Diastereoselective One-Pot Knoevenagel Condensation/Corey–Chaykovsky Cyclopropanation von Clemens, Jeremy J, Asgian, Juliana L, Busch, Brett B, Coon, Timothy, Ernst, Justin, Kaljevic, Leonard, Krenitsky, Paul J, Neubert, Timothy D, Schweiger, Edwin J, Termin, Andreas, Stamos, Dean

Volltext

Synthesis of the ( S, S, S)-diastereomer of the 15-membered biaryl ring system of RP 66453 von Krenitsky, Paul J., Boger, Dale L.

Volltext

Preparation of the 14-membered l, l-cycloisodityrosine subunit of RP 66453 von Krenitsky, Paul J., Boger, Dale L.

Volltext

CYCLIN-DEPENDENT KINASE DEGRADING COMPOUNDS von MENDY, Derek, MERCURIO, Frank, KRENITSKY, Paul J, XIE, Weilin, HAUGHEY, Michael P, ELSNER, Jan, PLANTEVIN-KRENITSKY, Veronique

Volltext bestellen

CK1 alpha AND DUAL CK1 alpha / GSPT1 DEGRADING COMPOUNDS von Sapienza, John, Haughey, Michael P, Elsner, Jan, Plantevin-Krenitsky, Veronique, Xie, Weilin, Mendy, Derek, Mercurio, Frank, Krenitsky, Paul J, Papa, Patrick W

Volltext bestellen

MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR von ZHOU, Jinglan, MILLER, Mark, Thomas, KHATUYA, Haripada, FRIEMAN, Bryan, A, CLEVELAND, Thomas, HADIDA RUAH, Sara S, BEAR, Brian, GROOTENHUIS, Peter, Diederik Jan, SILINA, Alina, COON, Timothy, Richard, UY, Johnny, KRENITSKY, Paul, J, CLEMENS, Jeremy

Volltext bestellen

MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR von ZHOU, Jinglan, MILLER, Mark, Thomas, KHATUYA, Haripada, FRIEMAN, Bryan, A, CLEVELAND, Thomas, HADIDA RUAH, Sara S, BEAR, Brian, GROOTENHUIS, Peter, Diederik Jan, SILINA, Alina, COON, Timothy, Richard, UY, Johnny, KRENITSKY, Paul, J, CLEMENS, Jeremy

Volltext bestellen

Divergent mechanisms for the dealkoxycarbonylation of a 2-(3-azetidinyl)malonate by chloride and cyanide von Gilligan, Paul J., Krenitsky, Paul J.

Volltext

MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR von ZHOU, Jinglan, MILLER, Mark, Thomas, KHATUYA, Haripada, FRIEMAN, Bryan, A, CLEVELAND, Thomas, HADIDA RUAH, Sara S, BEAR, Brian, GROOTENHUIS, Peter, Diederik Jan, SILINA, Alina, COON, Timothy, Richard, UY, Johnny, KRENITSKY, Paul, J, CLEMENS, Jeremy

Volltext bestellen

Modulators of cystic fibrosis transmembrane conductance regulator von Hadida Ruah, Sara S, Khatuya, Haripada, Cleveland, Thomas, Silina, Alina, Uy, Johnny, Frieman, Bryan A, Clemens, Jeremy, Coon, Timothy Richard, Grootenhuis, Peter Diederik Jan, Zhou, Jinglan, Miller, Mark Thomas, Bear, Brian, Krenitsky, Paul J

Volltext bestellen

MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR von ZHOU, Jinglan, MILLER, Mark, Thomas, KHATUYA, Haripada, FRIEMAN, Bryan, A, CLEVELAND, Thomas, HADIDA RUAH, Sara S, BEAR, Brian, GROOTENHUIS, Peter, Diederik Jan, SILINA, Alina, COON, Timothy, Richard, UY, Johnny, KRENITSKY, Paul, J, CLEMENS, Jeremy

Volltext bestellen

Synthesis of the (S,S,S)-Diastereomer (I) of the 15-Membered Biaryl Ring System of RP 66453 von Krenitsky, Paul J., Boger, Dale L.

Volltext

ChemInform Abstract: Preparation of the 14-Membered L,L-Cycloisodityrosine Subunit of RP 66453 von Krenitsky, Paul J., Boger, Dale L.

Volltext

MODULADOR DEL REGULADOR DE CONDUCTANCIA TRANSMEMBRANA DE FIBROSIS QUÍSTICA, COMPOSICIONES FARMACÉUTICAS, MÉTODOS DE TRATAMIENTO Y PROCESO PARA PRODUCIR EL MODULADOR von MILLER, MARK T, MCARTNEY, JASON, KHATUYA, HARIPADA, ALCACIO, TIMOTHY, ZHOU, JINGLAN, ANGELL, PAUL T, SHI, YI, HUGHES, ROBERT M, PARASELLI, PRASUNA, GROSS, RAYMOND S, SHRESTHA, MUNA, FERRIS, LORI ANN, CLEVELAND, THOMAS, KANG, PING, TERMIN, ANDREAS P, HSIA, CLARA KUANG, STAVROPOULOS, KATHY, KESHAVARZ-SHOKRI, ALI, PIERRE, FABRICE J. D, BAEK, MINSON, ABELA, ALEXANDER R, JOSHI, PRAMOD V, GULEVICH, ANTON, SIESEL, DAVID A, YOUNG, TIMOTHY JOHN, KRENITSKY, PAUL J, UY, JOHNNY, CLEMENS, JEREMY J, JU - HADIDA RUAH, SARA S, GROOTENHUIS, PETER D. J, ANDERSOY, COREY, VAN GOOR, FREDRICK F

