Novel Synthetic Inhibitors of Selectin-Mediated Cell Adhesion:  Synthesis of 1,6-Bis[3-(3-carboxymethylphenyl)-4-(2-α-d-mannopyranosyloxy)phenyl]hexane (TBC1269) von Kogan, Timothy P, Dupré, Brian, Bui, Huong, McAbee, Kathy L, Kassir, Jamal M, Scott, Ian L, Hu, Xin, Vanderslice, Peter, Beck, Pamela J, Dixon, Richard A. F

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Discovery of TBC11251, a Potent, Long Acting, Orally Active Endothelin Receptor-A Selective Antagonist von Wu, Chengde, Chan, Ming F, Stavros, Fiona, Raju, B, Okun, Ilya, Mong, Seymour, Keller, Karin M, Brock, Tommy, Kogan, Timothy P, Dixon, Richard A. F

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A Single Amino Acid Residue Can Determine the Ligand Specificity of E-selectin von Kogan, Timothy P., Revelle, B. Mitch, Tapp, Stephen, Scott, Dee, Beck, Pamela J.

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Rational Design and Synthesis of Small Molecule, Non-oligosaccharide Selectin Inhibitors: (.alpha.-D-Mannopyranosyloxy)biphenyl-Substituted Carboxylic Acids von Kogan, Timothy P, Dupre, Brian, Keller, Karin M, Scott, Ian L, Bui, Huong, Market, Robert V, Beck, Pamela J, Voytus, Jennifer A, Revelle, B. Mitch, Scott, Delores

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Small-molecule selectin inhibitor protects against liver inflammatory response after ischemia and reperfusion von Palma-Vargas, J.M, Toledo-Pereyra, Luis, Dean, Richard E, Harkema, James M, Dixon, Richard A.F, Kogan, Timothy P

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Novel inhibitors of α4β1 integrin receptor interactions through library synthesis and screening von Souers, Andrew J, Virgilio, Alex A, Schürer, Stephan S, Ellman, Jonathan A, Kogan, Timothy P, West, Henry E, Ankener, Wendy, Vanderslice, Peter

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Solution-phase combinatorial synthesis of ureas using nitrophenylcarbamates von Raju, B., Kassir, Jamal M., Kogan, Timothy P.

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Endothelin Antagonists:  Substituted Mesitylcarboxamides with High Potency and Selectivity for ETA Receptors von Wu, Chengde, Decker, E. Radford, Blok, Natalie, Bui, Huong, Chen, Qi, Raju, B, Bourgoyne, Andree R, Knowles, Vippra, Biediger, Ronald J, Market, Robert V, Lin, Shuqun, Dupré, Brian, Kogan, Timothy P, Holland, George W, Brock, Tommy A, Dixon, Richard A. F

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A Regio- and stereocontrolled total synthesis of (-)-indolactam-V von Kogan, Timothy P., Somers, Todd C., Venuti, Michael C.

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Selectin Blockade Prevents Antigen-induced Late Bronchial Responses and Airway Hyperresponsiveness in Allergic Sheep von ABRAHAM, WILLIAM M, AHMED, ASHFAQ, SABATER, JUAN R, LAUREDO, ISABEL T, BOTVINNIKOVA, YELENA, BJERCKE, ROBERT J, HU, X, REVELLE, B. MITCH, KOGAN, TIMOTHY P, SCOTT, IAN L, DIXON, RICHARD A. F, YEH, EDWARD T. H, BECK, PAMELA J

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Modification of CD4 Immunoadhesin with Monomethoxypoly(Ethylene Glycol) Aldehyde via Reductive Alkylation von Chamow, Steven M, Kogan, Timothy P, Venuti, Michael, Gadek, Thomas, Harris, Reed J, Peers, David H, Mordenti, Joyce, Shak, Steven, Ashkenazi, Avi

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Design, Synthesis, and Evaluation of Mitomycin-Tethered Phosphorothioate Oligodeoxynucleotides von Huh, Nam, Rege, Ajay A, Yoo, Byungwoo, Kogan, Timothy P, Kohn, Harold

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Substituted (1,2-Diarylethyl)amide Acyl-CoA:Cholesterol Acyltransferase Inhibitors: Effect of Polar Groups on in Vitro and in Vivo Activity von Clader, John W, Berger, Joel G, Burrier, Robert E, Davis, Harry R, Domalski, Martin, Dugar, Sundeep, Kogan, Timothy P, Salisbury, Brian, Vaccaro, Wayne

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Novastan® (Brand of Argatroban): A Small-Molecule, Direct Thrombin Inhibitor von Hursting, Marcie J., Alford, Kenneth L., Becker, Jeanclaude P., Brooks, R. Lynn, Joffrion, James L., Knappenberger, Gary D., Kogan, Patricia W., Kogan, Timothy P., Mckinney, Anthony A., Schwarz, Richard P.

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Selectin blockade prevents antigen-induced late bronchial responses and airway hyperresponsiveness in allergic sheep von ABRAHAM, W. M, AHMED, A, DIXON, R. A. F, YEH, E. T. H, BECK, P. J, SABATER, J. R, LAUREDO, I. T, BOTVINNIKOVA, Y, BJERCKE, R. J, HU, X, REVELLE, B. M, KOGAN, T. P, SCOTT, I. L

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Solid phase synthesis of sulfonamides using a carbamate linker von Raju, B., Kogan, Timothy P.

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State-of-the-Art Review: The Preclinical and Clinical Pharmacology of Novastan (Argatroban): A Small-Molecule, Direct Thrombin Inhibitor von Schwarz, Richard P., Becker, Jean-Claude P., Brooks, R. Lynn, Hursting, Marcie J., Joffrion, James L., Knappenberger, Gary D., Kogan, Timothy P., Kogan, Patricia W., McKinney, Anthony A.

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A 3D Structure Model of Integrin α4β1 Complex: I. Construction of a Homology Model of β1 and Ligand Binding Analysis von You, Tony J., Maxwell, David S., Kogan, Timothy P., Chen, Qi, Li, Jian, Kassir, Jamal, Holland, George W., Dixon, Richard A.F.

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Small peptide inhibitors of smooth muscle myosin light chain kinase von Gaeta, Federico C. A, Lehman de Gaeta, Laura S, Kogan, Timothy P, Or, Yat Sun, Foster, Carolyn, Czarniecki, Michael

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Use of halomethyl resins to immobilize amines: An efficient method for synthesis of sulfonamides and amides on a solid support von Raju, B., Kogan, Timothy P.

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