Asymmetric Ni(II)/Cr(II)-Mediated Coupling Reaction:  Catalytic Process von Choi, Hyeong-wook, Nakajima, Katsumasa, Demeke, Damtew, Kang, Fu-An, Jun, Hyuk-Sang, Wan, Zhao-Kui, Kishi, Yoshito

Volltext

Asymmetric Ni(II)/Cr(II)-Mediated Coupling Reaction:  Stoichiometric Process von Wan, Zhao-Kui, Choi, Hyeong-wook, Kang, Fu-An, Nakajima, Katsumasa, Demeke, Damtew, Kishi, Yoshito

Volltext

Discovery of Orally Active Inhibitors of Brahma Homolog (BRM)/SMARCA2 ATPase Activity for the Treatment of Brahma Related Gene 1 (BRG1)/SMARCA4-Mutant Cancers von Papillon, Julien P. N, Nakajima, Katsumasa, Adair, Christopher D, Hempel, Jonathan, Jouk, Andriana O, Karki, Rajeshri G, Mathieu, Simon, Möbitz, Henrik, Ntaganda, Rukundo, Smith, Troy, Visser, Michael, Hill, Susan E, Hurtado, Felipe Kellermann, Chenail, Gregg, Bhang, Hyo-Eun C, Bric, Anka, Xiang, Kay, Bushold, Geoffrey, Gilbert, Tamara, Vattay, Anthony, Dooley, Julie, Costa, Emily A, Park, Isabel, Li, Ailing, Farley, David, Lounkine, Eugen, Yue, Q. Kimberley, Xie, Xiaoling, Zhu, Xiaoping, Kulathila, Raviraj, King, Daniel, Hu, Tiancen, Vulic, Katarina, Cantwell, John, Luu, Catherine, Jagani, Zainab

Volltext

Enantioselective Synthesis of (−)-Pumiliotoxin C from a Chiral Amino Ester and an Acetylenic Sulfone that Acts as an Alkene Dipole Equivalent von Back, Thomas G, Nakajima, Katsumasa

Volltext

Identification of a PCSK9-LDLR disruptor peptide with in vivo function von Brousseau, Margaret E., Clairmont, Kevin B., Spraggon, Glen, Flyer, Alec N., Golosov, Andrei A., Grosche, Philipp, Amin, Jakal, Andre, Jerome, Burdick, Debra, Caplan, Shari, Chen, Guanjing, Chopra, Raj, Ames, Lisa, Dubiel, Diana, Fan, Li, Gattlen, Raphael, Kelly-Sullivan, Dawn, Koch, Alexander W., Lewis, Ian, Li, Jingzhou, Liu, Eugene, Lubicka, Danuta, Marzinzik, Andreas, Nakajima, Katsumasa, Nettleton, David, Ottl, Johannes, Pan, Meihui, Patel, Tajesh, Perry, Lauren, Pickett, Stephanie, Poirier, Jennifer, Reid, Patrick C., Pelle, Xavier, Seepersaud, Mohindra, Subramanian, Vanitha, Vera, Victoria, Xu, Mei, Yang, Lihua, Yang, Qing, Yu, Jinghua, Zhu, Guoming, Monovich, Lauren G.

Volltext

Design of Thioether Cyclic Peptide Scaffolds with Passive Permeability and Oral Exposure von Golosov, Andrei A, Flyer, Alec N, Amin, Jakal, Babu, Charles, Gampe, Christian, Li, Jingzhou, Liu, Eugene, Nakajima, Katsumasa, Nettleton, David, Patel, Tajesh J, Reid, Patrick C, Yang, Lihua, Monovich, Lauren G

Volltext

The Discovery of SWI/SNF Chromatin Remodeling Activity as a Novel and Targetable Dependency in Uveal Melanoma von Rago, Florencia, Elliott, GiNell, Li, Ailing, Sprouffske, Kathleen, Kerr, Grainne, Desplat, Aurore, Abramowski, Dorothee, Chen, Julie T., Farsidjani, Ali, Xiang, Kay X., Bushold, Geoffrey, Feng, Yun, Shirley, Matthew D., Bric, Anka, Vattay, Anthony, Moebitz, Henrik, Nakajima, Katsumasa, Adair, Christopher D., Mathieu, Simon, Ntaganda, Rukundo, Smith, Troy, Papillon, Julien P. N., Kauffmann, Audrey, Ruddy, David A., Bhang, Hyo-eun C., Castelletti, Deborah, Jagani, Zainab