Volltext bestellen

Automated multi-scale computational pathotyping (AMSCP) of inflamed synovial tissue von Bell, Richard D., Brendel, Matthew, Konnaris, Maxwell A., Xiang, Justin, Otero, Miguel, Fontana, Mark A., Bai, Zilong, Krenitsky, Daria M., Meednu, Nida, Rangel-Moreno, Javier, Scheel-Toellner, Dagmar, Carr, Hayley, Nayar, Saba, McMurray, Jack, DiCarlo, Edward, Anolik, Jennifer H., Donlin, Laura T., Orange, Dana E., Kenney, H. Mark, Schwarz, Edward M., Filer, Andrew, Ivashkiv, Lionel B., Wang, Fei

Volltext

When structure–affinity relationships meet structure–kinetics relationships: 3-((Inden-1-yl)amino)-1-isopropyl-cyclopentane-1-carboxamides as CCR2 antagonists von Vilums, Maris, Zweemer, Annelien J.M., Barmare, Farhana, van der Gracht, Anouk M.F., Bleeker, Dave C.T., Yu, Zhiyi, de Vries, Henk, Gross, Raymond, Clemens, Jeremy, Krenitsky, Paul, Brussee, Johannes, Stamos, Dean, Saunders, John, Heitman, Laura H., IJzerman, Adriaan P.

Volltext

Structure–Kinetic RelationshipsAn Overlooked Parameter in Hit-to-Lead Optimization: A Case of Cyclopentylamines as Chemokine Receptor 2 Antagonists von Vilums, Maris, Zweemer, Annelien J. M, Yu, Zhiyi, de Vries, Henk, Hillger, Julia M, Wapenaar, Hannah, Bollen, Ilse A. E, Barmare, Farhana, Gross, Raymond, Clemens, Jeremy, Krenitsky, Paul, Brussee, Johannes, Stamos, Dean, Saunders, John, Heitman, Laura H, IJzerman, Adriaan P

Volltext

Synthesis, Corticotropin-Releasing Factor Receptor Binding Affinity, and Pharmacokinetic Properties of Triazolo-, Imidazo-, and Pyrrolopyrimidines and -pyridines von Chorvat, Robert J, Bakthavatchalam, Rajagopal, Beck, James P, Gilligan, Paul J, Wilde, Richard G, Cocuzza, Anthony J, Hobbs, Frank W, Cheeseman, Robert S, Curry, Matthew, Rescinito, Joseph P, Krenitsky, Paul, Chidester, Dennis, Yarem, Jerry A, Klaczkiewicz, John D, Hodge, C. Nicholas, Aldrich, Paul E, Wasserman, Zelda R, Fernandez, Christine H, Zaczek, Robert, Fitzgerald, Lawrence W, Huang, Shiew-Mei, Shen, Helen L, Wong, Y. Nancy, Chien, Ben M, Quon, Check Y, Arvanitis, Argyrios

Volltext

MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR von Gross, Raymond Stanley, Clemens, Jeremy J, Cleveland, Thomas, Binch, Hayley Marie, Uy, Johnny, Nicholls, Georgia McGaughey, Marelius, Gulin Erdogan, Termin, Andreas P, Krenitsky, Paul John, Pierre, Fabrice Jean Denis, Khatuya, Haripada, Lin, Chun-Chieh, Silina, Alina, Conroy, Erica, McCartney, Jason, Frieman, Bryan A, Coon, Timothy Richard, Bear, Brian Richard, Arumugam, Vijayalaksmi, Grootenhuis, Peter Diederik Jan, Joshi, Pramod Virupax, Zhou, Jinglan, Miller, Mark Thomas, Melillo, Vito, Anderson, Corey, Hadida-Ruah, Sara Sabina

Volltext bestellen

MODULATOR OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR, PHARMACEUTICAL COMPOSITIONS, METHODS OF TREATMENT, AND PROCESS FOR MAKING THE MODULATOR von GROSS, Raymond, Stanley, ABELA, Alexander, Russell, MCCARTNEY, Jason, CLEVELAND, Thomas, KANG, Ping, KESHAVARZ-SHOKRI, Ali, JOSHI, Pramod, Virupax, STAVROPOULOS, Kathy, ALCACIO, Timothy, KHATUYA, KHATUYA, Haripada, TERMIN, Andreas, P, BAEK, Minson, SHI, Yi, SHRESTHA, Muna, FERRIS,, Lori, Ann, GROOTENHUIS, Peter Diederik, Jan, HSIA, Clara, Kuang-Ju, KRENITSKY, Paul, John, ANGELL, Paul, Timothy, MILLER, Mark, Thomas, ANDERSON, Corey, PARASELLI, Prasuna, YOUNG, Tomothy, John, ZHOU,, Jinglan, GULEVICH, Anton, VAN GOOR, Fredrik, F, UY, Johnny, CLEMENS, Jeremy, J, HADIDA RUAH, Sara, Sabina, PIERRE, Fa brice Jean, Denis, SIESEL, David, Andrew, HUGHES, Robert, M

Volltext bestellen