Identification of Diarylurea Inhibitors of the Cardiac-Specific Kinase TNNI3K by Designing Selectivity Against VEGFR2, p38α, and B‑Raf von Patterson, Jaclyn R, Graves, Alan P, Stoy, Patrick, Cheung, Mui, Desai, Tina A, Fries, Harvey, Gatto, Gregory J, Holt, Dennis A, Shewchuk, Lisa, Totoritis, Rachel, Wang, Liping, Kallander, Lara S

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4,6-Diaminopyrimidines as Highly Preferred Troponin I‑Interacting Kinase (TNNI3K) Inhibitors von Philp, Joanne, Lawhorn, Brian G, Graves, Alan P, Shewchuk, Lisa, Rivera, Katrina L, Jolivette, Larry J, Holt, Dennis A, Gatto, Gregory J, Kallander, Lara S

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Substituent Effects on Drug–Receptor H‑bond Interactions: Correlations Useful for the Design of Kinase Inhibitors von Lawhorn, Brian G, Philp, Joanne, Graves, Alan P, Holt, Dennis A, Gatto, Gregory J, Kallander, Lara S

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Identification of Purines and 7‑Deazapurines as Potent and Selective Type I Inhibitors of Troponin I‑Interacting Kinase (TNNI3K) von Lawhorn, Brian G, Philp, Joanne, Zhao, Yongdong, Louer, Christopher, Hammond, Marlys, Cheung, Mui, Fries, Harvey, Graves, Alan P, Shewchuk, Lisa, Wang, Liping, Cottom, Joshua E, Qi, Hongwei, Zhao, Huizhen, Totoritis, Rachel, Zhang, Guofeng, Schwartz, Benjamin, Li, Hu, Sweitzer, Sharon, Holt, Dennis A, Gatto, Gregory J, Kallander, Lara S

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In Vivo Half-Life Extension of BMP1/TLL Metalloproteinase Inhibitors Using Small-Molecule Human Serum Albumin Binders von Vantourout, Julien C, Mason, Andrew M, Yuen, Josephine, Simpson, Graham L, Evindar, Ghotas, Kuai, Letian, Hobbs, Michael, Edgar, Emma, Needle, Saul, Bai, Xiaopeng, Wilson, Steve, Scott-Stevens, Paul, Traylen, William, Lambert, Kim, Young, Neil, Bunally, Shenaz, Summerfield, Scott G, Snell, Richard, Lad, Rakesh, Shi, Eric, Skinner, Steven, Shewchuk, Lisa, Watson, Allan J.B, Chung, Chun-wa, Pal, Sandeep, Holt, Dennis A, Kallander, Lara S, Prendergast, Joanne, Rivera, Katrina, Washburn, David G, Harpel, Mark R, Arico-Muendel, Christopher, Isidro-Llobet, Albert

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GSK114: A selective inhibitor for elucidating the biological role of TNNI3K von Lawhorn, Brian G., Philp, Joanne, Graves, Alan P., Shewchuk, Lisa, Holt, Dennis A., Gatto, Gregory J., Kallander, Lara S.

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Empowering Women in Organic Chemistry (EWOC) at Five Years: Giving Back and Getting Back von Cantor, Elinor H, Faul, Margaret M, Huryn, Donna M, Kallander, Lara, Ruck, Rebecca T, Watson, Mary P

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Empowering Women in Organic Chemistry (EWOC) at Five Years: Giving Back and Getting Back von Cantor, Elinor H., Faul, Margaret M., Huryn, Donna M., Kallander, Lara, Ruck, Rebecca T., Watson, Mary P.

