PVC Formulation of Anastrepha suspensa Pheromones Suitable for Field Studies von Kuzmich, Daniel, Kawagoe, Zachary A., Walse, Spencer S.

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A GPBAR1 (TGR5) small molecule agonist shows specific inhibitory effects on myeloid cell activation in vitro and reduces experimental autoimmune encephalitis (EAE) in vivo von Lewis, Nuruddeen D, Patnaude, Lori A, Pelletier, Josephine, Souza, Donald J, Lukas, Susan M, King, F James, Hill, Jonathan D, Stefanopoulos, Dimitria E, Ryan, Kelli, Desai, Sudha, Skow, Donna, Kauschke, Stefan G, Broermann, Andre, Kuzmich, Daniel, Harcken, Christian, Hickey, Eugene R, Modis, Louise K

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Nonsteroidal Dissociated Glucocorticoid Agonists Containing Azaindoles as Steroid A-Ring Mimetics von Riether, Doris, Harcken, Christian, Razavi, Hossein, Kuzmich, Daniel, Gilmore, Thomas, Bentzien, Jörg, Pack, Edward J, Souza, Donald, Nelson, Richard M, Kukulka, Alison, Fadra, Tazmeen N, Zuvela-Jelaska, Ljiljana, Pelletier, Josephine, Dinallo, Roger, Panzenbeck, Mark, Torcellini, Carol, Nabozny, Gerald H, Thomson, David S

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CCR1 plays a critical role in modulating pain through hematopoietic and non-hematopoietic cells von Lewis, Nuruddeen D, Muthukumarana, Akalushi, Fogal, Steven E, Corradini, Laura, Stefanopoulos, Dimitria E, Adusumalli, Prathima, Pelletier, Josephine, Panzenbeck, Mark, Berg, Karen, Canfield, Melissa, Cook, Brian N, Razavi, Hossein, Kuzmich, Daniel, Anderson, Shawn, Allard, Devan, Harrison, Paul, Grimaldi, Christine, Souza, Donald, Harcken, Christian, Fryer, Ryan M, Modis, Louise K, Brown, Maryanne L

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Trifluoromethyl group as a pharmacophore : Effect of replacing a CF3 group on binding and agonist activity of a glucocorticoid receptor ligand von BETAGERI, Raj, YAN ZHANG, PAW, Zofia, SHIH, Daw-Tsun, SHIH, Cheng-Kon, ZUVELA-JELASKA, Ljiljana, NABOZNY, Gerald, THOMSON, David S, ZINDELL, Renee M, KUZMICH, Daniel, KIRRANE, Thomas M, BENTZIEN, Jörg, CARDOZO, Mario, CAPOLINO, Alison J, FADRA, Tazmeen N, NELSON, Richard M

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Non-steroidal dissociated glucocorticoid agonists: indoles as A-ring mimetics and function-regulating pharmacophores von Betageri, Raj, Gilmore, Thomas, Kuzmich, Daniel, Kirrane, Thomas M., Bentzien, Jörg, Wiedenmayer, Dieter, Bekkali, Younes, Regan, John, Berry, Angela, Latli, Bachir, Kukulka, Alison J., Fadra, Tazmeen N., Nelson, Richard M., Goldrick, Susan, Zuvela-Jelaska, Ljiljana, Souza, Don, Pelletier, Josephine, Dinallo, Roger, Panzenbeck, Mark, Torcellini, Carol, Lee, Heewon, Pack, Edward, Harcken, Christian, Nabozny, Gerald, Thomson, David S.

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The timing of diverse external stakeholder involvement during interfirm open innovation: The effects on new product speed to market and product lifespan von Fisher, Gregory J., John-Mariadoss, Babu, Kuzmich, Daniel, Qualls, William J.

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Free Radical Cyclizations in Alkaloid Total Synthesis:  (±)-21-Oxogelsemine and (±)-Gelsemine von Atarashi, Shogo, Choi, Joong-Kwon, Ha, Deok-Chan, Hart, David J, Kuzmich, Daniel, Lee, Chih-Shone, Ramesh, Subban, Wu, Shung C

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Identification of novel azaindazole CCR1 antagonist clinical candidates von Harcken, Christian, Kuzmich, Daniel, Cook, Brain, Mao, Can, Disalvo, Darren, Razavi, Hossein, Swinamer, Alan, Liu, Pingrong, Zhang, Qiang, Kukulka, Alison, Skow, Donna, Patel, Mita, Patel, Monica, Fletcher, Kimberly, Sherry, Tara, Joseph, David, Smith, Dustin, Canfield, Melissa, Souza, Donald, Bogdanffy, Matthew, Berg, Karen, Brown, Maryanne

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Identification of Highly Efficacious Glucocorticoid Receptor Agonists with a Potential for Reduced Clinical Bone Side Effects von Harcken, Christian, Riether, Doris, Kuzmich, Daniel, Liu, Pingrong, Betageri, Raj, Ralph, Mark, Emmanuel, Michel, Reeves, Jonathan T, Berry, Angela, Souza, Donald, Nelson, Richard M, Kukulka, Alison, Fadra, Tazmeen N, Zuvela-Jelaska, Ljiljana, Dinallo, Roger, Bentzien, Jörg, Nabozny, Gerald H, Thomson, David S

