Practical Considerations in Kinetic Resolution Reactions von Keith, John M., Larrow, Jay F., Jacobsen, Eric N.

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One-Step Conversion of Azine N-Oxides to α-1,2,4-Triazolo-, 1,2,3-Triazolo, Imidazolo-, and Pyrazoloheteroarenes von Keith, John M

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Asymmetric Hydrocyanation of Hydrazones Catalyzed by Lanthanide−PYBOX Complexes von Keith, John M, Jacobsen, Eric N

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Biochemical and Biological Properties of 4-(3-phenyl-[1,2,4] thiadiazol-5-yl)-piperazine-1-carboxylic acid phenylamide, a Mechanism-Based Inhibitor of Fatty Acid Amide Hydrolase von Karbarz, Mark J., Luo, Lin, Chang, Leon, Tham, Chui-Se, Palmer, James A., Wilson, Sandy J., Wennerholm, Michelle L., Brown, Sean M., Scott, Brian P., Apodaca, Richard L., Keith, John M., Wu, Jiejun, Breitenbucher, James Guy, Chaplan, Sandra R., Webb, Michael

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One-Step Conversion of Azine N‑Oxides to α‑N‑Aryltriflamidoazines von Keith, John M

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Lead identification of acetylcholinesterase inhibitors-histamine H3 receptor antagonists from molecular modeling von BEMBENEK, Scott D, KEITH, John M, LETAVIC, Michael A, APODACA, Richard, BARBIER, Ann J, DVORAK, Lisa, ALUISIO, Leah, MILLER, Kirsten L, LOVENBERG, Timothy W, CARRUTHERS, Nicholas I

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One-Step Conversion of Pyridine N-Oxides to Tetrazolo[1,5-a]pyridines von Keith, John M

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Selective ortho-cleavage of methoxymethyl- and 4-methoxybenzyl ethers von Keith, John M

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One Step Conversion of Heteroaromatic-N-Oxides to Imidazolo-Heteroarenes von Keith, John M

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Heteroarylureas with fused bicyclic diamine cores as inhibitors of fatty acid amide hydrolase von Keith, John M., Jones, William, Pierce, Joan M., Seierstad, Mark, Palmer, James A., Webb, Michael, Karbarz, Mark, Scott, Brian P., Wilson, Sandy J., Luo, Lin, Wennerholm, Michelle, Chang, Leon, Rizzolio, Michele, Rynberg, Raymond, Chaplan, Sandra, Guy Breitenbucher, J.

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Dual serotonin transporter/histamine H3 ligands : Optimization of the H3 pharmacophore von KEITH, John M, GOMEZ, Leslie A, MAZUR, Curt, LOVENBERG, Timothy W, CARRUTHERS, Nicholas I, LETAVIC, Michael A, LY, Kiev S, JABLONOWSKI, Jill A, SEIERSTAD, Mark, BARBIER, Ann J, WILSON, Sandy J, BOGGS, Jamin D, FRASER, Ian C

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Preclinical Characterization of the FAAH Inhibitor JNJ-42165279 von Keith, John M, Jones, William M, Tichenor, Mark, Liu, Jing, Seierstad, Mark, Palmer, James A, Webb, Michael, Karbarz, Mark, Scott, Brian P, Wilson, Sandy J, Luo, Lin, Wennerholm, Michelle L, Chang, Leon, Rizzolio, Michele, Rynberg, Raymond, Chaplan, Sandra R, Breitenbucher, J. Guy

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A Single Amino Acid Difference between Mouse and Human 5-Lipoxygenase Activating Protein (FLAP) Explains the Speciation and Differential Pharmacology of Novel FLAP Inhibitors von Blevitt, Jonathan M., Hack, Michael D., Herman, Krystal, Chang, Leon, Keith, John M., Mirzadegan, Tara, Rao, Navin L., Lebsack, Alec D., Milla, Marcos E.

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Exploration of the Mitsunobu Reaction with Tosyl- and Boc-Hydrazones as Nucleophilic Agents von Keith, John M, Gomez, Leslie

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Heteroarylureas with spirocyclic diamine cores as inhibitors of fatty acid amide hydrolase von Keith, John M., Jones, William M., Pierce, Joan M., Seierstad, Mark, Palmer, James A., Webb, Michael, Karbarz, Mark J., Scott, Brian P., Wilson, Sandy J., Luo, Lin, Wennerholm, Michelle L., Chang, Leon, Brown, Sean M., Rizzolio, Michele, Rynberg, Raymond, Chaplan, Sandra R., Breitenbucher, J. Guy

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Thiadiazolopiperazinyl ureas as inhibitors of fatty acid amide hydrolase von Keith, John M., Apodaca, Richard, Xiao, Wei, Seierstad, Mark, Pattabiraman, Kanaka, Wu, Jiejun, Webb, Michael, Karbarz, Mark J., Brown, Sean, Wilson, Sandy, Scott, Brian, Tham, Chui-Se, Luo, Lin, Palmer, James, Wennerholm, Michelle, Chaplan, Sandra, Breitenbucher, J. Guy

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The SAR of brain penetration for a series of heteroaryl urea FAAH inhibitors von Keith, John M., Tichenor, Mark S., Apodaca, Richard L., Xiao, Wei, Jones, William M., Seierstad, Mark, Pierce, Joan M., Palmer, James A., Webb, Michael, Karbarz, Mark J., Scott, Brian P., Wilson, Sandy J., Wennerholm, Michelle L., Rizzolio, Michele, Rynberg, Raymond, Chaplan, Sandra R., Breitenbucher, J. Guy

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1-Aryl-2-((6-aryl)pyrimidin-4-yl)amino)ethanols as competitive inhibitors of fatty acid amide hydrolase von Keith, John M, Hawryluk, Natalie, Apodaca, Richard L, Chambers, Allison, Pierce, Joan M, Seierstad, Mark, Palmer, James A, Webb, Michael, Karbarz, Mark J, Scott, Brian P, Wilson, Sandy J, Luo, Lin, Wennerholm, Michelle L, Chang, Leon, Rizzolio, Michele, Chaplan, Sandra R, Breitenbucher, J Guy

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Heteroaryl urea inhibitors of fatty acid amide hydrolase: Structure–mutagenicity relationships for arylamine metabolites von Tichenor, Mark S., Keith, John M., Jones, William M., Pierce, Joan M., Merit, Jeff, Hawryluk, Natalie, Seierstad, Mark, Palmer, James A., Webb, Michael, Karbarz, Mark J., Wilson, Sandy J., Wennerholm, Michelle L., Woestenborghs, Filip, Beerens, Dominiek, Luo, Lin, Brown, Sean M., Boeck, Marlies De, Chaplan, Sandra R., Breitenbucher, J. Guy

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Polypharmacology of Small-Molecule Modulators of the 5-Lipoxygenase Activating Protein (FLAP) Observed via a High-throughput Lipidomics Platform von Song, Jiao, Liu, Xuejun, Zhu, Jian, Tootoonchi, Mandana, Keith, John M., Meduna, Steven P., Dvorak, Curt A., Eccles, Wendy, Krawczuk, Paul J., Blevitt, Jonathan M., Wu, Jiejun, Rao, Navin L., Lebsack, Alec D., Milla, Marcos E.

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