Structure-guided enzymology of the lipid A acyltransferase LpxM reveals a dual activity mechanism von Dovala, Dustin, Rath, Christopher M., Hu, Qijun, Sawyer, William S., Shia, Steven, Elling, Robert A., Knapp, Mark S., Metzger, Louis E.

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Discovery of imidazo[1,2-a]-pyridine inhibitors of pan-PI3 kinases that are efficacious in a mouse xenograft model von Han, Wooseok, Menezes, Daniel L., Xu, Yongjin, Knapp, Mark S., Elling, Robert, Burger, Matthew T., Ni, Zhi-Jie, Smith, Aaron, Lan, Jiong, Williams, Teresa E., Verhagen, Joelle, Huh, Kay, Merritt, Hanne, Chan, John, Kaufman, Susan, Voliva, Charles F., Pecchi, Sabina

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Potent, Selective, and Orally Bioavailable Inhibitors of VPS34 Provide Chemical Tools to Modulate Autophagy in Vivo von Honda, Ayako, Harrington, Edmund, Cornella-Taracido, Ivan, Furet, Pascal, Knapp, Mark S, Glick, Meir, Triantafellow, Ellen, Dowdle, William E, Wiedershain, Dmitri, Maniara, Wieslawa, Moore, Christine, Finan, Peter M, Hamann, Lawrence G, Firestone, Brant, Murphy, Leon O, Keaney, Erin P

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Structure guided optimization of a fragment hit to imidazopyridine inhibitors of PI3K von Pecchi, Sabina, Ni, Zhi-Jie, Han, Wooseok, Smith, Aaron, Lan, Jiong, Burger, Matthew, Merritt, Hanne, Wiesmann, Marion, Chan, John, Kaufman, Susan, Knapp, Mark S., Janssen, Johanna, Huh, Kay, Voliva, Charles F.

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Identification and structure–activity relationship of 2-morpholino 6-(3-hydroxyphenyl) pyrimidines, a class of potent and selective PI3 kinase inhibitors von Pecchi, Sabina, Renhowe, Paul A., Taylor, Clarke, Kaufman, Susan, Merritt, Hanne, Wiesmann, Marion, Shoemaker, Kevin R., Knapp, Mark S., Ornelas, Elizabeth, Hendrickson, Thomas F., Fantl, Wendy, Voliva, Charles F.

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Selective VPS34 inhibitor blocks autophagy and uncovers a role for NCOA4 in ferritin degradation and iron homeostasis in vivo von Dowdle, William E., Nyfeler, Beat, Nagel, Jane, Elling, Robert A., Liu, Shanming, Triantafellow, Ellen, Menon, Suchithra, Wang, Zuncai, Honda, Ayako, Pardee, Gwynn, Cantwell, John, Luu, Catherine, Cornella-Taracido, Ivan, Harrington, Edmund, Fekkes, Peter, Lei, Hong, Fang, Qing, Digan, Mary Ellen, Burdick, Debra, Powers, Andrew F., Helliwell, Stephen B., D’Aquin, Simon, Bastien, Julie, Wang, Henry, Wiederschain, Dmitri, Kuerth, Jenny, Bergman, Philip, Schwalb, David, Thomas, Jason, Ugwonali, Savuth, Harbinski, Fred, Tallarico, John, Wilson, Christopher J., Myer, Vic E., Porter, Jeffery A., Bussiere, Dirksen E., Finan, Peter M., Labow, Mark A., Mao, Xiaohong, Hamann, Lawrence G., Manning, Brendan D., Valdez, Reginald A., Nicholson, Thomas, Schirle, Markus, Knapp, Mark S., Keaney, Erin P., Murphy, Leon O.

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Lenvatinib plus Pembrolizumab or Everolimus for Advanced Renal Cell Carcinoma von Motzer, Robert, Alekseev, Boris, Rha, Sun-Young, Porta, Camillo, Eto, Masatoshi, Powles, Thomas, Grünwald, Viktor, Hutson, Thomas E, Kopyltsov, Evgeny, Méndez-Vidal, María J, Kozlov, Vadim, Alyasova, Anna, Hong, Sung-Hoo, Kapoor, Anil, Alonso Gordoa, Teresa, Merchan, Jaime R, Winquist, Eric, Maroto, Pablo, Goh, Jeffrey C, Kim, Miso, Gurney, Howard, Patel, Vijay, Peer, Avivit, Procopio, Giuseppe, Takagi, Toshio, Melichar, Bohuslav, Rolland, Frederic, De Giorgi, Ugo, Wong, Shirley, Bedke, Jens, Schmidinger, Manuela, Dutcus, Corina E, Smith, Alan D, Dutta, Lea, Mody, Kalgi, Perini, Rodolfo F, Xing, Dongyuan, Choueiri, Toni K