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Reverse Hydroxamate Inhibitors of Bone Morphogenetic Protein 1 von Kallander, Lara S., Washburn, David, Hilfiker, Mark A., Eidam, Hilary Schenck, Lawhorn, Brian G., Prendergast, Joanne, Fox, Ryan, Dowdell, Sarah, Manns, Sharada, Hoang, Tram, Zhao, Steve, Ye, Guosen, Hammond, Marlys, Holt, Dennis A., Roethke, Theresa, Hong, Xuan, Reid, Robert A., Gampe, Robert, Zhang, Hong, Diaz, Elsie, Rendina, Alan R., Quinn, Amy M., Willette, Bob

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4-Aryl-1,2,3-triazole:  A Novel Template for a Reversible Methionine Aminopeptidase 2 Inhibitor, Optimized To Inhibit Angiogenesis in Vivo von Kallander, Lara S, Lu, Qing, Chen, Wenfang, Tomaszek, Thaddeus, Yang, Guang, Tew, David, Meek, Thomas D, Hofmann, Glenn A, Schulz-Pritchard, Christina K, Smith, Ward W, Janson, Cheryl A, Ryan, M. Dominic, Zhang, Gui-Feng, Johanson, Kyung O, Kirkpatrick, Robert B, Ho, Thau F, Fisher, Paul W, Mattern, Michael R, Johnson, Randall K, Hansbury, Michael J, Winkler, James D, Ward, Keith W, Veber, Daniel F, Thompson, Scott K

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Discovery of renin inhibitors containing a simple aspartate binding moiety that imparts reduced P450 inhibition von Lawhorn, Brian G., Tran, Tritin, Hong, Victor S., Morgan, Lisa A., Le, BaoChau T., Harpel, Mark R., Jolivette, Larry, Diaz, Elsie, Schwartz, Benjamin, Gross, Jeffrey W., Tomaszek, Thaddeus, Semus, Simon, Concha, Nestor, Smallwood, Angela, Holt, Dennis A., Kallander, Lara S.

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Empowering Women in Organic Chemistry (EWOC) at Five Years: Giving Back and Getting Back von Cantor, Elinor H., Faul, Margaret M., Huryn, Donna M., Kallander, Lara, Ruck, Rebecca T., Watson, Mary P.

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Empowering Women in Organic Chemistry (EWOC) at Five Years: Giving Back and Getting Back von Cantor, Elinor H., Faul, Margaret M., Huryn, Donna M., Kallander, Lara, Ruck, Rebecca T., Watson, Mary P.

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Empowering Women in Organic Chemistry (EWOC) at Five Years: Giving Back and Getting Back von Cantor, Elinor H., Faul, Margaret M., Huryn, Donna M., Kallander, Lara, Ruck, Rebecca T., Watson, Mary P.

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A Versatile Enantioselective Strategy Toward l-C-Nucleosides:  A Total Synthesis of l-Showdomycin von Trost, Barry M, Kallander, Lara S

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The discovery of tertiary-amine LXR agonists with potent cholesterol efflux activity in macrophages von Marino, Joseph P., Kallander, Lara S., Ma, Chun, Oh, Hye-Ja, Lee, Dennis, Gaitanopoulos, Dimitri E., Krawiec, John A., Parks, Derek J., Webb, Christine L., Ziegler, Kelly, Jaye, Michael, Thompson, Scott K.

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Improving the developability profile of pyrrolidine progesterone receptor partial agonists von Kallander, Lara S., Washburn, David G., Hoang, Tram H., Frazee, James S., Stoy, Patrick, Johnson, Latisha, Lu, Qing, Hammond, Marlys, Barton, Linda S., Patterson, Jaclyn R., Azzarano, Leonard M., Nagilla, Rakesh, Madauss, Kevin P., Williams, Shawn P., Stewart, Eugene L., Duraiswami, Chaya, Grygielko, Eugene T., Xu, Xiaoping, Laping, Nicholas J., Bray, Jeffrey D., Thompson, Scott K.

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Empowering Women in Organic Chemistry (EWOC) at Five Years: Giving Back and Getting Back von Cantor, Elinor H., Faul, Margaret M., Huryn, Donna M., Kallander, Lara, Ruck, Rebecca T., Watson, Mary P.

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Empowering Women in Organic Chemistry (EWOC) at Five Years: Giving Back and Getting Back von Cantor, Elinor H., Faul, Margaret M., Huryn, Donna M., Kallander, Lara, Ruck, Rebecca T., Watson, Mary P.

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Empowering Women in Organic Chemistry (EWOC) at Five Years: Giving Back and Getting Back von Cantor, Elinor H., Faul, Margaret M., Huryn, Donna M., Kallander, Lara, Ruck, Rebecca T., Watson, Mary P.

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