Chemical Epigenetics: The Impact of Chemical and Chemical Biology Techniques on Bromodomain Target Validation von Schiedel, Matthias, Moroglu, Mustafa, Ascough, David M. H., Chamberlain, Anna E. R., Kamps, Jos J. A. G., Sekirnik, Angelina R., Conway, Stuart J.

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Chemical basis for the recognition of trimethyllysine by epigenetic reader proteins von Kamps, Jos J.A.G., Huang, Jiaxin, Poater, Jordi, Xu, Chao, Pieters, Bas J.G.E., Dong, Aiping, Min, Jinrong, Sherman, Woody, Beuming, Thijs, Matthias Bickelhaupt, F., Li, Haitao, Mecinović, Jasmin

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Bicyclic Boronate VNRX-5133 Inhibits Metallo- and Serine-β-Lactamases von Krajnc, Alen, Brem, Jürgen, Hinchliffe, Philip, Calvopiña, Karina, Panduwawala, Tharindi D, Lang, Pauline A, Kamps, Jos J. A. G, Tyrrell, Jonathan M, Widlake, Emma, Saward, Benjamin G, Walsh, Timothy R, Spencer, James, Schofield, Christopher J

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The plant cysteine oxidases from Arabidopsis thaliana are kinetically tailored to act as oxygen sensors von White, Mark D., Kamps, Jos J. A.G., East, Samuel, Taylor Kearney, Leah J., Flashman, Emily

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How formaldehyde reacts with amino acids von Kamps, Jos J. A. G., Hopkinson, Richard J., Schofield, Christopher J., Claridge, Timothy D. W.

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Roles of 2-oxoglutarate oxygenases and isopenicillin N synthase in β-lactam biosynthesis von Rabe, Patrick, Kamps, Jos J. A. G, Schofield, Christopher J, Lohans, Christopher T

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Mass Spectrometric Assays Reveal Discrepancies in Inhibition Profiles for the SARS‐CoV‐2 Papain‐Like Protease von Brewitz, Lennart, Kamps, Jos J. A. G., Lukacik, Petra, Strain‐Damerell, Claire, Zhao, Yilin, Tumber, Anthony, Malla, Tika R., Orville, Allen M., Walsh, Martin A., Schofield, Christopher J.

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The adaptability of the ion-binding site by the Ag(I)/Cu(I) periplasmic chaperone SilF von Lithgo, Ryan M, Hanževački, Marko, Harris, Gemma, Kamps, Jos J A G, Holden, Ellie, Gianga, Tiberiu-Marius, Benesch, Justin L P, Jäger, Christof M, Croft, Anna K, Hussain, Rohannah, Hobman, Jon L, Orville, Allen M, Quigley, Andrew, Carr, Stephen B, Scott, David J

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Non‐Hydrolytic β‐Lactam Antibiotic Fragmentation by l,d‐Transpeptidases and Serine β‐Lactamase Cysteine Variants von Lohans, Christopher T., Chan, H. T. Henry, Malla, Tika R., Kumar, Kiran, Kamps, Jos J. A. G., McArdle, Darius J. B., van Groesen, Emma, de Munnik, Mariska, Tooke, Catherine L., Spencer, James, Paton, Robert S., Brem, Jürgen, Schofield, Christopher J.

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Installation of Trimethyllysine Analogs on Intact Histones via Cysteine Alkylation von Pieters, Bas J. G. E, Hintzen, Jordi C. J, Grobben, Yvonne, Al Temimi, Abbas H. K, Kamps, Jos J. A. G, Mecinović, Jasmin

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F NMR studies on γ-butyrobetaine hydroxylase provide mechanistic insights and suggest a dual inhibition mode von Le niak, Robert K, Rydzik, Anna M, Kamps, Jos J. A. G, Kahn, Amjad, Claridge, Timothy D. W, Schofield, Christopher J

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Structure activity relationship studies on rhodanines and derived enethiol inhibitors of metallo-β-lactamases von Zhang, Dong, Markoulides, Marios S., Stepanovs, Dmitrijs, Rydzik, Anna M., El-Hussein, Ahmed, Bon, Corentin, Kamps, Jos J.A.G., Umland, Klaus-Daniel, Collins, Patrick M., Cahill, Samuel T., Wang, David Y., von Delft, Frank, Brem, Jürgen, McDonough, Michael A., Schofield, Christopher J.

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Cation-π Interactions Contribute to Substrate Recognition in γ-Butyrobetaine Hydroxylase Catalysis von Kamps, Jos J. A. G., Khan, Amjad, Choi, Hwanho, Lesniak, Robert K., Brem, Jürgen, Rydzik, Anna M., McDonough, Michael A., Schofield, Christopher J., Claridge, Timothy D. W., Mecinović, Jasmin

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Hydroxylamine as an oxygen nucleophile: substitution of sulfonamide by a hydroxyl group in benzothiazole-2-sulfonamides von Kamps, Jos J A G, Belle, Roman, Mecinović, Jasmin

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X-ray free-electron laser studies reveal correlated motion during isopenicillin N synthase catalysis von Rabe, Patrick, Kamps, Jos J. A. G., Sutherlin, Kyle D., Linyard, James D. S., Aller, Pierre, Pham, Cindy C., Makita, Hiroki, Clifton, Ian, McDonough, Michael A., Leissing, Thomas M., Shutin, Denis, Lang, Pauline A., Butryn, Agata, Brem, Jurgen, Gul, Sheraz, Fuller, Franklin D., Kim, In-Sik, Cheah, Mun Hon, Fransson, Thomas, Bhowmick, Asmit, Young, Iris D., O'Riordan, Lee, Brewster, Aaron S., Pettinati, Ilaria, Doyle, Margaret, Joti, Yasumasa, Owada, Shigeki, Tono, Kensuke, Batyuk, Alexander, Hunter, Mark S., Alonso-Mori, Roberto, Bergmann, Uwe, Owen, Robin L., Sauter, Nicholas K., Claridge, Timothy D. W., Robinson, Carol V., Yachandra, Vittal K., Yano, Junko, Kern, Jan F., Orville, Allen M., Schofield, Christopher J.

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Reading and erasing of the phosphonium analogue of trimethyllysine by epigenetic proteins von Belle, Roman, Kamps, Jos J. A. G., Poater, Jordi, Kumar, Kiran, Pieters, Bas J. G. E., Salah, Eidarus, Claridge, Timothy D. W., Paton, Robert S., Bickelhaupt, F. Matthias, Kawamura, Akane, Schofield, Christopher J., Mecinović, Jasmin

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Cation-[pi] Interactions Contribute to Substrate Recognition in [gamma]-Butyrobetaine Hydroxylase Catalysis von Kamps, Jos J A G, Khan, Amjad, Choi, Hwanho, Lesniak, Robert K, Brem, Jurgen, Rydzik, Anna M, McDonough, Michael A, Schofield, Christopher J, Claridge, Timothy D W, Mecinovic, Jasmin

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Mechanism of biomolecular recognition of trimethyllysine by the fluorinated aromatic cage of KDM5A PHD3 finger von Pieters, Bas J. G. E., Wuts, Maud H. M., Poater, Jordi, Kumar, Kiran, White, Paul B., Kamps, Jos J. A. G., Sherman, Woody, Pruijn, Ger J. M., Paton, Robert S., Beuming, Thijs, Bickelhaupt, F. Matthias, Mecinović, Jasmin

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