Virtual and biomolecular screening converge on a selective agonist for GPR30 von Oprea, Tudor I, Prossnitz, Eric R, Bologa, Cristian G, Revankar, Chetana M, Young, Susan M, Edwards, Bruce S, Arterburn, Jeffrey B, Kiselyov, Alexander S, Parker, Matthew A, Tkachenko, Sergey E, Savchuck, Nikolay P, Sklar, Larry A

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Chemistry of N-fluoropyridinium salts von Kiselyov, Alexander S

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Novel inhibitors of VEGF receptors-1 and -2 based on azole-5-carboxamide templates von Kiselyov, Alexander S., Milligan, Daniel, Ouyang, Xiaohu

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Arylphthalazines. Part 2: 1-(Isoquinolin-5-yl)-4-arylamino phthalazines as potent inhibitors of VEGF receptors I and II von Duncton, Matthew A.J., Piatnitski, Evgueni L., Katoch-Rouse, Reeti, Smith, Leon M., Kiselyov, Alexander S., Milligan, Daniel L., Balagtas, Chris, Wong, Wai C., Kawakami, Joel, Doody, Jacqueline F.

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Quantitative 3D reconstruction of viral vector distribution in rodent and ovine brain following local delivery von Poceviciute, Roberta, Mitchell, Kenneth, Nikolakopoulou, Angeliki Maria, Cho, Suehyun K., Ma, Xiaobo, Chen, Phillip, Figueroa, Samantha, Sarmiento, Ethan J., Singh, Aryan, Hartstein, Oren, Loudon, William G., Cros, Florent, Kiselyov, Alexander S.

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3,4-Disubstituted isothiazoles: Novel potent inhibitors of VEGF receptors 1 and 2 von Kiselyov, Alexander S., Semenova, Marina, Semenov, Victor V.

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One-pot synthesis of polysubstituted pyrimidines von Kiselyov, Alexander S.

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(1,2,3-Triazol-4-yl)benzenamines: Synthesis and activity against VEGF receptors 1 and 2 von Kiselyov, Alexander S., Semenova, Marina, Semenov, Victor V.

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DNA triple-helix specific intercalators as antigene enhancers: Unfused aromatic cations von Wilson, W. David, Tanious, Farial A, Mizan, Shaikh, Yao, Shijie, Kiselyov, Alexander S, Zon, Gerald, Strekowski, Lucjan

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Oxadiazole derivatives as a novel class of antimitotic agents: Synthesis, inhibition of tubulin polymerization, and activity in tumor cell lines von Ouyang, Xiaohu, Piatnitski, Evgueni L., Pattaropong, Vatee, Chen, Xiaoling, He, Hai-Ying, Kiselyov, Alexander S., Velankar, Avdhoot, Kawakami, Joel, Labelle, Marc, Smith, Leon, Lohman, Julia, Lee, Sui Ping, Malikzay, Asra, Fleming, James, Gerlak, Jason, Wang, Ying, Rosler, Robin L., Zhou, Kai, Mitelman, Stan, Camara, Margarita, Surguladze, David, Doody, Jacqueline F., Tuma, M. Carolina

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Arylphthalazines as potent, and orally bioavailable inhibitors of VEGFR-2 von Duncton, Matthew A.J., Piatnitski Chekler, Eugene L., Katoch-Rouse, Reeti, Sherman, Dan, Wong, Wai C., Smith, Leon M., Kawakami, Joel K., Kiselyov, Alexander S., Milligan, Daniel L., Balagtas, Chris, Hadari, Yaron R., Wang, Ying, Patel, Sheetal N., Rolster, Robin L., Tonra, James R., Surguladze, David, Mitelman, Stan, Kussie, Paul, Bohlen, Peter, Doody, Jacqueline F.

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The o-Amino-Trifluoromethyl Functionality as a Novel Synthon for 4-Fluoroquinolines von Strekowski, Lucjan, Kiselyov, Alexander S, Hojjat, Maryam

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Discovery of Dual VEGFR-2 and Tubulin Inhibitors with in Vivo Efficacy von Chekler, Eugene L. Piatnitski, Kiselyov, Alexander S, Ouyang, Xiaohu, Chen, Xiaoling, Pattaropong, Vatee, Wang, Ying, Tuma, M. Carolina, Doody, Jacqueline F

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1-[4-(1 H-Benzoimidazol-2-yl)-phenyl]-3-[4-(1 H-benzoimidazol-2-yl)-phenyl]-urea derivatives as small molecule heparanase inhibitors von Pan, Weitao, Miao, Hua-Quan, Xu, Yong-Jiang, Navarro, Elizabeth C., Tonra, James R., Corcoran, Erik, Lahiji, Armin, Kussie, Paul, Kiselyov, Alexander S., Wong, Wai C., Liu, Hu

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Hetaryl imidazoles: A novel dual inhibitors of VEGF receptors I and II von Kiselyov, Alexander S., Semenova, Marina, Semenov, Victor V.

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Synthesis and structure–activity relationships of 1,2,4-triazoles as a novel class of potent tubulin polymerization inhibitors von Ouyang, Xiaohu, Chen, Xiaoling, Piatnitski, Evgueni L., Kiselyov, Alexander S., He, Hai-Ying, Mao, Yunyu, Pattaropong, Vatee, Yu, Yang, Kim, Ki H., Kincaid, John, Smith, Leon, Wong, Wai C., Lee, Sui Ping, Milligan, Daniel L., Malikzay, Asra, Fleming, James, Gerlak, Jason, Deevi, Dhanvanthri, Doody, Jacqueline F., Chiang, Hui-Hsien, Patel, Sheetal N., Wang, Ying, Rolser, Robin L., Kussie, Paul, Labelle, Marc, Tuma, M. Carolina

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Arylphthalazines: Identification of a new phthalazine chemotype as inhibitors of VEGFR kinase von Piatnitski, Evgueni L., Duncton, Matthew A.J., Kiselyov, Alexander S., Katoch-Rouse, Reeti, Sherman, Dan, Milligan, Daniel L., Balagtas, Chris, Wong, Wai C., Kawakami, Joel, Doody, Jacqueline F.

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Design and chemical synthesis of [1,2,4]triazol[1,5- c]pyrimidin-5-yl amines, a novel class of VEGFR-2 kinase inhibitors von Kiselyov, Alexander S., Piatnitski Chekler, Eugene L., Chernisheva, Natalia B., Salamandra, Lev K., Semenov, Victor V.

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Efficient Syntheses of the anti- and syn-Diol Epoxide Metabolites of the Carcinogenic Polycyclic Aromatic Hydrocarbon Benzo[g]chrysene von Kiselyov, Alexander S, Lee, Hongmee, Harvey, Ronald G

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4-(Azolylphenyl)-phthalazin-1-amines: Novel Inhibitors of VEGF Receptors I and II von Kiselyov, Alexander S., Semenov, Victor V., Milligan, Daniel

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