The Chemical Synthesis of Insulin: An Enduring Challenge von Karas, John A, Wade, John D, Hossain, Mohammed Akhter

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Total Chemical Synthesis of a Nonfibrillating Human Glycoinsulin von Hossain, Mohammed Akhter, Okamoto, Ryo, Karas, John A, Praveen, Praveen, Liu, Mengjie, Forbes, Briony E, Wade, John D, Kajihara, Yasuhiro

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The Antimicrobial Activity of Cannabinoids von Karas, John A., Wong, Labell J. M., Paulin, Olivia K. A., Mazeh, Amna C., Hussein, Maytham H., Li, Jian, Velkov, Tony

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A One-Pot Chemically Cleavable Bis-Linker Tether Strategy for the Synthesis of Heterodimeric Peptides von Patil, Nitin A., Tailhades, Julien, Karas, John A., Separovic, Frances, Wade, John D., Hossain, Mohammed Akhter

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2-Nitroveratryl as a Photocleavable Thiol-Protecting Group for Directed Disulfide Bond Formation in the Chemical Synthesis of Insulin von Karas, John A., Scanlon, Denis B., Forbes, Briony E., Vetter, Irina, Lewis, Richard J., Gardiner, James, Separovic, Frances, Wade, John D., Hossain, Mohammed A.

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The Killing Mechanism of Teixobactin against Methicillin-Resistant Staphylococcus aureus: an Untargeted Metabolomics Study von Hussein, Maytham, Karas, John A, Schneider-Futschik, Elena K, Chen, Fan, Swarbrick, James, Paulin, Olivia K A, Hoyer, Daniel, Baker, Mark, Zhu, Yan, Li, Jian, Velkov, Tony

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Chemical Synthesis and Characterization of an Equinatoxin II(1-85) Analogue von Karas, John A, Sani, Marc-Antoine, Separovic, Frances

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Modular Synthesis of Trifunctional Peptide-oligonucleotide Conjugates via Native Chemical Ligation von Dastpeyman, Mohadeseh, Karas, John A, Amin, Azin, Turner, Bradley J, Shabanpoor, Fazel

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Versatile New Bis(thiosemicarbazone) Bifunctional Chelators: Synthesis, Conjugation to Bombesin(7−14)-NH2, and Copper-64 Radiolabeling von Paterson, Brett M, Karas, John A, Scanlon, Denis B, White, Jonathan M, Donnelly, Paul S

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The effect of substance P and its common in vivo‐formed metabolites on MRGPRX2 and human mast cell activation von Hsin, Lin, Fernandopulle, Nithya A., Ding, Jie, Lumb, Chris, Veldhuis, Nicholas, Karas, John A., Northfield, Susan E., Mackay, Graham A.

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Modulation of Conotoxin Structure and Function Is Achieved through a Multienzyme Complex in the Venom Glands of Cone Snails von Safavi-Hemami, Helena, Gorasia, Dhana G., Steiner, Andrew M., Williamson, Nicholas A., Karas, John A., Gajewiak, Joanna, Olivera, Baldomero M., Bulaj, Grzegorz, Purcell, Anthony W.

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Rapid Optimization of a Peptide Inhibitor of Malaria Parasite Invasion by Comprehensive N-Methyl Scanning von Harris, Karen S., Casey, Joanne L., Coley, Andrew M., Karas, John A., Sabo, Jennifer K., Tan, Yen Yee, Dolezal, Olan, Norton, Raymond S., Hughes, Andrew B., Scanlon, Denis, Foley, Michael

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Structure of micelle bound cationic peptides by NMR spectroscopy using a lanthanide shift reagent von Swarbrick, James D, Karas, John A, Li, Jian, Velkov, Tony

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1,3-Dichloroacetone: A Robust Reagent for Preparing Bicyclic Peptides von Lin, Qingqing, Hopper, Denham, Zhang, Haoyue, Sfyris Qoon, Jordan, Shen, Zihan, Karas, John A, Hughes, Richard A, Northfield, Susan E

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Thiol-Cyanobenzothiazole Ligation for the Efficient Preparation of Peptide–PNA Conjugates von Patil, Nitin A, Karas, John A, Turner, Bradley J, Shabanpoor, Fazel

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Semisynthesis of A6–A11 lactam insulin von Xu, Rong, Jap, Edwina, Gubbins, Ben, Hagemeyer, Christoph E., Karas, John A.

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Structure–Activity Relationships of Daptomycin Lipopeptides von Karas, John A, Carter, Glen P, Howden, Benjamin P, Turner, Adrianna M, Paulin, Olivia K. A, Swarbrick, James D, Baker, Mark. A, Li, Jian, Velkov, Tony

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Differential MRGPRX2-dependent activation of human mast cells by polymyxins and octapeptins von Ding, Jie, Zhang, Stephanie S., Fernandopulle, Nithya A., Karas, John A., Li, Jian, Ziogas, James, Velkov, Tony, Mackay, Graham A.

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Endosomal escape cell-penetrating peptides significantly enhance pharmacological effectiveness and CNS activity of systemically administered antisense oligonucleotides von Dastpeyman, Mohadeseh, Sharifi, Ramin, Amin, Azin, Karas, John A., Cuic, Brittany, Pan, Yijun, Nicolazzo, Joseph A., Turner, Bradley J., Shabanpoor, Fazel

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An Engineered Nanosugar Enables Rapid and Sustained Glucose‐Responsive Insulin Delivery in Diabetic Mice von Xu, Rong, Bhangu, Sukhvir Kaur, Sourris, Karly C., Vanni, Domitilla, Sani, Marc‐Antoine, Karas, John A., Alt, Karen, Niego, Be'eri, Ale, Anukreity, Besford, Quinn A., Dyett, Brendan, Patrick, Joshua, Carmichael, Irena, Shaw, Jonathan E., Caruso, Frank, Cooper, Mark E., Hagemeyer, Christoph E., Cavalieri, Francesca

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