Low intrinsic efficacy for G protein activation can explain the improved side effect profiles of new opioid agonists von Gillis, Alexander, Gondin, Arisbel B, Kliewer, Andrea, Sanchez, Julie, Lim, Herman D, Alamein, Claudia, Manandhar, Preeti, Santiago, Marina, Fritzwanker, Sebastian, Schmiedel, Frank, Katte, Timothy A, Reekie, Tristan, Grimsey, Natasha L, Kassiou, Michael, Kellam, Barrie, Krasel, Cornelius, Halls, Michelle L, Connor, Mark, Lane, J Robert, Schulz, Stefan, Christie, Macdonald J, Canals, Meritxell

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Identification of a novel toxicophore in anti-cancer chemotherapeutics that targets mitochondrial respiratory complex I von Stephenson, Zoe A, Harvey, Robert F, Pryde, Kenneth R, Mistry, Sarah, Hardy, Rachel E, Serreli, Riccardo, Chung, Injae, Allen, Timothy Eh, Stoneley, Mark, MacFarlane, Marion, Fischer, Peter M, Hirst, Judy, Kellam, Barrie, Willis, Anne E

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Development of novel fluorescent histamine H1-receptor antagonists to study ligand-binding kinetics in living cells von Stoddart, Leigh A., Vernall, Andrea J., Bouzo-Lorenzo, Monica, Bosma, Reggie, Kooistra, Albert J., de Graaf, Chris, Vischer, Henry F., Leurs, Rob, Briddon, Stephen J., Kellam, Barrie, Hill, Stephen J.

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NanoBiT Complementation to Monitor Agonist-Induced Adenosine A1 Receptor Internalization von Soave, Mark, Kellam, Barrie, Woolard, Jeanette, Briddon, Stephen J., Hill, Stephen J.

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Novel selective β1‐adrenoceptor antagonists for concomitant cardiovascular and respiratory disease von Baker, Jillian G., Gardiner, Sheila M., Woolard, Jeanette, Fromont, Christophe, Jadhav, Gopal P., Mistry, Shailesh N., Thompson, Kevin S. J., Kellam, Barrie, Hill, Stephen J., Fischer, Peter M.

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Ligand-directed covalent labelling of a GPCR with a fluorescent tag in live cells von Stoddart, Leigh A., Kindon, Nicholas D., Otun, Omolade, Harwood, Clare R., Patera, Foteini, Veprintsev, Dmitry B., Woolard, Jeanette, Briddon, Stephen J., Franks, Hester A., Hill, Stephen J., Kellam, Barrie

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A novel and selective fluorescent ligand for the study of adenosine A2B receptors von Patera, Foteini, Mistry, Sarah J., Kindon, Nicholas D., Comeo, Eleonora, Goulding, Joelle, Kellam, Barrie, Kilpatrick, Laura E., Franks, Hester, Hill, Stephen J.

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A Non-imaging High Throughput Approach to Chemical Library Screening at the Unmodified Adenosine-A3 Receptor in Living Cells von Arruda, Maria Augusta, Stoddart, Leigh A., Gherbi, Karolina, Briddon, Stephen J., Kellam, Barrie, Hill, Stephen J.

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Visualizing Ligand Binding to a GPCR In Vivo Using NanoBRET von Alcobia, Diana C., Ziegler, Alexandra I., Kondrashov, Alexander, Comeo, Eleonora, Mistry, Sarah, Kellam, Barrie, Chang, Aeson, Woolard, Jeanette, Hill, Stephen J., Sloan, Erica K.

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Subtype selective fluorescent ligands based on ICI 118,551 to study the human β2‐adrenoceptor in CRISPR/Cas9 genome‐edited HEK293T cells at low expression levels von Goulding, Joëlle, Mistry, Sarah J., Soave, Mark, Woolard, Jeanette, Briddon, Stephen J., White, Carl W., Kellam, Barrie, Hill, Stephen J.

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Insights into low molecular mass organic gelators: a focus on drug delivery and tissue engineering applications von Skilling, Kathryn J, Citossi, Francesca, Bradshaw, Tracey D, Ashford, Marianne, Kellam, Barrie, Marlow, Maria

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The evolving small‐molecule fluorescent‐conjugate toolbox for Class A GPCRs von Vernall, Andrea J, Hill, Stephen J, Kellam, Barrie

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Accelerated formation of multicellular 3-D structures by cell-to-cell cross-linking von De Bank, Paul A., Hou, Qingpu, Warner, Robert M., Wood, Ian V., Ali, Bahaa E., MacNeil, Sheila, Kendall, David A., Kellam, Barrie, Shakesheff, Kevin M., Buttery, Lee D.K.

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Collaborating for better care von White, Simon, Kellam, Barrie, Bond, Christine, Donyai, Parastou

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Drug-like Antagonists of P2Y ReceptorsFrom Lead Identification to Drug Development von Conroy, Sean, Kindon, Nicholas, Kellam, Barrie, Stocks, Michael J

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Modulators of CXCR4 and CXCR7/ACKR3 Function von Adlere, Ilze, Caspar, Birgit, Arimont, Marta, Dekkers, Sebastian, Visser, Kirsten, Stuijt, Jeffrey, de Graaf, Chris, Stocks, Michael, Kellam, Barrie, Briddon, Stephen, Wijtmans, Maikel, de Esch, Iwan, Hill, Stephen, Leurs, Rob

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Monitoring Allosteric Interactions with CXCR4 Using NanoBiT Conjugated Nanobodies von Soave, Mark, Heukers, Raimond, Kellam, Barrie, Woolard, Jeanette, Smit, Martine J., Briddon, Stephen J., Hill, Stephen J.

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Science and Practice back together again von White, Simon, Kellam, Barrie, Bond, Christine, Donyai, Parastou

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Allosteric interactions at adenosine A1 and A3 receptors: new insights into the role of small molecules and receptor dimerization von Hill, Stephen J, May, Lauren T, Kellam, Barrie, Woolard, Jeanette

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Subtype-Selective Fluorescent Ligands as Pharmacological Research Tools for the Human Adenosine A2A Receptor von Comeo, Eleonora, Kindon, Nicholas D, Soave, Mark, Stoddart, Leigh A, Kilpatrick, Laura E, Scammells, Peter J, Hill, Stephen J, Kellam, Barrie

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