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Development of an Enantioselective Hydrogenation Route to (S)‑1-(2-(Methylsulfonyl)pyridin-4-yl)propan-1-amine von Reeves, Jonathan T, Tan, Zhulin, Reeves, Diana C, Song, Jinhua J, Han, Zhengxu S, Xu, Yibo, Tang, Wenjun, Yang, Bing-Shiou, Razavi, Hossein, Harcken, Christian, Kuzmich, Daniel, Mahaney, Paige E, Lee, Heewon, Busacca, Carl A, Senanayake, Chris H

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Substituted phenyl as a steroid A-ring mimetic: Providing agonist activity to a class of arylsulfonamide nonsteroidal glucocorticoid ligands von DiSalvo, Darren, Kuzmich, Daniel, Bentzien, Jörg, Regan, John, Kukulka, Alison, Fadra-Khan, Tazmeen, Nelson, Richard, Harcken, Christian, Thomson, David, Nabozny, Gerald

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Function-regulating pharmacophores in a sulfonamide class of glucocorticoid receptor agonists von Kuzmich, Daniel, Bentzien, Jörg, Betageri, Raj, DiSalvo, Darren, Fadra-Khan, Tazmeen, Harcken, Christian, Kukulka, Alison, Nabozny, Gerald, Nelson, Richard, Pack, Edward, Souza, Donald, Thomson, David

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Synthesis of 2-Aryl-1-hydroxyazaindolesand 2-Arylazaindoles via Oxidation of o- Hydroxyaminostyrylpyridines von Kuzmich, Daniel, Mulrooney, Carol

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Late-stage optimization of a tercyclic class of S1P 3 -sparing, S1P 1 receptor agonists von Horan, Joshua C., Kuzmich, Daniel, Liu, Pingrong, DiSalvo, Darren, Lord, John, Mao, Can, Hopkins, Tamara D., Yu, Hui, Harcken, Christian, Betageri, Raj, Hill-Drzewi, Melissa, Patenaude, Lori, Patel, Monica, Fletcher, Kimberly, Terenzzio, Donna, Linehan, Brian, Xia, Heather, Patel, Mita, Studwell, Debbie, Miller, Craig, Hickey, Eugene, Levin, Jeremy I., Smith, Dustin, Kemper, Raymond A., Modis, Louise K., Bannen, Lynne C., Chan, Diva S., Mac, Morrison B., Ng, Stephanie, Wang, Yong, Xu, Wei, Lemieux, René M.

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A GPBAR1 von Lewis, Nuruddeen D, Patnaude, Lori A, Pelletier, Josephine, Souza, Donald J, Lukas, Susan M, King, F. James, Hill, Jonathan D, Stefanopoulos, Dimitria E, Ryan, Kelli, Desai, Sudha, Skow, Donna, Kauschke, Stefan G, Broermann, Andre, Kuzmich, Daniel, Harcken, Christian, Hickey, Eugene R, Modis, Louise K

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A GPBAR1 In Vivo von Lewis, Nuruddeen D, Patnaude, Lori A, Pelletier, Josephine, Souza, Donald J, Lukas, Susan M, King, F. James, Hill, Jonathan D, Stefanopoulos, Dimitria E, Ryan, Kelli, Desai, Sudha, Skow, Donna, Kauschke, Stefan G, Broermann, Andre, Kuzmich, Daniel, Harcken, Christian, Hickey, Eugene R, Modis, Louise K

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Trifluoromethyl group as a pharmacophore: Effect of replacing a CF 3 group on binding and agonist activity of a glucocorticoid receptor ligand von Betageri, Raj, Zhang, Yan, Zindell, Renee M., Kuzmich, Daniel, Kirrane, Thomas M., Bentzien, Jörg, Cardozo, Mario, Capolino, Alison J., Fadra, Tazmeen N., Nelson, Richard M., Paw, Zofia, Shih, Daw-Tsun, Shih, Cheng-Kon, Zuvela-Jelaska, Ljiljana, Nabozny, Gerald, Thomson, David S.

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Late-stage optimization of a tercyclic class of S1P3-sparing, S1P1 receptor agonists von Horan, Joshua C., Kuzmich, Daniel, Liu, Pingrong, DiSalvo, Darren, Lord, John, Mao, Can, Hopkins, Tamara D., Yu, Hui, Harcken, Christian, Betageri, Raj, Hill-Drzewi, Melissa, Patenaude, Lori, Patel, Monica, Fletcher, Kimberly, Terenzzio, Donna, Linehan, Brian, Xia, Heather, Patel, Mita, Studwell, Debbie, Miller, Craig, Hickey, Eugene, Levin, Jeremy I., Smith, Dustin, Kemper, Raymond A., Modis, Louise K., Bannen, Lynne C., Chan, Diva S., Mac, Morrison B., Ng, Stephanie, Wang, Yong, Xu, Wei, Lemieux, René M.

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G Protein–Coupled Bile Acid Receptor 1 Stimulation Mediates Arterial Vasodilation through a K Ca 1.1 (BK Ca )–Dependent Mechanism von Fryer, Ryan M., Ng, Khing Jow, Nodop Mazurek, Suzanne G., Patnaude, Lori, Skow, Donna J., Muthukumarana, Akalushi, Gilpin, Kyle E., Dinallo, Roger M., Kuzmich, Daniel, Lord, John, Sanyal, Sulagna, Yu, Hui, Harcken, Christian, Cerny, Matthew A., Hickey, Eugene R., Modis, Louise K.

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