Epigenetics and beyond: targeting writers of protein lysine methylation to treat disease von Bhat, Kamakoti P., Ümit Kaniskan, H., Jin, Jian, Gozani, Or

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Inhibitors of Protein Methyltransferases and Demethylases von Kaniskan, H. Ümit, Martini, Michael L, Jin, Jian

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Advancing targeted protein degradation for cancer therapy von Dale, Brandon, Cheng, Meng, Park, Kwang-Su, Kaniskan, H. Ümit, Xiong, Yue, Jin, Jian

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TF-PROTACs Enable Targeted Degradation of Transcription Factors von Liu, Jing, Chen, He, Kaniskan, H. Ümit, Xie, Ling, Chen, Xian, Jin, Jian, Wei, Wenyi

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Cancer Selective Target Degradation by Folate-Caged PROTACs von Liu, Jing, Chen, He, Liu, Yi, Shen, Yudao, Meng, Fanye, Kaniskan, H. Ümit, Jin, Jian, Wei, Wenyi

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Artificial intelligence and machine learning‐aided drug discovery in central nervous system diseases: State‐of‐the‐arts and future directions von Vatansever, Sezen, Schlessinger, Avner, Wacker, Daniel, Kaniskan, H. Ümit, Jin, Jian, Zhou, Ming‐Ming, Zhang, Bin

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An MDM2 degrader for treatment of acute leukemias von Marcellino, Bridget K., Yang, Xiaobao, Ümit Kaniskan, H., Brady, Claudia, Chen, He, Chen, Karie, Qiu, Xing, Clementelli, Cara, Herschbein, Lauren, Li, Zhijun, Elghaity-Beckley, Sebastian, Arandela, Joann, Kelly, Brianna, Hoffman, Ronald, Liu, Jing, Xiong, Yue, Jin, Jian, Shih, Alan H.

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Selective Inhibitors of Protein Methyltransferases von Kaniskan, H. Ümit, Konze, Kyle D, Jin, Jian

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TF-DUBTACs Stabilize Tumor Suppressor Transcription Factors von Liu, Jing, Yu, Xufen, Chen, He, Kaniskan, H. Ümit, Xie, Ling, Chen, Xian, Jin, Jian, Wei, Wenyi

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Folate-Guided Protein Degradation by Immunomodulatory Imide Drug-Based Molecular Glues and Proteolysis Targeting Chimeras von Chen, He, Liu, Jing, Kaniskan, H. Ümit, Wei, Wenyi, Jin, Jian

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Telomere Targeting Chimera Enables Targeted Destruction of Telomeric Repeat-Binding Factor Proteins von Wang, Zhen, Liu, Jing, Chen, He, Qiu, Xing, Xie, Ling, Kaniskan, H. Ümit, Chen, Xian, Jin, Jian, Wei, Wenyi

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Harnessing the E3 Ligase KEAP1 for Targeted Protein Degradation von Wei, Jieli, Meng, Fanye, Park, Kwang-Su, Yim, Hyerin, Velez, Julia, Kumar, Prashasti, Wang, Li, Xie, Ling, Chen, He, Shen, Yudao, Teichman, Emily, Li, Dongxu, Wang, Gang Greg, Chen, Xian, Kaniskan, H. Ümit, Jin, Jian

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Chemically induced degradation of epigenetic targets von Kabir, Md, Yu, Xufen, Kaniskan, H. Ümit, Jin, Jian

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Acetylation Targeting Chimera Enables Acetylation of the Tumor Suppressor p53 von Kabir, Md, Sun, Ning, Hu, Xiaoping, Martin, Tiphaine C., Yi, Jingjie, Zhong, Yue, Xiong, Yan, Kaniskan, H. Ümit, Gu, Wei, Parsons, Ramon, Jin, Jian

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Discovery of the First Lactate Dehydrogenase Proteolysis Targeting Chimera Degrader for the Treatment of Pancreatic Cancer von Sun, Ning, Kabir, Md, Lee, Youngeun, Xie, Ling, Hu, Xiaoping, Velez, Julia, Chen, Xian, Kaniskan, H. Ümit, Jin, Jian

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Recent advances in developing degraders & inhibitors of lysine methyltransferases von Velez, Julia, Kaniskan, H. Ümit, Jin, Jian

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Light-induced control of protein destruction by opto-PROTAC von Liu, Jing, Chen, He, Ma, Leina, He, Zhixiang, Wang, Dong, Liu, Yi, Lin, Qian, Zhang, Tinghu, Gray, Nathanael, Kaniskan, H Ümit, Jin, Jian, Wei, Wenyi

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Structure–Activity Relationship Studies for Enhancer of Zeste Homologue 2 (EZH2) and Enhancer of Zeste Homologue 1 (EZH1) Inhibitors von Yang, Xiaobao, Li, Fengling, Konze, Kyle D, Meslamani, Jamel, Ma, Anqi, Brown, Peter J, Zhou, Ming-Ming, Arrowsmith, Cheryl H, Kaniskan, H. Ümit, Vedadi, Masoud, Jin, Jian

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Discovery of the First-in-Class G9a/GLP PROTAC Degrader von Velez, Julia, Han, Yulin, Yim, Hyerin, Yang, Peiyi, Deng, Zhijie, Park, Kwang-su, Kabir, Md, Kaniskan, H. Ümit, Xiong, Yan, Jin, Jian

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Structurally Specific Z‑DNA Proteolysis Targeting Chimera Enables Targeted Degradation of Adenosine Deaminase Acting on RNA 1 von Wang, Zhen, Zhang, Dingpeng, Qiu, Xing, Inuzuka, Hiroyuki, Xiong, Yan, Liu, Jing, Chen, Li, Chen, He, Xie, Ling, Kaniskan, H. Ümit, Chen, Xian, Jin, Jian, Wei, Wenyi

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