A new type of synthetic peptide library for identifying ligand-binding activity von Lam, Kit S, Salmon, Sydney E, Hersh, Evan M, Hruby, Victor J, Kazmierski, Wieslaw M, Knapp, Richard J

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The CCR5 Receptor-Based Mechanism of Action of 873140, a Potent Allosteric Noncompetitive HIV Entry Inhibitor von Watson, Christian, Jenkinson, Stephen, Kazmierski, Wieslaw, Kenakin, Terry

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764 IN VITRO PROFILING OF GSK2336805, A POTENT AND SELECTIVE INHIBITOR OF HCV NS5A von Bechtel, J, Crosby, R, Wang, A, Woldu, E, Van Horn, S, Horton, J, Creech, K, Caballo, L.H, Voitenleitner, C, Vamathevan, J, Duan, M, Spaltenstein, A, Kazmierski, W, Roberts, C, Hamatake, R

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Emerging approaches in the molecular design of receptor-selective peptide ligands: conformational, topographical and dynamic considerations von Hruby, V J, al-Obeidi, F, Kazmierski, W

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Novel inhibitors of HIV protease : Design, synthesis and biological evaluation of picomolar inhibitors containing cyclic P1/P2 scaffolds von SPALTENSTEIN, A, ALMOND, M. R, BOCK, W. J, CLEARY, D. G, FURFINE, E. S, HAZEN, R. J, KAZMIERSKI, W. M, SALITURO, F. G, TUNG, R. D, WRIGHT, L. L

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Recent progress in discovery of small-molecule CCR5 chemokine receptor ligands as HIV-1 inhibitors von KAZMIERSKI, Wieslaw, BIFULCO, Neil, YANG, Hanbiao, BOONE, Larry, DEANDA, Felix, WATSON, Chris, KENAKIN, Terry

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TARGETING THE NS5A PROTEIN OF HCV: AN EMERGING OPTION von Cordek, D G, Bechtel, J T, Maynard, A T, Kazmierski, W M, Cameron, C E

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Iron Chelates Bind Nitric Oxide and Decrease Mortality in an Experimental Model of Septic Shock von Kazmierski, Wieslaw M., Wolberg, Gerald, Wilson, Joan G., Smith, Sheila R., Williams, Darryl S., Thorp, H. Holden, Molina, Luis

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New Amino Acids for the Topographical Control of Peptide Conformation: Synthesis of All the Isomers of .alpha.,.beta.-Dimethylphenylalanine and .alpha.,.beta.-Dimethyl-1,2,3,4-tetr... von Kazmierski, Wieslaw M, Urbanczyk-Lipkowska, Zofia, Hruby, Victor J

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Topographic design of peptide neurotransmitters and hormones on stable backbone templates: relation of conformation and dynamics to bioactivity von Kazmierski, Wieslaw M, Yamamura, Henry I, Hruby, Victor J

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Inhibitors of Human Immunodeficiency Virus Type 1 Derived from gp41 Transmembrane Protein:  Structure−Activity Studies von Kazmierski, Wieslaw M, Hazen, Richard J, Aulabaugh, Ann, StClair, Marty H

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4,4-Disubstituted Cyclohexylamine based CCR5 Chemokine Receptor Antagonists as Anti-HIV-1 agents von Duan, Maosheng, Kazmierski, Wieslaw, Aquino, Christopher, Ferris, Rob, Kenakin, Terry, Watson, Chris, Wheelan, Pat

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Small-molecule CCR5 Ligands that may Spare the CCR5 Function: Opportunity for New Antiviral Discovery? von Kazmierski, Wieslaw, Muniz-Medina, Vanessa, Danehower, Susan, Jones, Stacey, Kenakin, Terry

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Recent advances in the design and synthesis of small-molecule mimetic drugs von Kazmierski, Wieslaw M.

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Discovery of potent pyrrolidone-based HIV-1 protease inhibitors with enhanced drug-like properties von KAZMIERSKI, Wieslaw M, ANDREWS, Webb, FURFINE, Eric, SPALTENSTEIN, Andrew, WRIGHT, Lois

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Unexpected antinociceptive potency of cyclic [D-Tca 1]CTAP: potential for a novel mechanism of action von Horan, Peter J., Wild, Kenneth D., Kazmierski, Wieslaw W., Ferguson, Ronald, Hruby, Victor J., Weber, Steven J., Davis, Thomas P., Fang, Lei, Knapp, Richard J., Yamamura, Henry I., Kramer, Thomas H., Burks, Thomas F., Bowen, Wayne D., Takemori, A.E., Porreca, Frank

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A solid-phase approach to analogues of the antibiotic mureidomycin von Bozzoli, Andrea, Kazmierski, Wieslaw, Kennedy, Gordon, Pasquarello, Alessandra, Pecunioso, Angelo

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CONSTRAINED PHENYLALANINE ANALOGS - PREFERRED CONFORMATION OF THE 1,2,3,4-TETRAHYDROISOQUINOLINE-3-CARBOXYLIC ACID (TIC) RESIDUE von VALLE, G, KAZMIERSKI, WM, CRISMA, M, BONORA, GM, TONIOLO, C, HRUBY, VJ

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Potent inhibitors of the HIV-1 protease incorporating cyclic urea P1-P2 scaffold von KAZMIERSKI, Wieslaw M, FURFINE, Eric, GRAY-NUNEZ, Yolanda, SPALTENSTEIN, Andrew, WRIGHT, Lois

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Peptide, Peptidomimetic and Small-molecule Drug Discovery Targeting HIV-1 Host-cell Attachment and Entry through gp120, gp41, CCR5 and CXCR4 von Kazmierski, Wieslaw M., Kenakin, Terry P., Gudmundsson, Kristjan S.

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