Synthesis and SAR of novel 2-arylthiazolidinones as selective analgesic N-type calcium channel blockers von Knutsen, Lars J.S., Hobbs, Christopher J., Earnshaw, Christopher G., Fiumana, Andrea, Gilbert, Jenny, Mellor, Sarah L., Radford, Fleur, Smith, Nichola J., Birch, Philip J., Russell Burley, J., Ward, Stuart D.C., James, Iain F.

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N-substituted adenosines as novel neuroprotective A(1) agonists with diminished hypotensive effects von Knutsen, L J, Lau, J, Petersen, H, Thomsen, C, Weis, J U, Shalmi, M, Judge, M E, Hansen, A J, Sheardown, M J

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Synthesis of Novel GABA Uptake Inhibitors. 3. Diaryloxime and Diarylvinyl Ether Derivatives of Nipecotic Acid and Guvacine as Anticonvulsant Agents von Knutsen, Lars J. S, Andersen, Knud Erik, Lau, Jesper, Lundt, Behrend F, Henry, Rodger F, Morton, Howard E, Nærum, Lars, Petersen, Hans, Stephensen, Henrik, Suzdak, Peter D, Swedberg, Michael D. B, Thomsen, Christian, Sørensen, Per O

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Synthesis of Novel GABA Uptake Inhibitors. 4. Bioisosteric Transformation and Successive Optimization of Known GABA Uptake Inhibitors Leading to a Series of Potent Anticonvulsant D... von Andersen, Knud Erik, Sørensen, Jan L, Huusfeldt, Per O, Knutsen, Lars J. S, Lau, Jesper, Lundt, Behrend F, Petersen, Hans, Suzdak, Peter D, Swedberg, Michael D. B

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Characterization of tiagabine (NO-328), a new potent and selective GABA uptake inhibitor von Nielsen, Erik B., Suzdak, Peter D., Andersen, Knud E., Knutsen, Lars J.S., Sonnewald, Ursula, Braestrup, Claus

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The synthesis of novel GABA uptake inhibitors. 1. Elucidation of the structure-activity studies leading to the choice of (R)-1-[4,4-bis(3-methyl-2-thienyl)-3-butenyl]-3-piperidinec... von Andersen, Knud Erik, Braestrup, Claus, Groenwald, Frederik C, Joergensen, Anker S, Nielsen, Erik B, Sonnewald, Ursula, Soerensen, Per O, Suzdak, Peter D, Knutsen, Lars J. S

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NNC-711, a novel potent and selective γ-aminobutyric acid uptake inhibitor: pharmacological characterization von Suzdak, Peter D., Frederiksen, Kristen, Andersen, Knud Erik, Sørensen, Per O., Knutsen, Lars J.S., Nielsen, Erik B.

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(R)‐N‐[4,4‐Bis(3‐Methyl‐2‐Thienyl)but‐3‐en‐1‐yl]Nipecotic Acid Binds with High Affinity to the Brain γ‐Aminobutyric Acid Uptake Carrier von Braestrup, Claus, Nielsen, Erik B., Sonnewald, Ursula, Knutsen, Lars J. S., Andersen, Knud Erik, Jansen, Jens Aas, Frederiksen, Kristen, Andersen, Peter H., Mortensen, Alicja, Suzdak, Peter D.

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N-Substituted Adenosines as Novel Neuroprotective A sub(1) Agonists with Diminished Hypotensive Effects von Knutsen, LJS, Lau, J, Petersen, H, Thomsen, C, Weis, JU, Shalmi, M, Judge, ME, Hansen, A J, Sheardown, MJ

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Stereoselective conversion of 2′,3′-dideoxydidehydro carbocyclic nucleosides into 2′-deoxy carbocyclic nucleosides von Barkley, James V., Dhanda, Anupma, Nielsen, May-Britt, Roberts, Stanley M., Knutsen, Lars J. S., Varley, David R.

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super(14)C-labelling of a novel antiischaemic adenosine A sub(1) agonist at purine C-8 von Valsborg, J S, Knutsen, LJS, Foged, C

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In vivo labeling of the central GABA uptake carrier with super(3)H-tiagabine von Suzdak, P D, Swedberg, MDB, Andersen, KE, Knutsen, LJS, Braestrup, C

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Facile conversion of 4-endo-hydroxy-2-oxabicyclo[3.3.0]oct-7-en-3-one into carbocyclic 2′-deoxyribonucleoside analogues von Dhanda, Anupma, Knutsen, Lars J. S., Nielsen, May-Britt, Roberts, Stanley M., Varley, David R.

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(R)-N-(4,4-Bis(3-methyl-2-thienyl)but-3-en-1-yl)nipecotic acid binds with high affinity to the brain gamma -aminobutyric acid uptake carrier von Braestrup, C, Nielsen, E B, Sonnewald, U, Knutsen, LJS, Andersen, KE, Jansen, JA, Frederiksen, K, Andersen, PH, Mortensen, A, Suzdak, P D

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Synthesis and antiviral properties of 5-(2-substituted vinyl)-6-aza-2'-deoxyuridines von Mitchell, William L, Ravenscroft, Paul, Hill, Malcolm L, Knutsen, Lars J. S, Judkins, Brian D, Newton, Roger F, Scopes, David I. C

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The Chemistry of 2′-Deoxyribo-C-Nucleosides von Knutsen, Lars J. S.

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Coupling-elimination reactions of 2,5-anhydro-3,4,6-tri- O-benzoyl- d-allonic acid: synthesis of 2′-deoxyribo- C-nucleosides von Knutsen, Lars J.S., Newton, Roger F., Scopes, David I.C., Klinkert, Graham

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Synthesis of imidazo-fused bridgehead-nitrogen 2'-deoxyribo-C-nucleosides: coupling-elimination reactions of 2,5-anhydro-3,4,6-tri-O-benzoyl-D-allonic acid von KNUTSEN, L. J. S, JUDKINS, B. D, NEWTON, R. F, SCOPES, D. I. C, KLINKERT, G

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Synthesis of imidazo-fused bridgehead-nitrogen C-nucleosides via dehydrative coupling reactions of 2,5-anhydro-3,4,6-tri-O-benzoyl-D-allonic acid von KNUTSEN, L. J. S, JUDKINS, B. D, MITCHELL, W. L, NEWTON, R. F, SCOPES, D. I. C

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Reduction of the carboxyl-function in aromatic carboxylic acids by alkali metal–liquid ammonia solutions von Franks, David, Grossel, Martin C., Hayward, Rodney C., Knutsen, Lars J. S.

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