Biologically active compounds based on the privileged 2-imidazoline scaffold: The world beyond adrenergic/imidazoline receptor modulators von Krasavin, Mikhail

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Spirocyclic Motifs in Natural Products von Chupakhin, Evgeny, Babich, Olga, Prosekov, Alexander, Asyakina, Lyudmila, Krasavin, Mikhail

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Synthetic Studies towards CH‐Diazomethane Sulfonamides: a Novel Type of Diazo Reagents von Bubyrev, Andrey, Dar'in, Dmitry, Kantin, Grigory, Krasavin, Mikhail

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Multicomponent Reactions Involving Diazo Reagents: A 5-Year Update von Bakulina, Olga, Inyutina, Anna, Dar'in, Dmitry, Krasavin, Mikhail

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Diazocarbonyl and Related Compounds in the Synthesis of Azoles von Budeev, Anton, Kantin, Grigory, Dar'in, Dmitry, Krasavin, Mikhail

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Conjugates of Iron-Transporting N-Hydroxylactams with Ciprofloxacin von Bakulina, Olga, Bannykh, Anton, Levashova, Ekaterina, Krasavin, Mikhail

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Exploration of Spirocyclic Derivatives of Ciprofloxacin as Antibacterial Agents von Lukin, Alexei, Chudinov, Mikhail, Vedekhina, Tatiana, Rogacheva, Elizaveta, Kraeva, Lyudmila, Bakulina, Olga, Krasavin, Mikhail

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Synthesis of spirocyclic tetrahydroisoquinolines (spiroTHIQs) via the Castagnoli-Cushman reaction von Safrygin, Alexander, Dar'in, Dmitry, Bakulina, Olga, Krasavin, Mikhail

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Discovery of 2‑[1-(4,4-Difluorocyclohexyl)piperidin-4-yl]-6-fluoro-3-oxo-2,3-dihydro‑1H‑isoindole-4-carboxamide (NMS-P118): A Potent, Orally Available, and Highly Selective PARP‑1... von Papeo, Gianluca, Posteri, Helena, Borghi, Daniela, Busel, Alina A., Caprera, Francesco, Casale, Elena, Ciomei, Marina, Cirla, Alessandra, Corti, Emiliana, D’Anello, Matteo, Fasolini, Marina, Forte, Barbara, Galvani, Arturo, Isacchi, Antonella, Khvat, Alexander, Krasavin, Mikhail Y., Lupi, Rosita, Orsini, Paolo, Perego, Rita, Pesenti, Enrico, Pezzetta, Daniele, Rainoldi, Sonia, Riccardi-Sirtori, Federico, Scolaro, Alessandra, Sola, Francesco, Zuccotto, Fabio, Felder, Eduard R., Donati, Daniele, Montagnoli, Alessia

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Preparation and Synthetic Applications of Five-to-Seven-Membered Cyclic α-Diazo Monocarbonyl Compounds von Zhukovsky, Daniil, Dar'in, Dmitry, Bakulina, Olga, Krasavin, Mikhail

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Carbonic Anhydrase IX Inhibitors as Candidates for Combination Therapy of Solid Tumors von Kalinin, Stanislav, Malkova, Anna, Sharonova, Tatiana, Sharoyko, Vladimir, Bunev, Alexander, Supuran, Claudiu T., Krasavin, Mikhail

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A novel approach to biologically relevant oxazolo[5,4-d]pyrimidine-5,7-diones via readily available diazobarbituric acid derivatives von Gecht, Martha, Kantin, Grigory, Dar'in, Dmitry, Krasavin, Mikhail

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The Use of Aryl-Substituted Homophthalic Anhydrides in the Castagnoli-Cushman Reaction Provides Access to Novel Tetrahydroisoquinolone Carboxylic Acid Bearing an All-Carbon Quatern... von Moshnenko, Nazar, Kazantsev, Alexander, Bakulina, Olga, Dar'in, Dmitry, Krasavin, Mikhail

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One-Pot Sequence of Staudinger/aza-Wittig/Castagnoli-Cushman Reactions Provides Facile Access to Novel Natural-like Polycyclic Ring Systems von Lebedev, Rodion, Dar'in, Dmitry, Kantin, Grigory, Bakulina, Olga, Krasavin, Mikhail

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Extending the Scope of the New Variant of the Castagnoli–Cushman Cyclocondensation onto o-Methyl Benzoic Acids Bearing Various Electron-Withdrawing Groups in the α-Position von Guranova, Natalia, Yakovleva, Lyudmila, Bakulina, Olga, Dar’in, Dmitry, Krasavin, Mikhail

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Inhibitory activity against carbonic anhydrase IX and XII as a candidate selection criterion in the development of new anticancer agents von Krasavin, Mikhail, Kalinin, Stanislav, Sharonova, Tatiana, Supuran, Claudiu T.

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Synthesis and Antibacterial Evaluation of Ciprofloxacin Congeners with Spirocyclic Amine Periphery von Lukin, Alexei, Komarova, Kristina, Vinogradova, Lyubov, Rogacheva, Elizaveta, Kraeva, Lyudmila, Krasavin, Mikhail

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Dicarboxylic Acid Monoesters in β- and δ-Lactam Synthesis von Ananeva, Anna, Bakulina, Olga, Dar'in, Dmitry, Kantin, Grigory, Krasavin, Mikhail

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Facile and diastereoselective arylation of the privileged 1,4-dihydroisoquinolin-3(2 H )-one scaffold von Dar'in, Dmitry, Kantin, Grigory, Bunev, Alexander, Krasavin, Mikhail

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Two Annulated Azaheterocyclic Cores Readily Available from a Single Tetrahydroisoquinolonic Castagnoli-Cushman Precursor von Karchuganova, Elizaveta, Bakulina, Olga, Dar'in, Dmitry, Krasavin, Mikhail

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