Sulfonimidamides in Medicinal and Agricultural Chemistry von Chinthakindi, Praveen K., Naicker, Tricia, Thota, Niranjan, Govender, Thavendran, Kruger, Hendrik G., Arvidsson, Per I.

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Safety and pharmacodynamics of dalazatide, a Kv1.3 channel inhibitor, in the treatment of plaque psoriasis: A randomized phase 1b trial von Tarcha, Eric J, Olsen, Chelsea M, Probst, Peter, Peckham, David, Muñoz-Elías, Ernesto J, Kruger, James G, Iadonato, Shawn P

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EZH2 Is Required for Germinal Center Formation and Somatic EZH2 Mutations Promote Lymphoid Transformation von Béguelin, Wendy, Popovic, Relja, Teater, Matt, Jiang, Yanwen, Bunting, Karen L., Rosen, Monica, Shen, Hao, Yang, Shao Ning, Wang, Ling, Ezponda, Teresa, Martinez-Garcia, Eva, Zhang, Haikuo, Zheng, Yupeng, Verma, Sharad K., McCabe, Michael T., Ott, Heidi M., Van Aller, Glenn S., Kruger, Ryan G., Liu, Yan, McHugh, Charles F., Scott, David W., Chung, Young Rock, Kelleher, Neil, Shaknovich, Rita, Creasy, Caretha L., Gascoyne, Randy D., Wong, Kwok-Kin, Cerchietti, Leandro, Levine, Ross L., Abdel-Wahab, Omar, Licht, Jonathan D., Elemento, Olivier, Melnick, Ari M.

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A DNA Hypomethylation Signature Predicts Antitumor Activity of LSD1 Inhibitors in SCLC von Mohammad, Helai P., Smitheman, Kimberly N., Kamat, Chandrashekhar D., Soong, David, Federowicz, Kelly E., Van Aller, Glenn S., Schneck, Jess L., Carson, Jeffrey D., Liu, Yan, Butticello, Michael, Bonnette, William G., Gorman, Shelby A., Degenhardt, Yan, Bai, Yuchen, McCabe, Michael T., Pappalardi, Melissa B., Kasparec, Jiri, Tian, Xinrong, McNulty, Kenneth C., Rouse, Meagan, McDevitt, Patrick, Ho, Thau, Crouthamel, Michelle, Hart, Timothy K., Concha, Nestor O., McHugh, Charles F., Miller, William H., Dhanak, Dashyant, Tummino, Peter J., Carpenter, Christopher L., Johnson, Neil W., Hann, Christine L., Kruger, Ryan G.

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Targeting enhancer switching overcomes non-genetic drug resistance in acute myeloid leukaemia von Bell, Charles C., Fennell, Katie A., Chan, Yih-Chih, Rambow, Florian, Yeung, Miriam M., Vassiliadis, Dane, Lara, Luis, Yeh, Paul, Martelotto, Luciano G., Rogiers, Aljosja, Kremer, Brandon E., Barbash, Olena, Mohammad, Helai P., Johanson, Timothy M., Burr, Marian L., Dhar, Arindam, Karpinich, Natalie, Tian, Luyi, Tyler, Dean S., MacPherson, Laura, Shi, Junwei, Pinnawala, Nathan, Yew Fong, Chun, Papenfuss, Anthony T., Grimmond, Sean M., Dawson, Sarah-Jane, Allan, Rhys S., Kruger, Ryan G., Vakoc, Christopher R., Goode, David L., Naik, Shalin H., Gilan, Omer, Lam, Enid Y. N., Marine, Jean-Christophe, Prinjha, Rab K., Dawson, Mark A.

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Mutation of A677 in histone methyltransferase EZH2 in human B-cell lymphoma promotes hypertrimethylation of histone H3 on lysine 27 (H3K27) von McCabe, Michael T, Graves, Alan P, Ganji, Gopinath, Diaz, Elsie, Halsey, Wendy S, Jiang, Yong, Smitheman, Kimberly N, Ott, Heidi M, Pappalardi, Melissa B, Allen, Kimberly E, Chen, Stephanie B, Della Pietra, Anthony III, Dul, Edward, Hughes, Ashley M, Gilbert, Seth A, Thrall, Sara H, Tummino, Peter J, Kruger, Ryan G, Brandt, Martin, Schwartz, Benjamin, Creasy, Caretha L

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Design of Ionic Liquid 3-Methyl-1-sulfonic Acid Imidazolium Nitrate as Reagent for the Nitration of Aromatic Compounds by in Situ Generation of NO2 in Acidic Media von Zolfigol, Mohammad A, Khazaei, Ardeshir, Moosavi-Zare, Ahmad R, Zare, Abdolkarim, Kruger, Hendrik G, Asgari, Zhila, Khakyzadeh, Vahid, Kazem-Rostami, Masoud

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Effect of nozzle selection on deposition of thiamethoxam in Actara® spray drift and implications for off-field risk assessment von Perine, J., Anderson, J.C., Kruger, G.R., Abi-Akar, F., Overmyer, J.

