A Whole Proteome Inventory of Background Photocrosslinker Binding von Kleiner, Philipp, Heydenreuter, Wolfgang, Stahl, Matthias, Korotkov, Vadim S., Sieber, Stephan A.

Volltext

Chemical Cross-Linking Enables Drafting ClpXP Proximity Maps and Taking Snapshots of In Situ Interaction Networks von Fux, Anja, Korotkov, Vadim S., Schneider, Markus, Antes, Iris, Sieber, Stephan A.

Volltext

Repurposing human kinase inhibitors to create an antibiotic active against drug-resistant Staphylococcus aureus, persisters and biofilms von Le, Philipp, Kunold, Elena, Macsics, Robert, Rox, Katharina, Jennings, Megan C., Ugur, Ilke, Reinecke, Maria, Chaves-Moreno, Diego, Hackl, Mathias W., Fetzer, Christian, Mandl, Franziska A. M., Lehmann, Johannes, Korotkov, Vadim S., Hacker, Stephan M., Kuster, Bernhard, Antes, Iris, Pieper, Dietmar H., Rohde, Manfred, Wuest, William M., Medina, Eva, Sieber, Stephan A.

Volltext

Hydantoin analogs inhibit the fully assembled ClpXP protease without affecting the individual peptidase and chaperone domains von Fetzer, Christian, Korotkov, Vadim S, Sieber, Stephan A

Volltext

Selective Activation of Human Caseinolytic Protease P (ClpP) von Stahl, Matthias, Korotkov, Vadim S., Balogh, Dóra, Kick, Leonhard M., Gersch, Malte, Pahl, Axel, Kielkowski, Pavel, Richter, Klaus, Schneider, Sabine, Sieber, Stephan A.

Volltext

Design and synthesis of tailored human caseinolytic protease P inhibitors von Gronauer, Thomas F, Mandl, Melanie M, Lakemeyer, Markus, Hackl, Mathias W, Meßner, Martina, Korotkov, Vadim S, Pachmayr, Johanna, Sieber, Stephan A

Volltext

Oligosubstituted Pyrroles Directly from Substituted Methyl Isocyanides and Acetylenes von Lygin, Alexander V., Larionov, Oleg V., Korotkov, Vadim S., de Meijere, Armin

Volltext

A chemical compound inhibiting the Aha1–Hsp90 chaperone complex von Stiegler, Sandrine C., Rübbelke, Martin, Korotkov, Vadim S., Weiwad, Matthias, John, Christine, Fischer, Gunter, Sieber, Stephan A., Sattler, Michael, Buchner, Johannes

Volltext

A Chemical Disruptor of the ClpX Chaperone Complex Attenuates the Virulence of Multidrug‐Resistant Staphylococcus aureus von Fetzer, Christian, Korotkov, Vadim S., Thänert, Robert, Lee, Kyu Myung, Neuenschwander, Martin, von Kries, Jens Peter, Medina, Eva, Sieber, Stephan A.

Volltext

The Mechanism of Caseinolytic Protease (ClpP) Inhibition von Gersch, Malte, Gut, Felix, Korotkov, Vadim S., Lehmann, Johannes, Böttcher, Thomas, Rusch, Marion, Hedberg, Christian, Waldmann, Herbert, Klebe, Gerhard, Sieber, Stephan A.

Volltext

Dual Inhibitor of Staphylococcus aureus Virulence and Biofilm Attenuates Expression of Major Toxins and Adhesins von Hofbauer, Barbara, Vomacka, Jan, Stahl, Matthias, Korotkov, Vadim S, Jennings, Megan C, Wuest, William M, Sieber, Stephan A

Volltext

Reversible Inhibitors Arrest ClpP in a Defined Conformational State that Can Be Revoked by ClpX Association von Pahl, Axel, Lakemeyer, Markus, Vielberg, Marie-Theres, Hackl, Mathias W., Vomacka, Jan, Korotkov, Vadim S., Stein, Martin L., Fetzer, Christian, Lorenz-Baath, Katrin, Richter, Klaus, Waldmann, Herbert, Groll, Michael, Sieber, Stephan A.

Volltext

A Minimal β-Lactone Fragment for Selective β5c or β5i Proteasome Inhibitors von Groll, Michael, Korotkov, Vadim S., Huber, Eva M., de Meijere, Armin, Ludwig, Antje

Volltext

A Minimal [beta]-Lactone Fragment for Selective [beta]5c or [beta]5i Proteasome Inhibitors von Groll, Michael, Korotkov, Vadim S, Huber, Eva M, deMeijere, Armin, Ludwig, Antje

Volltext

Development and characterization of improved β-lactone-based anti-virulence drugs targeting ClpP von Zeiler, Evelyn, Korotkov, Vadim S., Lorenz-Baath, Katrin, Böttcher, Thomas, Sieber, Stephan A.

Volltext

GaCl3-catalyzed insertion of diazene derivatives into the cyclopropane ring von KOROTKOV, Vadim S, LARIONOV, Oleg V, HOFMEISTER, Anja, MAGULL, Jorg, DE MEIJERE, Armin

Volltext

A β-Lactone-Based Antivirulence Drug Ameliorates Staphylococcus aureus Skin Infections in Mice von Weinandy, Franziska, Lorenz-Baath, Katrin, Korotkov, Vadim S., Böttcher, Thomas, Sethi, Shneh, Chakraborty, Trinad, Sieber, Stephan A.

Volltext

An Aromatic Hydroxyamide Attenuates Multiresistant Staphylococcus aureus Toxin Expression von Vomacka, Jan, Korotkov, Vadim S., Bauer, Bianca, Weinandy, Franziska, Kunzmann, Martin H., Krysiak, Joanna, Baron, Oliver, Böttcher, Thomas, Lorenz-Baath, Katrin, Sieber, Stephan A.

Volltext

Synthesis and biological activity of optimized belactosin C congeners von Korotkov, Vadim S, Ludwig, Antje, Larionov, Oleg V, Lygin, Alexander V, Groll, Michael, de Meijere, Armin

Volltext

Neocarzilin A Is a Potent Inhibitor of Cancer Cell Motility Targeting VAT‑1 Controlled Pathways von Gleissner, Carolin M.-L, Pyka, Carolin L, Heydenreuter, Wolfgang, Gronauer, Thomas F, Atzberger, Carina, Korotkov, Vadim S, Cheng, Weiting, Hacker, Stephan M, Vollmar, Angelika M, Braig, Simone, Sieber, Stephan A

Volltext