Sodium channels and nociception: recent concepts and therapeutic opportunities von Krafte, Douglas S, Bannon, Anthony W

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Discovery and Biological Evaluation of 5-Aryl-2-furfuramides, Potent and Selective Blockers of the Nav1.8 Sodium Channel with Efficacy in Models of Neuropathic and Inflammatory Pai... von Kort, Michael E, Drizin, Irene, Gregg, Robert J, Scanio, Marc J. C, Shi, Lei, Gross, Michael F, Atkinson, Robert N, Johnson, Matthew S, Pacofsky, Gregory J, Thomas, James B, Carroll, William A, Krambis, Michael J, Liu, Dong, Shieh, Char-Chang, Zhang, XuFeng, Hernandez, Gricelda, Mikusa, Joseph P, Zhong, Chengmin, Joshi, Shailen, Honore, Prisca, Roeloffs, Rosemarie, Marsh, Kennan C, Murray, Bernard P, Liu, Jinrong, Werness, Stephen, Faltynek, Connie R, Krafte, Douglas S, Jarvis, Michael F, Chapman, Mark L, Marron, Brian E

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The Effect of κ-Opioid Receptor Agonists on Tetrodotoxin-Resistant Sodium Channels in Primary Sensory Neurons von Su, Xin, Castle, Neil A., Antonio, Brett, Roeloffs, Rosemarie, Thomas, James B., Krafte, Douglas S., Chapman, Mark L.

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Pharmacological modulation of human cardiac Na + channels von Krafte, Douglas S., Davison, Kathleen, Dugrenier, Nancy, Estep, Kimberly, Josef, Kurt, Barchi, Robert L., Kallen, Roland G., Silver, Paul J., Ezrin, Alan M.

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Discovery of potent furan piperazine sodium channel blockers for treatment of neuropathic pain von Drizin, Irene, Gregg, Robert J., Scanio, Marc J.C., Shi, Lei, Gross, Michael F., Atkinson, Robert N., Thomas, James B., Johnson, Matthew S., Carroll, William A., Marron, Brian E., Chapman, Mark L., Liu, Dong, Krambis, Michael J., Shieh, Char-Chang, Zhang, XuFeng, Hernandez, Gricelda, Gauvin, Donna M., Mikusa, Joseph P., Zhu, Chang Z., Joshi, Shailen, Honore, Prisca, Marsh, Kennan C., Roeloffs, Rosemarie, Werness, Stephen, Krafte, Douglas S., Jarvis, Michael F., Faltynek, Connie R., Kort, Michael E.

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Direct Activation of an Inwardly Rectifying Potassium Channel by Arachidonic Acid von Liu, Y, Liu, D, Heath, L, Meyers, D M, Krafte, D S, Wagoner, P K, Silvia, C P, Yu, W, Curran, M E

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Tenidap, a novel anti-inflammatory agent, is an opener of the inwardly rectifying K + channel hKir2.3 von Liu, Yi, Liu, Dong, Printzenhoff, David, Coghlan, Michael J., Harris, Richard, Krafte, Douglas S.

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A rat brain na + channel α subunit with novel gating properties von Auld, Vanessa J., Goldin, Alan L., Krafte, Douglas S., Marshall, John, Dunn, James M., Catterall, William A., Lester, Henry A., Davidson, Norman, Dunn, Robert J.

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Decrease of inward rectification as a mechanism for arachidonic acid-induced potentiation of hKir2.3 von Liu, Yi, Liu, Dong, Krafte, Douglas S

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Identification of Three Separate Binding Sites on SHK Toxin, a Potent Inhibitor of Voltage-Dependent Potassium Channels in Human T-Lymphocytes and Rat Brain von Pennington, M.W., Mahnir, V.M., Krafte, D.S., Zaydenberg, I., Byrnes, M.E., Khaytin, I., Crowley, K., Kem, W.R.

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A Neutral Amino Acid Change in Segment IIS4 Dramatically Alters the Gating Properties of the Voltage-Dependent Sodium Channel von Auld, V. J., Goldin, A. L., Krafte, D. S., Catterall, W. A., Lester, H. A., Davidson, N., Dunn, R. J.

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Block of Nav1.8 by Small Molecules von Krafte, Douglas S., Chapman, Mark, Marron, Brian, Atkinson, Robert, Liu, Yi, Yu, Fei, Kort, Michael, Jarvis, Michael F.

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Synthesis and Structure-Activity Relationships of 6-Heterocyclic-Substituted Purines as Inactivation Modifiers of Cardiac Sodium Channels von Estep, Kimberly G, Josef, Kurt A, Bacon, Edward R, Carabateas, Philip M, Rumney, Squire, Pilling, Garry M, Krafte, Douglas S, Volberg, Walter A, Dillon, Kathleen, Dugrenier, Nancy, Briggs, G. Maurice, Canniff, Paul C, Gorczyca, William P, Stankus, Gerald P, Ezrin, Alan M

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Voltage-dependent modulation of Ca channel current in heart cells by Bay K8644 von SANGUINETTI, M. C, KRAFTE, D. S, KASS, R. S

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Hydrogen ion modulation of Ca channel current in cardiac ventricular cells. Evidence for multiple mechanisms von Krafte, D S, Kass, R S

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Novel Inhibitors of Potassium Ion Channels on Human T Lymphocytes von Michne, William F, Guiles, Joseph W, Treasurywala, Adi M, Castonguay, Laurie A, Weigelt, Carolyn A, Oconnor, Bernard, Volberg, Walter A, Grant, Alison M, Chadwick, Christopher C, Krafte, Douglas S, Hill, Roger J

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Inactivation of cloned Na channels expressed in Xenopus oocytes von KRAFTE, D. S, GOLDIN, A. L, AULD, V. J, DUNN, R. J, DAVIDSON, N, LESTER, H. A

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WIN 17317-3: novel nonpeptide antagonist of voltage-activated K+ channels in human T lymphocytes von Hill, R J, Grant, A M, Volberg, W, Rapp, L, Faltynek, C, Miller, D, Pagani, K, Baizman, E, Wang, S, Guiles, J W

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Voltage Dependence of Cardiac Delayed Rectifier Block by Methanesulfonamide Class III Antiarrhythmic Agents von Krafte, Douglas S, Volberg, Walter A

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Identification of a Specific Radioligand for the Cardiac Rapidly Activating Delayed Rectifier K+ Channel von Chadwick, Christopher C, Ezrin, Alan M, OʼConnor, Bernard, Volberg, Walter A, Smith, David I, Wedge, Karen J, Hill, Roger J, Briggs, G Maurice, Pagani, Edward D, Silver, Paul J, Krafte, Douglas S

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