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Potential of brain mast cells for therapeutic application in the immune response to bacterial and viral infections von Natarajan, Satheesh, Govender, Kamini, Shobo, Adeola, Baijnath, Sooraj, Arvidsson, Per I., Govender, Thavendran, Lin, Johnson, Maguire, Glenn EM, Naicker, Tricia, Kruger, Hendrik. G.

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Enantioselective Organocatalyzed Transformations of β‑Ketoesters von Govender, Thavendran, Arvidsson, Per I, Maguire, Glenn E. M, Kruger, Hendrik G, Naicker, Tricia

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Crystal, spectroscopic and quantum mechanics studies of Schiff bases derived from 4-nitrocinnamaldehyde von Ani, Friday E., Ibeji, Collins U., Obasi, Nnamdi L., Kelani, Monsuru T., Ukogu, Kingsley, Tolufashe, Gideon F., Ogundare, Segun A., Oyeneyin, Oluwatoba E., Maguire, Glenn E. M., Kruger, Hendrik G.

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In vitro and in vivo induction of fetal hemoglobin with a reversible and selective DNMT1 inhibitor von Gilmartin, Aidan G, Groy, Arthur, Gore, Elizabeth R, Atkins, Charity, Long, Edward R, Montoute, Monica N, Wu, Zining, Halsey, Wendy, McNulty, Dean E, Ennulat, Daniela, Rueda, Lourdes, Pappalardi, Melissa, Kruger, Ryan G, McCabe, Michael T, Raoof, Ali, Butlin, Roger, Stowell, Alexandra, Cockerill, Mark, Waddell, Ian, Ogilvie, Donald, Luengo, Juan, Jordan, Allan, Benowitz, Andrew B

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Nanotechnology and the treatment of HIV infection von Parboosing, Raveen, Maguire, Glenn E M, Govender, Patrick, Kruger, Hendrik G

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Targeting Histone Methylation in Cancer von McCabe, Michael T, Mohammad, Helai P, Barbash, Olena, Kruger, Ryan G

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Interrogating the lack of diversity of thought in the pandemic response that led to mistakes - holistic evidence-based approach to deal with future pandemics von Aldous, Colleen, Kruger, Hendrik G

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Lysine specific demethylase 1 inactivation enhances differentiation and promotes cytotoxic response when combined with all- trans retinoic acid in acute myeloid leukemia across sub... von Smitheman, Kimberly N, Severson, Tesa M, Rajapurkar, Satyajit R, McCabe, Michael T, Karpinich, Natalie, Foley, James, Pappalardi, Melissa B, Hughes, Ashley, Halsey, Wendy, Thomas, Elizabeth, Traini, Christopher, Federowicz, Kelly E, Laraio, Jenny, Mobegi, Fredrick, Ferron-Brady, Geraldine, Prinjha, Rabinder K, Carpenter, Christopher L, Kruger, Ryan G, Wessels, Lodewyk, Mohammad, Helai P

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The effect of N-methylation of amino acids (Ac-X-OMe) on solubility and conformation: a DFT study von Md Abdur Rauf, Shah, Arvidsson, Per I, Albericio, Fernando, Govender, Thavendran, Maguire, Glenn E M, Kruger, Hendrik G, Honarparvar, Bahareh

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A Synthesis of “Dual Warhead” β‑Aryl Ethenesulfonyl Fluorides and One-Pot Reaction to β‑Sultams von Chinthakindi, Praveen K, Govender, Kimberleigh B, Kumar, A. Sanjeeva, Kruger, Hendrik G, Govender, Thavendran, Naicker, Tricia, Arvidsson, Per I

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Assembly of the SIR Complex and Its Regulation by O-Acetyl-ADP-Ribose, a Product of NAD-Dependent Histone Deacetylation von Liou, Gunn-Guang, Tanny, Jason C., Kruger, Ryan G., Walz, Thomas, Moazed, Danesh

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Smyd3 regulates cancer cell phenotypes and catalyzes histone H4 lysine 5 methylation von Van Aller, Glenn S, Reynoird, Nicolas, Barbash, Olena, Huddleston, Michael, Liu, Shichong, Zmoos, Anne-Flore, McDevitt, Patrick, Sinnamon, Robert, Le, BaoChau, Mas, Gloria, Annan, Roland, Sage, Julien, Garcia, Benjamin A, Tummino, Peter J, Gozani, Or, Kruger, Ryan G

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