Bioisosteric approach to the discovery of imidazo[1,2-a]pyrazines as potent Aurora kinase inhibitors von Meng, Zhaoyang, Kulkarni, Bheemashankar A., Kerekes, Angela D., Mandal, Amit K., Esposite, Sara J., Belanger, David B., Reddy, Panduranga Adulla, Basso, Andrea D., Tevar, Seema, Gray, Kimberly, Jones, Jennifer, Smith, Elizabeth B., Doll, Ronald J., Siddiqui, M. Arshad

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Exploring Chemical Diversity of Epoxyquinoid Natural Products:  Synthesis and Biological Activity of (−)-Jesterone and Related Molecules von Hu, Yongbo, Li, Chaomin, Kulkarni, Bheemashankar A, Strobel, Gary, Lobkovsky, Emil, Torczynski, Richard M, Porco, John A

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Solution-phase combinatorial synthesis of 4-hydroxyquinolin-2(1H)-ones von Kulkarni, Bheemashankar A., Ganesan, A.

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Ion-Exchange Resins for Combinatorial Synthesis: 2,4-Pyrrolidinediones by Dieckmann Condensation von Kulkarni, Bheemashankar A., Ganesan, Arasu

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A New Series of Orally Bioavailable Chemokine Receptor 9 (CCR9) Antagonists; Possible Agents for the Treatment of Inflammatory Bowel Disease von Kalindjian, S. Barret, Kadnur, Sanjay V, Hewson, Christopher A, Venkateshappa, Chandregowda, Juluri, Suresh, Kristam, Rajendra, Kulkarni, Bheemashankar, Mohammed, Zainuddin, Saxena, Rohit, Viswanadhan, Vellarkad N, Aiyar, Jayashree, McVey, Donna

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Discovery and pharmacological evaluation of indole derivatives as potent and selective RORγt inverse agonist for multiple autoimmune conditions von Shaikh, Nadim S., Iyer, Jitesh P., Munot, Yogesh S., Mukhopadhyay, Partha P., Raje, Amol A., Nagaraj, Ranganayaki, Jamdar, Vijay, Gavhane, Ravindra, Lohote, Mahendra, Sherkar, Prasad, Bala, Madhu, Petla, Rajkanth, Meru, Ashwinkumar, Umrani, Dhananjay, Rouduri, Sreekanth, Joshi, Sachin, Reddy, Satyanarayan, Kandikere, Vishwottam, Bhuniya, Debnath, Kulkarni, Bheemashankar, Mookhtiar, Kasim A.

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Discovery and evaluation of 1H-pyrrolo[2,3-b]pyridine based selective and reversible small molecule BTK inhibitors for the treatment of rheumatoid arthritis von Thakkar, Mahesh, Bhuniya, Debnath, Kaduskar, Rahul, Mengawade, Tanaji, Naik, Keshav, Salunkhe, Videsh, Bhalerao, Amit, Kurhade, Santosh, Mavinahalli, Jagadeesh, Jain, Vaibhav, Petla, Rajkanth, Avaragolla, Satheesh, Ray, Swagatam, Rouduri, Sreekanth, Dhanave, Avinash, De, Siddhartha, Pathade, Vishal, Tambe, Ashwini, Raje, Amol A., Madgula, Vamsi, Joshi, Sachin, Nadeem, Ahmed, bala, Madhu, Umrani, Dhananjay, Hariharan, Narayanan, Kulkarni, Bheemashankar, Mookhtiar, Kasim A.

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Discovery and optimization of N-acyl and N-aroylpyrazolines as B-Raf kinase inhibitors von Blackburn, Christopher, Duffey, Matthew O., Gould, Alexandra E., Kulkarni, Bheemashankar, Liu, Jane X., Menon, Saurabh, Nagayoshi, Masayuki, Vos, Tricia J., Williams, Juliet

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Discovery and evaluation of 1 H -pyrrolo[2,3- b ]pyridine based selective and reversible small molecule BTK inhibitors for the treatment of rheumatoid arthritis von Thakkar, Mahesh, Bhuniya, Debnath, Kaduskar, Rahul, Mengawade, Tanaji, Naik, Keshav, Salunkhe, Videsh, Bhalerao, Amit, Kurhade, Santosh, Mavinahalli, Jagadeesh, Jain, Vaibhav, Petla, Rajkanth, Avaragolla, Satheesh, Ray, Swagatam, Rouduri, Sreekanth, Dhanave, Avinash, De, Siddhartha, Pathade, Vishal, Tambe, Ashwini, Raje, Amol A., Madgula, Vamsi, Joshi, Sachin, Nadeem, Ahmed, bala, Madhu, Umrani, Dhananjay, Hariharan, Narayanan, Kulkarni, Bheemashankar, Mookhtiar, Kasim A.

