Anticancer and Structure Activity Relationship of Non-Symmetrical Choline Kinase Inhibitors von Schiaffino-Ortega, Santiago, Mariotto, Elena, Luque-Navarro, Pilar María, Kimatrai-Salvador, María, Rios-Marco, Pablo, Hurtado-Guerrero, Ramon, Marco, Carmen, Carrasco-Jimenez, María Paz, Viola, Giampietro, López-Cara, Luisa Carlota

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One-pot synthesis and biological evaluation of 2-pyrrolidinyl-4-amino-5-(3′,4′,5′-trimethoxybenzoyl)thiazole: A unique, highly active antimicrotubule agent von Romagnoli, Romeo, Baraldi, Pier Giovanni, Lopez Cara, Carlota, Kimatrai Salvador, Maria, Bortolozzi, Roberta, Basso, Giuseppe, Viola, Giampietro, Balzarini, Jan, Brancale, Andrea, Fu, Xian-Hua, Li, Jun, Zhang, Su-Zhan, Hamel, Ernest

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Synthesis and Biological Evaluation of 2‑(Alkoxycarbonyl)-3-Anilinobenzo[b]thiophenes and Thieno[2,3‑b]pyridines as New Potent Anticancer Agents von Romagnoli, Romeo, Baraldi, Pier Giovanni, Kimatrai Salvador, Maria, Preti, Delia, Aghazadeh Tabrizi, Mojgan, Bassetto, Marcella, Brancale, Andrea, Hamel, Ernest, Castagliuolo, Ignazio, Bortolozzi, Roberta, Basso, Giuseppe, Viola, Giampietro

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Design, synthesis and biological evaluation of novel vicinal diaryl-substituted 1H-Pyrazole analogues of combretastatin A-4 as highly potent tubulin polymerization inhibitors von Romagnoli, Romeo, Oliva, Paola, Salvador, Maria Kimatrai, Camacho, Maria Encarnacion, Padroni, Chiara, Brancale, Andrea, Ferla, Salvatore, Hamel, Ernest, Ronca, Roberto, Grillo, Elisabetta, Bortolozzi, Roberta, Rruga, Fatlum, Mariotto, Elena, Viola, Giampietro

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Synthesis and Antitumor Molecular Mechanism of Agents Based on Amino 2-(3′,4′,5′-Trimethoxybenzoyl)benzo[b]furan: Inhibition of Tubulin and Induction of Apoptosis von Romagnoli, Romeo, Baraldi, Pier Giovanni, Lopez-Cara, Carlota, Cruz-Lopez, Olga, Carrion, Maria Dora, Kimatrai Salvador, Maria, Bermejo, Jaime, Estévez, Sara, Estévez, Francisco, Balzarini, Jan, Brancale, Andrea, Ricci, Antonio, Chen, Longchuan, Kim, Jae Gwan, Hamel, Ernest

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Design, synthesis and biological evaluation of 2-alkoxycarbonyl-3-anilinoindoles as a new class of potent inhibitors of tubulin polymerization von Romagnoli, Romeo, Prencipe, Filippo, Oliva, Paola, Kimatrai Salvador, Maria, Brancale, Andrea, Ferla, Salvatore, Hamel, Ernest, Viola, Giampietro, Bortolozzi, Roberta, Persoons, Leentje, Balzarini, Jan, Liekens, Sandra, Schols, Dominique

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2-Alkoxycarbonyl-3-arylamino-5-substituted thiophenes as a novel class of antimicrotubule agents: Design, synthesis, cell growth and tubulin polymerization inhibition von Romagnoli, Romeo, Kimatrai Salvador, Maria, Schiaffino Ortega, Santiago, Baraldi, Pier Giovanni, Oliva, Paola, Baraldi, Stefania, Lopez-Cara, Luisa Carlota, Brancale, Andrea, Ferla, Salvatore, Hamel, Ernest, Balzarini, Jan, Liekens, Sandra, Mattiuzzo, Elena, Basso, Giuseppe, Viola, Giampietro

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Design, synthesis and biological evaluation of 3,5-disubstituted 2-amino thiophene derivatives as a novel class of antitumor agents von Romagnoli, Romeo, Baraldi, Pier Giovanni, Lopez-Cara, Carlota, Salvador, Maria Kimatrai, Preti, Delia, Tabrizi, Mojgan Aghazadeh, Balzarini, Jan, Nussbaumer, Peter, Bassetto, Marcella, Brancale, Andrea, Fu, Xian-Hua, Yang-Gao, Li, Jun, Zhang, Su-Zhan, Hamel, Ernest, Bortolozzi, Roberta, Basso, Giuseppe, Viola, Giampietro

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Synthesis and biological effects of novel 2-amino-3-(4-chlorobenzoyl)-4-substituted thiophenes as allosteric enhancers of the A1 adenosine receptor von Romagnoli, Romeo, Baraldi, Pier Giovanni, Carrion, Maria Dora, Lopez Cara, Carlota, Kimatrai Salvador, Maria, Preti, Delia, Aghazadeh Tabrizi, Mojgan, Moorman, Allan R., Vincenzi, Fabrizio, Borea, Pier Andrea, Varani, Katia

