A Clinical-Stage Cysteine Protease Inhibitor blocks SARS-CoV‑2 Infection of Human and Monkey Cells von Mellott, Drake M, Tseng, Chien-Te, Drelich, Aleksandra, Fajtová, Pavla, Chenna, Bala C, Kostomiris, Demetrios H, Hsu, Jason, Zhu, Jiyun, Taylor, Zane W, Kocurek, Klaudia I, Tat, Vivian, Katzfuss, Ardala, Li, Linfeng, Giardini, Miriam A, Skinner, Danielle, Hirata, Ken, Yoon, Michael C, Beck, Sungjun, Carlin, Aaron F, Clark, Alex E, Beretta, Laura, Maneval, Daniel, Hook, Vivian, Frueh, Felix, Hurst, Brett L, Wang, Hong, Raushel, Frank M, O’Donoghue, Anthony J, de Siqueira-Neto, Jair Lage, Meek, Thomas D, McKerrow, James H

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Dissecting the Kinetic Mechanism of Human Lysine Methyltransferase 2D and Its Interactions with the WRAD2 Complex von Edwardes, Lucy V., Caswell, Sarah J., Giurrandino, Mariacarmela, Zhai, Xiang, Gohlke, Andrea, Kostomiris, Demetrios H., Pollard, Hannah K., Pflug, Alexander, Hamm, Gregory R., Jervis, Kate V., Clarkson, Paul N., Syson, Karl

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Optimization of Potent, Efficacious, Selective and Blood–Brain Barrier Penetrating Inhibitors Targeting EGFR Exon20 Insertion Mutations von Thomson, Clare, Braybrooke, Erin, Colclough, Nicola, Davies, Nichola L., Floc’h, Nicolas, Greenwood, Ryan, Guérot, Carine, Hargreaves, David, Johnstrom, Peter, Khurana, Puneet, Kostomiris, Demetrios H., Li, Songlei, Lister, Andrew, Lorthioir, Olivier, Martin, Scott, McCoull, William, McLean, Neville J., McWilliams, Lisa, Orme, Jonathan P., Packer, Martin J., Pearson, Stuart, Swaih, Aisha M., Tentarelli, Sharon, Tucker, Michael J., Ward, Richard A., Wilkinson, Stephen, Winlow, Poppy, Wood, Isabel L.

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