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A selenide linker for "traceless" solid-phase organic synthesis von Li, Zhengong, Kulkarni, Bheemashankar A., Ganesan, A.

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Discovery of a Potent and Orally Bioavailable Benzolactam-Derived Inhibitor of Polo-Like Kinase 1 (MLN0905) von Duffey, Matthew O, Vos, Tricia J, Adams, Ruth, Alley, Jennifer, Anthony, Justin, Barrett, Cynthia, Bharathan, Indu, Bowman, Douglas, Bump, Nancy J, Chau, Ryan, Cullis, Courtney, Driscoll, Denise L, Elder, Amy, Forsyth, Nancy, Frazer, Jonathan, Guo, Jianping, Guo, Luyi, Hyer, Marc L, Janowick, David, Kulkarni, Bheemashankar, Lai, Su-Jen, Lasky, Kerri, Li, Gang, Li, Jing, Liao, Debra, Little, Jeremy, Peng, Bo, Qian, Mark G, Reynolds, Dominic J, Rezaei, Mansoureh, Scott, Margaret Porter, Sells, Todd B, Shinde, Vaishali, Shi, Qiuju Judy, Sintchak, Michael D, Soucy, Francois, Sprott, Kevin T, Stroud, Stephen G, Nestor, Michelle, Visiers, Irache, Weatherhead, Gabriel, Ye, Yingchun, D’Amore, Natalie

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Design and Optimization of Potent and Orally Bioavailable Tetrahydronaphthalene Raf Inhibitors von Gould, Alexandra E, Adams, Ruth, Adhikari, Sharmila, Aertgeerts, Kathleen, Afroze, Roushan, Blackburn, Christopher, Calderwood, Emily F, Chau, Ryan, Chouitar, Jouhara, Duffey, Matthew O, England, Dylan B, Farrer, Cheryl, Forsyth, Nancy, Garcia, Khristofer, Gaulin, Jeffery, Greenspan, Paul D, Guo, Ribo, Harrison, Sean J, Huang, Shih-Chung, Iartchouk, Natalia, Janowick, Dave, Kim, Mi-Sook, Kulkarni, Bheemashankar, Langston, Steven P, Liu, Jane X, Ma, Li-Ting, Menon, Saurabh, Mizutani, Hirotake, Paske, Erin, Renou, Christelle C, Rezaei, Mansoureh, Rowland, R. Scott, Sintchak, Michael D, Smith, Michael D, Stroud, Stephen G, Tregay, Ming, Tian, Yuan, Veiby, Ole P, Vos, Tricia J, Vyskocil, Stepan, Williams, Juliet, Xu, Tianlin, Yang, Johnny J, Yano, Jason, Zeng, Hongbo, Zhang, Dong Mei, Zhang, Qin, Galvin, Katherine M

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Synthesis of racemic and each enantiomer of 3-methylnonacosanol, a new plant growth regulator from Lowsonia inermis von Kulkarni, Bheemashankar A, Sankaranarayanan, Sivaraman, Subbaraman, Ayalur S, Chattopadhyay, Subrata

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Discovery and optimization of pyrazoline compounds as B-Raf inhibitors von Duffey, Matthew O., Adams, Ruth, Blackburn, Christopher, Chau, Ryan W., Chen, Susan, Galvin, Katherine M., Garcia, Khristofer, Gould, Alexandra E., Greenspan, Paul D., Harrison, Sean, Huang, Shih-Chung, Kim, Mi-Sook, Kulkarni, Bheemashankar, Langston, Steven, Liu, Jane X., Ma, Li-Ting, Menon, Saurabh, Nagayoshi, Masayuki, Rowland, R. Scott, Vos, Tricia J., Xu, Tianlin, Yang, Johnny J., Yu, Shaoxia, Zhang, Qin

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A solid-phase equivalent of van Leusen's TosMIC, and its application in oxazole synthesis von Kulkarni, Bheemashankar A., Ganesan, A.

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Solution-phase parallel oxazole synthesis with TosMIC von Kulkarni, Bheemashankar A., Ganesan, A.

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A Facile Synthesis of (10Z,15Z)-Eicosa-10,15-dienoic Acid, a Marine Natural Product von Kulkarni, Bheemashankar A, Chattopadhyay, Angshuman, Mamdapur, Vasant R

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Synthesis of the Marine Compound (2R,5Z,9Z)-2-Methoxyhexacosa-5,9-dienoic Acid via a Lipase-Catalyzed Resolution and a Novel O-Alkylation Protocol von Kulkarni, Bheemashankar A., Sharma, Anubha, Gamre, Sunita, Chattopadhyay, Subrata

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Process for preparation of patiromer von Kulkarni, Bheemashankar, Pavaskar, Sarita Mohan, Anand, Sivadas

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Solid-phase synthesis of tetramic acids von Kulkarni, Bheemashankar A., Ganesan, A.

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