Synthesis of Novel GABA Uptake Inhibitors. 3. Diaryloxime and Diarylvinyl Ether Derivatives of Nipecotic Acid and Guvacine as Anticonvulsant Agents von Knutsen, Lars J. S, Andersen, Knud Erik, Lau, Jesper, Lundt, Behrend F, Henry, Rodger F, Morton, Howard E, Nærum, Lars, Petersen, Hans, Stephensen, Henrik, Suzdak, Peter D, Swedberg, Michael D. B, Thomsen, Christian, Sørensen, Per O

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Synthesis of Novel GABA Uptake Inhibitors. 4. Bioisosteric Transformation and Successive Optimization of Known GABA Uptake Inhibitors Leading to a Series of Potent Anticonvulsant D... von Andersen, Knud Erik, Sørensen, Jan L, Huusfeldt, Per O, Knutsen, Lars J. S, Lau, Jesper, Lundt, Behrend F, Petersen, Hans, Suzdak, Peter D, Swedberg, Michael D. B

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Characterization of tiagabine (NO-328), a new potent and selective GABA uptake inhibitor von Nielsen, Erik B., Suzdak, Peter D., Andersen, Knud E., Knutsen, Lars J.S., Sonnewald, Ursula, Braestrup, Claus

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NNC-711, a novel potent and selective γ-aminobutyric acid uptake inhibitor: pharmacological characterization von Suzdak, Peter D., Frederiksen, Kristen, Andersen, Knud Erik, Sørensen, Per O., Knutsen, Lars J.S., Nielsen, Erik B.

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The synthesis of new adenosine A3 selective ligands containing bioisosteric isoxazoles von MOGENSEN, J. P, ROBERTS, S. M, BOWLER, A. N, THOMSEN, C, KNUTSEN, L. J. S

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Contrasting effects of adenosine A1 and A2 receptor ligands in different chemoconvulsive rodent models von KLITGAARD, H, KNUTSEN, L. J. S, THOMSEN, C

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N-Substituted Adenosines as Novel Neuroprotective A1 Agonists with Diminished Hypotensive Effects von Knutsen, Lars J. S, Lau, Jesper, Petersen, Hans, Thomsen, Christian, Weis, Jan U, Shalmi, Michael, Judge, Martin E, Hansen, Anker Jon, Sheardown, Malcolm J

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N-substituted adenosines as novel neuroprotective A(1) agonists with diminished hypotensive effects von Knutsen, L J, Lau, J, Petersen, H, Thomsen, C, Weis, J U, Shalmi, M, Judge, M E, Hansen, A J, Sheardown, M J

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The synthesis of novel GABA uptake inhibitors. 1. Elucidation of the structure-activity studies leading to the choice of (R)-1-[4,4-bis(3-methyl-2-thienyl)-3-butenyl]-3-piperidinec... von Andersen, Knud Erik, Braestrup, Claus, Groenwald, Frederik C, Joergensen, Anker S, Nielsen, Erik B, Sonnewald, Ursula, Soerensen, Per O, Suzdak, Peter D, Knutsen, Lars J. S

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(R)‐N‐[4,4‐Bis(3‐Methyl‐2‐Thienyl)but‐3‐en‐1‐yl]Nipecotic Acid Binds with High Affinity to the Brain γ‐Aminobutyric Acid Uptake Carrier von Braestrup, Claus, Nielsen, Erik B., Sonnewald, Ursula, Knutsen, Lars J. S., Andersen, Knud Erik, Jansen, Jens Aas, Frederiksen, Kristen, Andersen, Peter H., Mortensen, Alicja, Suzdak, Peter D.

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In vivo labeling of the central GABA uptake carrier with 3H-tiagabine von SUZDAK, P. D, SWEDBERG, M. D. B, ANDERSEN, K. E, KNUTSEN, L. J. S, BRAESTRUP, C

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Unexpected neuroprotection observed with the adenosine A2A receptor agonist CGS 21680 von Sheardown, Malcolm J., Knutsen, Lars J.S.

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Adenosine A1 and A3 selective N-alkoxypurines as novel cytokine modulators and neuroprotectants von Knutsen, Lars J.S., Sheardown, Malcolm J., Roberts, Stanley M., Mogensen, John P., Olsen, Uffe Bang, Thomsen, Christian, Bowler, Andrew N.

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The synthesis and biochemical evaluation of new A1 selective adenosine receptor agonists containing 6-hydrazinopurine moieties von KNUTSEN, L. J. S, LAU, J, SHEARDOWN, M. J, THOMSEN, C

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14C-labelling of a novel antiischaemic adenosine A1 agonist at purine C-8 von Valsborg, Jacob S., Knutsen, Lars J. S., Foged, Christian

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Synthesis and antiviral properties of 5-(2-substituted vinyl)-6-aza-2'-deoxyuridines von Mitchell, William L, Ravenscroft, Paul, Hill, Malcolm L, Knutsen, Lars J. S, Judkins, Brian D, Newton, Roger F, Scopes, David I. C

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Synthesis of [8-14C]-2,6-dichloro-9H-purine, a radiolabelled precursor for 14C-nucleosides von Valsborg, Jacob S., Knutsen, Lars J. S., Lundt, Inge, Foged, Christian

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The synthesis of novel GABA uptake inhibitors. I: Elucidation of the structure-activity studies leading to the choice of (R)-1-[4,4-bis(3-methyl-2-thienyl)-3-butenyl]-3-piperidinec... von ANDERSEN, K. E, BRAESTRUP, C, GRØNWALD, F. C, JØRGENSEN, A. S, NIELSEN, E. B, SONNEWALD, U, SØRENSEN, P. O, SUZDAK, P. D, KNUTSEN, L. J. S

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The Chemistry of 2′-Deoxyribo-C-Nucleosides von Knutsen, Lars J. S.

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(R)-N-[4,4-bis(3-methyl-2-thienyl)but-3-en-1-yl]nipecotic acids binds with high affinity to the brain γ-aminobutyric acid uptake carrier von BRAESTRUP, C, NIELSEN, E. B, SONNEWALD, U, KNUTSEN, L. J. S, ANDERSEN, K. E, JANSEN, J. A, FREDERIKSEN, K, ANDERSEN, P. H, MORTENSEN, A, SUZDAK, P. D

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