Design and Identification of a GPR40 Full Agonist (SCO-267) Possessing a 2‑Carbamoylphenyl Piperidine Moiety von Furukawa, Hideki, Miyamoto, Yasufumi, Hirata, Yasuhiro, Watanabe, Koji, Hitomi, Yuko, Yoshitomi, Yayoi, Aida, Jumpei, Noguchi, Naoyoshi, Takakura, Nobuyuki, Takami, Kazuaki, Miwatashi, Seiji, Hirozane, Yoshihiko, Hamada, Teruki, Ito, Ryo, Ookawara, Mitsugi, Moritoh, Yusuke, Watanabe, Masanori, Maekawa, Tsuyoshi

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Stereoselective Hydrothiolation of Alkynes Catalyzed by Cesium Base:  Facile Access to (Z)-1-Alkenyl Sulfides von Kondoh, Azusa, Takami, Kazuaki, Yorimitsu, Hideki, Oshima, Koichiro

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Trans-Hydrometalation of Alkynes by a Combination of InCl3 and DIBAL-H:  One-Pot Access to Functionalized (Z)-Alkenes von Takami, Kazuaki, Yorimitsu, Hideki, Oshima, Koichiro

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Triethylborane-Mediated Hydrogallation and Hydroindation:  Novel Access to Organogalliums and Organoindiums von Takami, Kazuaki, Mikami, Satoshi, Yorimitsu, Hideki, Shinokubo, Hiroshi, Oshima, Koichiro

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Discovery of a novel series of GPR119 agonists: Design, synthesis, and biological evaluation of N-(Piperidin-4-yl)-N-(trifluoromethyl)pyrimidin-4-amine derivatives von Kubo, Osamu, Takami, Kazuaki, Kamaura, Masahiro, Watanabe, Koji, Miyashita, Hirohisa, Abe, Shinichi, Matsuda, Kae, Tsujihata, Yoshiyuki, Odani, Tomoyuki, Iwasaki, Shinji, Kitazaki, Tomoyuki, Murata, Toshiki, Sato, Kenjiro

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Discovery of Pyrazolo[1,5-a]pyrazin-4-ones as Potent and Brain Penetrant GluN2A-Selective Positive Allosteric Modulators Reducing AMPA Receptor Binding Activity von Sakurai, Fumie, Yukawa, Takafumi, Kina, Asato, Murakami, Masataka, Takami, Kazuaki, Morimoto, Sachie, Seto, Masaki, Kamata, Makoto, Yamashita, Tohru, Nakashima, Kosuke, Narita, Naohiro, Bettini, Ezio, Ugolini, Annarosa, Corsi, Mauro, Hasui, Tomoaki

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Discovery of Brain-Penetrant Glucosylceramide Synthase Inhibitors with a Novel Pharmacophore von Tanaka, Yuta, Seto, Masaki, Kakegawa, Keiko, Takami, Kazuaki, Kikuchi, Fumiaki, Yamamoto, Takeshi, Nakamura, Minoru, Daini, Masaki, Murakami, Masataka, Ohashi, Tomohiro, Kasahara, Takahito, Wang, Junsi, Ikeda, Zenichi, Wada, Yasufumi, Puenner, Florian, Fujii, Takahiro, Inazuka, Masakazu, Sato, Sho, Suzaki, Tomohiko, Oak, Jeong-Ho, Takai, Yuichi, Kohara, Hiroshi, Kimoto, Kouya, Oki, Hideyuki, Mikami, Satoshi, Sasaki, Minoru, Tanaka, Yuta

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Discovery of a novel series of medium-sized cyclic enteropeptidase inhibitors von Kikuchi, Fumiaki, Ikeda, Zenichi, Kakegawa, Keiko, Nishikawa, Youichi, Sasaki, Shigekazu, Fukuda, Koichiro, Takami, Kazuaki, Banno, Yoshihiro, Nishikawa, Hitoaki, Taya, Naohiro, Nakahata, Takashi, Itono, Sachiko, Yashiro, Hiroaki, Tsuchimori, Kazue, Hiyoshi, Hideyuki, Sasaki, Masako, Tohyama, Kimio, Matsumiya, Kouta, Ishihara, Youko, Kawamoto, Tetsuji, Kamaura, Masahiro, Watanabe, Masanori, Kitazaki, Tomoyuki, Maekawa, Tsuyoshi, Sasaki, Minoru