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1H and 13C NMR spectral assignments of 1,1′-(((ethane-1,2-diylbis(oxy))bis(4,1-phenylene))bis(methylene))-bispyridinium and -bisquinolinium bromide derivatives von Schiaffino-Ortega, Santiago, Kimatrai-Salvador, María, Baglioni, Eleonora, Gallo, Miguel Angel, Entrena Guadix, Antonio, Lopez-Cara, Luisa Carlota

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Allosteric modulation of A1-adenosine receptor: a review von Kimatrai-Salvador, María, Baraldi, Pier Giovanni, Romagnoli, Romeo

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Design, Synthesis, and Biological Evaluation of 6‑Substituted Thieno[3,2‑d]pyrimidine Analogues as Dual Epidermal Growth Factor Receptor Kinase and Microtubule Inhibitors von Romagnoli, Romeo, Prencipe, Filippo, Oliva, Paola, Baraldi, Stefania, Baraldi, Pier Giovanni, Schiaffino Ortega, Santiago, Chayah, Mariem, Kimatrai Salvador, Maria, Lopez-Cara, Luisa Carlota, Brancale, Andrea, Ferla, Salvatore, Hamel, Ernest, Ronca, Roberto, Bortolozzi, Roberta, Mariotto, Elena, Mattiuzzo, Elena, Viola, Giampietro

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Synthesis and Evaluation of 1,5-Disubstituted Tetrazoles as Rigid Analogues of Combretastatin A-4 with Potent Antiproliferative and Antitumor Activity von Romagnoli, Romeo, Baraldi, Pier Giovanni, Salvador, Maria Kimatrai, Preti, Delia, Aghazadeh Tabrizi, Mojgan, Brancale, Andrea, Fu, Xian-Hua, Li, Jun, Zhang, Su-Zhan, Hamel, Ernest, Bortolozzi, Roberta, Basso, Giuseppe, Viola, Giampietro

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2-Alkoxycarbonyl-3-arylamino-5-substituted thiophenes as a novel class of antimicrotubule agents: Design, synthesis, cell growth and tubulin polymerization inhibition von Romagnoli, Romeo, Kimatrai Salvador, Maria, Schiaffino Ortega, Santiago, Baraldi, Pier Giovanni, Oliva, Paola, Baraldi, Stefania, Lopez-Cara, Luisa Carlota, Brancale, Andrea, Ferla, Salvatore, Hamel, Ernest, Balzarini, Jan, Liekens, Sandra, Mattiuzzo, Elena, Basso, Giuseppe, Viola, Giampietro

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A facile synthesis of diaryl pyrroles led to the discovery of potent colchicine site antimitotic agents von Romagnoli, Romeo, Oliva, Paola, Salvador, Maria Kimatrai, Manfredini, Stefano, Padroni, Chiara, Brancale, Andrea, Ferla, Salvatore, Hamel, Ernest, Ronca, Roberto, Maccarinelli, Federica, Rruga, Fatlum, Mariotto, Elena, Viola, Giampietro, Bortolozzi, Roberta

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Design, synthesis and biological evaluation of 3-substituted-2-oxindole hybrid derivatives as novel anticancer agents von Romagnoli, Romeo, Baraldi, Pier Giovanni, Prencipe, Filippo, Oliva, Paola, Baraldi, Stefania, Salvador, Maria Kimatrai, Lopez-Cara, Luisa Carlota, Bortolozzi, Roberta, Mattiuzzo, Elena, Basso, Giuseppe, Viola, Giampietro

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Synthesis, Antimitotic and Antivascular Activity of 1‑(3′,4′,5′-Trimethoxybenzoyl)-3-arylamino-5-amino-1,2,4-triazoles von Romagnoli, Romeo, Baraldi, Pier Giovanni, Salvador, Maria Kimatrai, Prencipe, Filippo, Bertolasi, Valerio, Cancellieri, Michela, Brancale, Andrea, Hamel, Ernest, Castagliuolo, Ignazio, Consolaro, Francesca, Porcù, Elena, Basso, Giuseppe, Viola, Giampietro

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Anticancer activity of novel hybrid molecules containing 5-benzylidene thiazolidine-2,4-dione von Romagnoli, Romeo, Baraldi, Pier Giovanni, Salvador, Maria Kimatrai, Camacho, M. Encarnacion, Balzarini, Jan, Bermejo, Jaime, Estévez, Francisco

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Design, Synthesis, in Vitro, and in Vivo Anticancer and Antiangiogenic Activity of Novel 3‑Arylaminobenzofuran Derivatives Targeting the Colchicine Site on Tubulin von Romagnoli, Romeo, Baraldi, Pier Giovanni, Salvador, Maria Kimatrai, Prencipe, Filippo, Lopez-Cara, Carlota, Schiaffino Ortega, Santiago, Brancale, Andrea, Hamel, Ernest, Castagliuolo, Ignazio, Mitola, Stefania, Ronca, Roberto, Bortolozzi, Roberta, Porcù, Elena, Basso, Giuseppe, Viola, Giampietro

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Synthesis and biological evaluation of 2-substituted-4-(3′,4′,5′-trimethoxyphenyl)-5-aryl thiazoles as anticancer agents von Romagnoli, Romeo, Baraldi, Pier Giovanni, Salvador, Maria Kimatrai, Camacho, M. Encarnacion, Preti, Delia, Tabrizi, Mojgan Aghazadeh, Bassetto, Marcella, Brancale, Andrea, Hamel, Ernest, Bortolozzi, Roberta, Basso, Giuseppe, Viola, Giampietro

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