Volltext

Abstract 10516: Identification of a PCSK9-LDLR Disruptor Macrocycle with in vivo Function von Brousseau, Margaret E, Clairmont, Kevin B, Spraggon, Glen, Flyer, Alec N, Golosov, Andrei A, Grosche, Philipp, André, Jérôme, Caplan, Shari, Chen, Guanjing, Fan, Li, Gattlen, Raphael, Koch, Alexander, Lewis, Ian, Li, Jingzhou, Liu, Eugene, Lubicka, Danuta, Marzinzik, Andreas, Nakajima, Katsumasa, Nettleton, David, Ottl, Johannes, Pan, Meihui, Patel, Tajesh, Pickett, Stephanie, Poirier, Jennifer, Reid, Patrick C, Pelle, Xavier, Subramanian, Vanitha, Vera, Victoria, Xu, Mei, Yang, Lihua, Yang, Qing, yu, jinghua, Zhu, Guoming, Monovich, Lauren G

Volltext

Tandem Conjugate Additions and 3-Aza-Cope Rearrangements of Tertiary Allyl Amines and Cyclic α-Vinylamines with Acetylenic Sulfones. Applications to Simple and Iterative Ring Expan... von Weston, Mitchell H, Nakajima, Katsumasa, Back, Thomas G

Volltext

Discovery of an Orally Bioavailable Benzimidazole Diacylglycerol Acyltransferase 1 (DGAT1) Inhibitor That Suppresses Body Weight Gain in Diet-Induced Obese Dogs and Postprandial Tr... von Nakajima, Katsumasa, Chatelain, Ricardo, Clairmont, Kevin B, Commerford, Renee, Coppola, Gary M, Daniels, Thomas, Forster, Cornelia J, Gilmore, Thomas A, Gong, Yongjin, Jain, Monish, Kanter, Aaron, Kwak, Youngshin, Li, Jingzhou, Meyers, Charles D, Neubert, Alan D, Szklennik, Paul, Tedesco, Vivienne, Thompson, James, Truong, David, Yang, Qing, Hubbard, Brian K, Serrano-Wu, Michael H

Volltext

Use of an acetylenic sulfone as an alkene dipole equivalent in the synthesis of (±)-pumiliotoxin C von Back, Thomas G., Nakajima, Katsumasa

Volltext

Discovery of diamide compounds as diacylglycerol acyltransferase 1 (DGAT1) inhibitors von Nakajima, Katsumasa, April, Myriam, Brewer, Jason T., Daniels, Thomas, Forster, Cornelia J., Gilmore, Thomas A., Jain, Monish, Kanter, Aaron, Kwak, Youngshin, Li, Jingzhou, McQuire, Les, Serrano-Wu, Michael H., Streeper, Ryan, Szklennik, Paul, Thompson, James, Wang, Bing

Volltext

A Convenient New Route to Piperidines, Pyrrolizidines, Indolizidines, and Quinolizidines by Cyclization of Acetylenic Sulfones with β- and γ-Chloroamines. Enantioselective Total Sy... von Back, Thomas G, Nakajima, Katsumasa

Volltext

Ring-expansion of tertiary cyclic alpha-vinylamines by tandem conjugate addition to (p-toluenesulfonyl)ethyne and formal 3-aza-Cope rearrangement von Weston, Mitchell H, Nakajima, Katsumasa, Parvez, Masood, Back, Thomas G

Volltext

Synthetic studies on the marine natural product halichondrins von Choi, Hyeong-wook, Demeke, Damtew, Kang, F.-A., Kishi, Y., Nakajima, K., Nowak, P., Wan, Z.-K., Xie, C.

Volltext

Chemically modified messenger RNA's von Caplan, Shari Lynn, Nakajima, Katsumasa

Volltext bestellen

Synthesis of Substituted Piperidines, Indolizidines, Quinolizidines, and Pyrrolizidines via a Cycloaddition Strategy Using Acetylenic Sulfones as Alkene Dipole Equivalents von Back, Thomas G, Nakajima, Katsumasa

Volltext

Unsymmetrical Ozonolysis of a Diels−Alder Adduct:  Practical Preparation of a Key Intermediate for Heme Total Synthesis von Taber, Douglass F, Nakajima, Katsumasa

Volltext

UREA COMPOUNDS AND COMPOSITIONS AS SMARCA2/BRM ATPASE INHIBITORS von ADAIR, Christopher, Ntaganda, Rukundo, Nakajima, Katsumasa, Smith, Troy Douglas, Papillon, Julien

Volltext bestellen

CHEMICALLY MODIFIED MESSENGER RNA'S von NAKAJIMA, Katsumasa, CAPLAN, Shari Lynn

Volltext bestellen