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Efficient and Stereoselective Syntheses of Isomerically Pure 4‑Aminotetrahydro‑2H‑thiopyran 1‑Oxide Derivatives von Mizojiri, Ryo, Takami, Kazuaki, Ito, Tatsuya, Maeda, Hiroyuki, Yamano, Mitsuhisa, Kawamoto, Tetsuji

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Efficient and Stereoselective Syntheses of Isomerically Pure 4-Aminotetrahydro-2 H -thiopyran 1-Oxide Derivatives von Mizojiri, Ryo, Takami, Kazuaki, Ito, Tatsuya, Maeda, Hiroyuki, Yamano, Mitsuhisa, Kawamoto, Tetsuji

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Abstract 2793: Design, synthesis and evaluations of novel class of orally bioavailable eIF4A3-selective inhibitors von Mizojiri, Ryo, Nakata, Daisuke, Satoh, Yoshihiko, Morishita, Daisuke, Shibata, Sachio, Iwatani-Yoshihara, Misa, Kosugi, Yohei, Kosaka, Mai, Takeda, Junpei, Sasaki, Shigekazu, Takami, Kazuaki, Fukuda, Koichiro, Kamaura, Masahiro, Sasaki, Shinobu, Arai, Ryosuke, Cary, Douglas R., Imaeda, Yasuhiro

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Discovery of Novel 5‑(Piperazine-1-carbonyl)pyridin-2(1H)‑one Derivatives as Orally eIF4A3-Selective Inhibitors von Mizojiri, Ryo, Nakata, Daisuke, Satoh, Yoshihiko, Morishita, Daisuke, Shibata, Sachio, Iwatani-Yoshihara, Misa, Kosugi, Yohei, Kosaka, Mai, Takeda, Junpei, Sasaki, Shigekazu, Takami, Kazuaki, Fukuda, Koichiro, Kamaura, Masahiro, Sasaki, Shinobu, Arai, Ryosuke, Cary, Douglas R, Imaeda, Yasuhiro

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Radical Alkenylation of α-Halo Carbonyl Compounds with Alkenylindiums von Takami, Kazuaki, Yorimitsu, Hideki, Oshima, Koichiro

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Palladium-Catalyzed Cross-Coupling Reaction of Organoindiums with Aryl Halides in Aqueous Media von Takami, Kazuaki, Yorimitsu, Hideki, Shinokubo, Hiroshi, Matsubara, Seijiro, Oshima, Koichiro

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Synthesis, Structure–Activity Relationship, and Pharmacological Studies of Novel Melanin-Concentrating Hormone Receptor 1 Antagonists 3-Aminomethylquinolines: Reducing Human Ether-... von Kasai, Shizuo, Kamata, Makoto, Masada, Shinichi, Kunitomo, Jun, Kamaura, Masahiro, Okawa, Tomohiro, Takami, Kazuaki, Ogino, Hitomi, Nakano, Yoshihide, Ashina, Shuntarou, Watanabe, Kaoru, Kaisho, Tomoko, Imai, Yumi N, Ryu, Sunghi, Nakayama, Masaharu, Nagisa, Yasutaka, Takekawa, Shiro, Kato, Koki, Murata, Toshiki, Suzuki, Nobuhiro, Ishihara, Yuji

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Radical Allylation, Vinylation, Alkynylation, and Phenylation Reactions of α-Halo Carbonyl Compounds with Organoboron, Organogallium, and Organoindium Reagents von Takami, Kazuaki, Usugi, Shin-ichi, Yorimitsu, Hideki, Oshima, Koichiro

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Triethylborane-induced radical reactions with gallium- and indium hydrides von Takami, Kazuaki, Mikami, Satoshi, Yorimitsu, Hideki, Shinokubo, Hiroshi, Oshima, Koichiro

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On the “musicality” of emotional speech: Calculating harmony using fundamental frequencies von FUJISAWA, Takashi, TAKAMI, Kazuaki, COOK, Norman D.

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Reaction of Silyldihalomethyllithiums with Nitriles:  Formation of α-Keto Acylsilanes via Azirines and 1,3-Rearrangement of Silyl Group from C to N von Yagi, Kazunari, Tsuritani, Takayuki, Takami, Kazuaki, Shinokubo, Hiroshi, Oshima, Koichiro

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Evaluation of the affective valence of speech using pitch substructure von Cook, N.D., Fujisawa, T.X., Takami, K.

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