Orally bioavailable, indole-based nonpeptide GnRH receptor antagonists with high potency and functional activity von Ashton, Wallace T., Sisco, Rosemary M., Kieczykowski, Gerard R., Yang, Yi Tien, Yudkovitz, Joel B., Cui, Jisong, Mount, George R., Ren, Rena Ning, Wu, Tsuei-Ju, Shen, Xiaolan, Lyons, Kathryn A., Mao, An-Hua, Carlin, Josephine R., Karanam, Bindhu V., Vincent, Stella H., Cheng, Kang, Goulet, Mark T.

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Total synthesis of (.+-.)-vernolepin von Kieczykowski, G. R, Schlessinger, R. H

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Total synthesis of the indole alkaloids dl-eburnamonine and dl-vincamine von Herrmann, J. L, Cregge, R. J, Richman, J. E, Kieczykowski, G. R, Normandin, S. N, Quesada, M. L, Semmelhack, C. L, Poss, A. J, Schlessinger, R. H

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Preparation of (4-Amino-1-Hydroxybutylidene)bisphosphonic Acid Sodium Salt, MK-217 (Alendronate Sodium). An Improved Procedure for the Preparation of 1-Hydroxy-1,1-bisphosphonic Ac... von Kieczykowski, Gerard R, Jobson, Ronald B, Melillo, David G, Reinhold, Donald. F, Grenda, Victor J, Shinkai, Ichiro

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Prostaglandins. An efficient synthesis of a 2-alkyl-4-hydroxycyclopentenone von Kieczykowski, G. R, Pogonowski, C. S, Richman, J. E, Schlessinger, Richard H

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Total synthesis of dl-bisnorvernolepin von Kieczykowski, G. R, Quesada, Martha L, Schlessinger, R. H

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Regiospecific monoalkylation of unsaturated imines derived from crotonaldehyde von Kieczykowski, G.R., Schlessinger, R.H., Sulsky, R.B.

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Regiospecific monoalkylation of 3-butenenitrile von Kieczykowski, G.R., Schlessinger, R.H., Sulsky, R.B.

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Discovery of substituted 8,9-dicarboxyldibenzo [2,3:5,6] bicyclo [5.2.0] nonan-4-ones with moderate binding affinity to the endothelin ETA and ETB receptors von Rivero, R.A., Greenlee, W.J., Williams, P.D., Kieczykowski, G.R., Williams, D.L.

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Deconjugative alkylation of the enolate anion derived from ethyl crotonate von Herrmann, J.L., Kieczykowski, G.R., Schlessinger, R.H.

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Synthesis of sesquiterpene antitumor lactones. 2. A new stereocontrolled total synthesis of (.+-.)-vernolepin von Isobe, Minoru, Iio, Hideo, Kawai, Tatsuhiko, Goto, Toshio

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Ketene thioacetal monoxides: Some conjugate addition-alkylation reactions leading to unsymmetrical 1,4-dicarbonyl systems von Herrmann, J.L., Kieczykowski, G.R., Romanet, R.F., Schlessinger, R.H.

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Ketene thioacetal monoxides: A novel and versatile class of two-carbon michael receptors von Herrmann, J.L., Kieczykowski, G.R., Romanet, R.F., Wepplo, P.J., Schlessinger, R.H.

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A mild, selective reduction of alkoxysulfonium salts: Reductions of sulfoxides using sodium cyanohydridoborate and crown ethers von Durst, H.Dupont, Zubrick, J.W., Kieczykowski, G.R.

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Ring-opening reactions of .alpha.-oxy epoxides with tert-butyl dilithioacetoacetate von Kieczykowski, Gerard R, Roberts, Michael R, Schlessinger, Richard H

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Catalytic, Enantioselective Synthesis of Taranabant, a Novel, Acyclic Cannabinoid-1 Receptor Inverse Agonist for the Treatment of Obesity von Chen, Cheng-yi, Frey, Lisa F, Shultz, Scott, Wallace, Debra J, Marcantonio, Karen, Payack, Joeseph F, Vazquez, Enrique, Springfield, Shawn A, Zhou, George, Liu, Ping, Kieczykowski, Gerard R, Chen, Alex M, Phenix, Brian D, Singh, Utpal, Strine, Jeff, Izzo, Brianne, Krska, Shane W

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Synthesis and characterization of a potent, selective, radiolabeled substance-P antagonist for NK1 receptor quantitation: ([18F]SPA-RQ) von Solin, Olof, Eskola, Olli, Hamill, Terence G, Bergman, Jörgen, Lehikoinen, Pertti, Grönroos, Tove, Forsback, Sarita, Haaparanta, Merja, Viljanen, Tapio, Ryan, Christine, Gibson, Raymond, Kieczykowski, Gerard, Hietala, Jarmo, Hargreaves, Richard, Burns, H Donald

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Procédé de préparation d'acide amino-4 hydroxy-1 butylidéne-bisphosphonique-1,1 ou de ses sels von BRENNER GERALD S, KIECZYKOWSKI GERALD R, JOBSON RONALD B, MELILLO DAVID G

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Fremgangsmåte for fremstilling av 4-amino-1-hydroxybutyliden-1,2-bisfosfonsyresalter von KIECZYKOWSKI, GERARD R, JOBSON, RONALD B, MELILLO, DAVID G

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Fremgangsmåte for fremstilling av 4-amino-1-hydroxybutyliden-1,2-bisfosfonsyresalter von KIECZYKOWSKI, GERARD R, JOBSON, RONALD B, MELILLO, DAVID G

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