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Identification of Novel Small Molecule Ligands That Bind to Tetanus Toxin von Lightstone, Felice C., Prieto, Maria C., Singh, Anup K., Piqueras, Mari Carmen, Whittal, Randy M., Knapp, Mark S., Balhorn, Rod, Roe, Diana C.

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Cloning, Expression, and One-Step Purification of the Minimal Essential Domain of the Light Chain of Botulinum Neurotoxin Type A von Kadkhodayan, Saloumeh, Knapp, Mark S., Schmidt, James J., Fabes, Sarah E., Rupp, Bernhard, Balhorn, Rod

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SYSTEM ARCHITECTURE FOR THERMAL IMAGING AND THERMOGRAPHY CAMERAS von NEAL HENRY W, KNAPP MARK S, SOUTHERLAND RICHARD L, BLETTNER DOUGLAS A, MALONE II JAMES K, EMMETT JEFF R

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System architecture for thermal imaging and thermography cameras von Malone, II James K, Emmett Jeff R, Knapp Mark S, Neal Henry W, Blettner Douglas A, Southerland Richard L

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SYSTEM ARCHITECTURE FOR THERMAL IMAGING AND THERMOGRAPHY CAMERAS von MALONE II, JAMES K, BLETTNER, DOUGLAS A, NEAL, HENRY W, KNAPP, MARK S, EMMETT, JEFF R, SOUTHERLAND, RICHARD L

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SYSTEM ARCHITECTURE FOR THERMAL IMAGING AND THERMOGRAPHY CAMERAS von MALONE II, JAMES K, BLETTNER, DOUGLAS A, NEAL, HENRY W, KNAPP, MARK S, EMMETT, JEFF R, SOUTHERLAND, RICHARD L

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SYSTEM ARCHITECTURE FOR THERMAL IMAGING AND THERMOGRAPHY CAMERAS von MALONE, II JAMES K, NEAL HENRY W, KNAPP MARK S, SOUTHERLAND RICHARD L, BLETTNER DOUGLAS A, EMMETT JEFF R

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SYSTEM ARCHITECTURE FOR THERMAL IMAGING AND THERMOGRAPHY CAMERAS von MALONE II, JAMES K, BLETTNER, DOUGLAS A, NEAL, HENRY W, KNAPP, MARK S, EMMETT, JEFF R, SOUTHERLAND, RICHARD L

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SYSTEM ARCHITECTURE FOR THERMAL IMAGING AND THERMOGRAPHY CAMERAS von BLETTNER, Douglas A, SOUTHERLAND, Richard L, KNAPP, Mark S, EMMETT, Jeff R, MALONE II, James K, NEAL, Henry W

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Nocturnal polyuria and saluresis in renal allograft recipients von Knapp, M S, Pownall, R, Heath, M J, Trimble, I, Kowanko, I C

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Drought, Tree Mortality, and Wildfire in Forests Adapted to Frequent Fire von STEPHENS, SCOTT L., COLLINS, BRANDON M., FETTIG, CHRISTOPHER J., FINNEY, MARK A., HOFFMAN, CHAD M., KNAPP, ERIC E., NORTH, MALCOLM P., SAFFORD, HUGH, WAYMAN, REBECCA B.

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In Vitro Pharmacological Characterization of Buprenorphine, Samidorphan, and Combinations Being Developed as an Adjunctive Treatment of Major Depressive Disorder von Bidlack, Jean M, Knapp, Brian I, Deaver, Daniel R, Plotnikava, Margarita, Arnelle, Derrick, Wonsey, Angela M, Fern Toh, May, Pin, Sokhom S, Namchuk, Mark N

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Bayesian Self‐Optimization for Telescoped Continuous Flow Synthesis von Clayton, Adam D., Pyzer‐Knapp, Edward O., Purdie, Mark, Jones, Martin F., Barthelme, Alexandre, Pavey, John, Kapur, Nikil, Chamberlain, Thomas W., Blacker, A. John, Bourne, Richard A.

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