Concise Syntheses of Meridianins by Carbonylative Alkynylation and a Four-Component Pyrimidine Synthesis von Karpov, Alexei S., Merkul, Eugen, Rominger, Frank, Müller, Thomas J. J.

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New Entry to a Three-Component Pyrimidine Synthesis by TMS−Ynones via Sonogashira Coupling von Karpov, Alexei S, Müller, Thomas J. J

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Optimization of a Dibenzodiazepine Hit to a Potent and Selective Allosteric PAK1 Inhibitor von Karpov, Alexei S, Amiri, Payman, Bellamacina, Cornelia, Bellance, Marie-Helene, Breitenstein, Werner, Daniel, Dylan, Denay, Regis, Fabbro, Doriano, Fernandez, Cesar, Galuba, Inga, Guerro-Lagasse, Stephanie, Gutmann, Sascha, Hinh, Linda, Jahnke, Wolfgang, Klopp, Julia, Lai, Albert, Lindvall, Mika K, Ma, Sylvia, Möbitz, Henrik, Pecchi, Sabina, Rummel, Gabriele, Shoemaker, Kevin, Trappe, Joerg, Voliva, Charles, Cowan-Jacob, Sandra W, Marzinzik, Andreas L

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Nicotinamide Phosphoribosyltransferase Inhibitor as a Novel Payload for Antibody–Drug Conjugates von Karpov, Alexei S, Abrams, Tinya, Clark, Suzanna, Raikar, Ankita, D’Alessio, Joseph A, Dillon, Michael P, Gesner, Thomas G, Jones, Darryl, Lacaud, Marion, Mallet, William, Martyniuk, Piotr, Meredith, Erik, Mohseni, Morvarid, Nieto-Oberhuber, Cristina M, Palacios, Daniel, Perruccio, Francesca, Piizzi, Grazia, Zurini, Mauro, Bialucha, Carl Uli

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Modular synthesis and modification of novel bifunctional dendrons von Tulli, Ludovico G, Miranda, Daniela, Lee, Cameron C, Sullivan, Yang, Grotzfeld, Robert, Hollingworth, Gregory, Kneuer, Rainer, Karpov, Alexei S

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Facile One-Pot Coupling−Aminovinylation Approach to Push−Pull Chromophores:  Alkyne Activation by Sonogashira Coupling von Karpov, Alexei S, Rominger, Frank, Müller, Thomas J. J

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Benzimidazolyl-pyrazolo[3,4‑b]pyridinones, Selective Inhibitors of MOLT‑4 Leukemia Cell Growth and Sea Urchin Embryo Spiculogenesis: Target Quest von Lichitsky, Boris V, Komogortsev, Andrey N, Dudinov, Arkady A, Krayushkin, Mikhail M, Khodot, Evgenii N, Samet, Alexander V, Silyanova, Eugenia A, Konyushkin, Leonid D, Karpov, Alexei S, Gorses, Delphine, Radimerski, Thomas, Semenova, Marina N, Kiselyov, Alex S, Semenov, Victor V

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Discovery of Potent and Selective Antibody–Drug Conjugates with Eg5 Inhibitors through Linker and Payload Optimization von Karpov, Alexei S, Nieto-Oberhuber, Cristina M, Abrams, Tinya, Beng-Louka, Edwige, Blanco, Enrique, Chamoin, Sylvie, Chene, Patrick, Dacquignies, Isabelle, Daniel, Dylan, Dillon, Michael P, Doumampouom-Metoul, Lionel, Drosos, Nikolaos, Fedoseev, Pavel, Furegati, Markus, Granda, Brian, Grotzfeld, Robert M, Hess Clark, Suzanna, Joly, Emilie, Jones, Darryl, Lacaud-Baumlin, Marion, Lagasse-Guerro, Stephanie, Lorenzana, Edward G, Mallet, William, Martyniuk, Piotr, Marzinzik, Andreas L, Mesrouze, Yannick, Nocito, Sandro, Oei, Yoko, Perruccio, Francesca, Piizzi, Grazia, Richard, Etienne, Rudewicz, Patrick J, Schindler, Patrick, Velay, Mélanie, Venstrom, Kristine, Wang, Peiyin, Zurini, Mauro, Lafrance, Marc

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A novel one-pot three-component synthesis of 3-halofurans and sequential Suzuki coupling von Karpov, Alexei S, Merkul, Eugen, Oeser, Thomas, Müller, Thomas J J

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A novel one-pot four-component access to tetrahydro-beta-carbolines by a coupling-amination-aza-annulation-Pictet-Spengler sequence (CAAPS) von Karpov, Alexei S, Oeser, Thomas, Müller, Thomas J J

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A diversity oriented four-component approach to tetrahydro-beta-carbolines initiated by Sonogashira coupling von Karpov, Alexei S, Rominger, Frank, Müller, Thomas J J

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A new convenient approach to chiral β-aryl(heteroaryl)alkylamines von Nenajdenko, Valentine G, Karpov, Alexei S, Balenkova, Elizabeth S

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Straightforward Novel One-Pot Enaminone and Pyrimidine Syntheses by Coupling-Addition-Cyclocondensation Sequences von Karpov, Alexei S., Müller, Thomas J.

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One-Pot Three-Component Synthesis of 3-Halofurans and 3-Chloro-4-iodofurans von Karpov, Alexei S., Merkul, Eugen, Oeser, Thomas, Müller, Thomas J. J.

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Kurze Meridianin‐Synthesen durch carbonylierende Alkinylierung; eine Vierkomponenten‐Pyrimidin‐Synthese von Karpov, Alexei S., Merkul, Eugen, Rominger, Frank, Müller, Thomas J. J.

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Straightforward Novel One-Pot Enaminone and Pyrimidine Syntheses by Coupling-Addition-Cyclocondensation Sequences von Karpov, Alexei S., Mueller, Thomas J. J.

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New Entry to a Three-Component Pyrimidine Synthesis by TMS-Ynones via Sonogashira Coupling von Karpov, Alexei S., Mueller, Thomas J. J.

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A Novel One-Pot Four-Component Access to Tetrahydro-β-carbolines by a Coupling-Amination-Aza-Annulation-Pictet-Spengler Sequence (CAAPS) von Karpov, Alexei S., Oeser, Thomas, Mueller, Thomas J. J.

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One-Pot Three-Component Synthesis of 3-Halofurans and 3-Chloro-4-iodofurans von Karpov, Alexei S., Merkul, Eugen, Oeser, Thomas, Mueller, Thomas J. J.

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Facile One-Pot Coupling-Aminovinylation Approach to Push-Pull Chromophores: Alkyne Activation by Sonogashira Coupling von Karpov, Alexei S., Rominger, Frank, Mueller, Thomas J. J.

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