New developments in antiinfectives research for tropical infectious diseases von Chibale, Kelly

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Quinine fever von Woodland, John G., Chibale, Kelly

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The Role of Natural Products in Drug Discovery and Development against Neglected Tropical Diseases von Cheuka, Peter Mubanga, Mayoka, Godfrey, Mutai, Peggoty, Chibale, Kelly

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Antiviral drug discovery: preparing for the next pandemic von Adamson, Catherine S, Chibale, Kelly, Goss, Rebecca J. M, Jaspars, Marcel, Newman, David J, Dorrington, Rosemary A

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First fully-automated AI/ML virtual screening cascade implemented at a drug discovery centre in Africa von Turon, Gemma, Hlozek, Jason, Woodland, John G., Kumar, Ankur, Chibale, Kelly, Duran-Frigola, Miquel

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Strategies to Combat Multi-Drug Resistance in Tuberculosis von Singh, Vinayak, Chibale, Kelly

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Synthesis and In Vitro Antiprotozoan Evaluation of 4-/8-Aminoquinoline-based Lactams and Tetrazoles von Tukulula, Matshawandile, Louw, Stefan, Njoroge, Mathew, Chibale, Kelly

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Multistage and transmission-blocking targeted antimalarials discovered from the open-source MMV Pandemic Response Box von Reader, Janette, van der Watt, Mariëtte E., Taylor, Dale, Le Manach, Claire, Mittal, Nimisha, Ottilie, Sabine, Theron, Anjo, Moyo, Phanankosi, Erlank, Erica, Nardini, Luisa, Venter, Nelius, Lauterbach, Sonja, Bezuidenhout, Belinda, Horatscheck, Andre, van Heerden, Ashleigh, Spillman, Natalie J., Cowell, Anne N., Connacher, Jessica, Opperman, Daniel, Orchard, Lindsey M., Llinás, Manuel, Istvan, Eva S., Goldberg, Daniel E., Boyle, Grant A., Calvo, David, Mancama, Dalu, Coetzer, Theresa L., Winzeler, Elizabeth A., Duffy, James, Koekemoer, Lizette L., Basarab, Gregory, Chibale, Kelly, Birkholtz, Lyn-Marié

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Including African data in drug discovery and development von Veale, Clinton G. L., Edkins, Adrienne L., Winks, Susan, Njoroge, Mathew, Chibale, Kelly

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Structure elaboration of isoniazid: synthesis, in silico molecular docking and antimycobacterial activity of isoniazid–pyrimidine conjugates von Kaur, Hardeep, Singh, Lovepreet, Chibale, Kelly, Singh, Kamaljit

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How can natural products serve as a viable source of lead compounds for the development of new/novel anti-malarials? von Guantai, Eric, Chibale, Kelly

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Eliminating malaria transmission requires targeting immature and mature gametocytes through lipoidal uptake of antimalarials von Naude, Mariska, van Heerden, Ashleigh, Reader, Janette, van der Watt, Mariëtte, Niemand, Jandeli, Joubert, Dorè, Siciliano, Giulia, Alano, Pietro, Njoroge, Mathew, Chibale, Kelly, Herreros, Esperanza, Leroy, Didier, Birkholtz, Lyn-Marié

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Recent Approaches to Chemical Discovery and Development Against Malaria and the Neglected Tropical Diseases Human African Trypanosomiasis and Schistosomiasis von Njoroge, Mathew, Njuguna, Nicholas M., Mutai, Peggoty, Ongarora, Dennis S. B., Smith, Paul W., Chibale, Kelly

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Synthesis and evaluation of the performance of a small molecule library based on diverse tropane-related scaffolds von Lowe, Robert A., Taylor, Dale, Chibale, Kelly, Nelson, Adam, Marsden, Stephen P.

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Novel antimycobacterial C-21 amide derivatives of the antibiotic fusidic acid: synthesis, pharmacological evaluation and rationalization of media-dependent activity using molecular... von Dziwornu, Godwin Akpeko, Kamunya, Stephanie, Ntsabo, Tando, Chibale, Kelly

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Working toward a Globally Diverse and Inclusive Community of Medicinal Chemists of the Future

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Dihydroartemisinin inhibits prostate cancer via JARID2/miR-7/miR-34a-dependent downregulation of Axl von Paccez, Juliano D., Duncan, Kristal, Sekar, Durairaj, Correa, Ricardo G., Wang, Yihong, Gu, Xuesong, Bashin, Manoj, Chibale, Kelly, Libermann, Towia A., Zerbini, Luiz F.

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Model‐Informed Approaches to Optimizing Therapeutics in the African Patient Populations von Mulubwa, Mwila, Chibale, Kelly

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Synthetic medicinal chemistry of selected antimalarial natural products von Kumar, Vipan, Mahajan, Aman, Chibale, Kelly

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4-Aminoquinoline Antimalarials Containing a Benzylmethylpyridylmethylamine Group Are Active against Drug Resistant Plasmodium falciparum and Exhibit Oral Activity in Mice von Joshi, Mukesh C, Okombo, John, Nsumiwa, Samkele, Ndove, Jeffrey, Taylor, Dale, Wiesner, Lubbe, Hunter, Roger, Chibale, Kelly, Egan, Timothy J

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