy J, Cleveland, Thomas, Binch, Hayley Marie, Uy, Johnny, Nicholls, Georgia McGaughey, Marelius, Gulin Erdogan, Termin, Andreas P, Krenitsky, Paul John, Pierre, Fabrice Jean Denis, Khatuya, Haripada, Lin, Chun-Chieh, Silina, Alina, Conroy, Erica, McCartney, Jason, Frieman, Bryan A, Coon, Timothy Richard, Bear, Brian Richard, Arumugam, Vijayalaksmi, Grootenhuis, Peter Diederik Jan, Joshi, Pramod Virupax, Zhou, Jinglan, Miller, Mark Thomas, Melillo, Vito, Anderson, Corey, Hadida-Ruah, Sara Sabina

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MODULATOR OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR, PHARMACEUTICAL COMPOSITIONS, METHODS OF TREATMENT, AND PROCESS FOR MAKING THE MODULATOR von GROSS, Raymond, Stanley, ABELA, Alexander, Russell, MCCARTNEY, Jason, CLEVELAND, Thomas, KANG, Ping, KESHAVARZ-SHOKRI, Ali, JOSHI, Pramod, Virupax, STAVROPOULOS, Kathy, ALCACIO, Timothy, KHATUYA, KHATUYA, Haripada, TERMIN, Andreas, P, BAEK, Minson, SHI, Yi, SHRESTHA, Muna, FERRIS,, Lori, Ann, GROOTENHUIS, Peter Diederik, Jan, HSIA, Clara, Kuang-Ju, KRENITSKY, Paul, John, ANGELL, Paul, Timothy, MILLER, Mark, Thomas, ANDERSON, Corey, PARASELLI, Prasuna, YOUNG, Tomothy, John, ZHOU,, Jinglan, GULEVICH, Anton, VAN GOOR, Fredrik, F, UY, Johnny, CLEMENS, Jeremy, J, HADIDA RUAH, Sara, Sabina, PIERRE, Fa brice Jean, Denis, SIESEL, David, Andrew, HUGHES, Robert, M

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Modulators of cystic fibrosis transmembrane conductance regulator von Gross, Raymond Stanley, Mccartney, Jason, Clemens, Jeremy J, Cleveland, Thomas, Binch, Hayley Marie, Uy, Johnny, Marelius, Gulin Erdogan, Termin, Andreas P, Krenitsky, Paul John, Pierre, Fabrice Jean Denis, Khatuya, Haripada, Lin, Chun-Chieh, Silina, Alina, Conroy, Erica, Frieman, Bryan A, Coon, Timothy Richard, Bear, Brian Richard, Arumugam, Vijayalaksmi, Grootenhuis, Peter Diederik Jan, Joshi, Pramod Virupax, Nicholls, Georgia Mcgaughey, Zhou, Jinglan, Miller, Mark Thomas, Melillo, Vito, Anderson, Corey, Hadida-Ruah, Sara Sabina

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