Discovery of potent furan piperazine sodium channel blockers for treatment of neuropathic pain von Drizin, Irene, Gregg, Robert J., Scanio, Marc J.C., Shi, Lei, Gross, Michael F., Atkinson, Robert N., Thomas, James B., Johnson, Matthew S., Carroll, William A., Marron, Brian E., Chapman, Mark L., Liu, Dong, Krambis, Michael J., Shieh, Char-Chang, Zhang, XuFeng, Hernandez, Gricelda, Gauvin, Donna M., Mikusa, Joseph P., Zhu, Chang Z., Joshi, Shailen, Honore, Prisca, Marsh, Kennan C., Roeloffs, Rosemarie, Werness, Stephen, Krafte, Douglas S., Jarvis, Michael F., Faltynek, Connie R., Kort, Michael E.

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Discovery and biological evaluation of potent, selective, orally bioavailable, pyrazine-based blockers of the Na sub(v)1.8 sodium channel with efficacy in a model of neuropathic pa... von Scanio, MJ, Shi, L, Drizin, I, Gregg, R J, Atkinson, R N, Thomas, J B, Johnson, MS, Chapman, M L, Liu, D, Krambis, MJ, Liu, Y, Shieh, C C, Zhang, X, Simler, G H, Joshi, S, Honore, P, Marsh, K C, Knox, A, Werness, S, Antonio, B, Krafte, D S, Jarvis, M F, Faltynek, C R, Marron, B E, Kort, ME

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