Metal‐Free Electrochemical Synthesis of Sulfonamides Directly from (Hetero)arenes, SO2, and Amines von Blum, Stephan P., Karakaya, Tarik, Schollmeyer, Dieter, Klapars, Artis, Waldvogel, Siegfried R.

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Investigating the Underappreciated Hydrolytic Instability of 1,8-Diazabicyclo[5.4.0]undec-7-ene and Related Unsaturated Nitrogenous Bases von Hyde, Alan M, Calabria, Ralph, Arvary, Rebecca, Wang, Xiao, Klapars, Artis

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A multifunctional catalyst that stereoselectively assembles prodrugs von DiRocco, Daniel A., Ji, Yining, Sherer, Edward C., Klapars, Artis, Reibarkh, Mikhail, Dropinski, James, Mathew, Rose, Maligres, Peter, Hyde, Alan M., Limanto, John, Brunskill, Andrew, Ruck, Rebecca T., Campeau, Louis-Charles, Davies, Ian W.

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Frontispiece: Metal‐Free Electrochemical Synthesis of Sulfonamides Directly from (Hetero)arenes, SO2, and Amines von Blum, Stephan P., Karakaya, Tarik, Schollmeyer, Dieter, Klapars, Artis, Waldvogel, Siegfried R.

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A General and Efficient Copper Catalyst for the Amidation of Aryl Halides von Klapars, Artis, Huang, Xiaohua, Buchwald, Stephen L

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Mechanism-Based Solution to the ProTide Synthesis Problem: Selective Access to Sofosbuvir, Acelarin, and INX-08189 von Simmons, Bryon, Liu, Zhuqing, Klapars, Artis, Bellomo, Ana, Silverman, Steven M

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Multi-column ultra-high performance liquid chromatography screening with chaotropic agents and computer-assisted separation modeling enables process development of new drug substan... von Haidar Ahmad, Imad A, Chen, Wenyong, Halsey, Holst M, Klapars, Artis, Limanto, John, Pirrone, Gregory F, Nowak, Timothy, Bennett, Raffeal, Hartman, Robert, Makarov, Alexey A, Mangion, Ian, Regalado, Erik L

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Unlocking the Potential of High-Throughput Experimentation for Electrochemistry with a Standardized Microscale Reactor von Rein, Jonas, Annand, James R, Wismer, Michael K, Fu, Jiantao, Siu, Juno C, Klapars, Artis, Strotman, Neil A, Kalyani, Dipannita, Lehnherr, Dan, Lin, Song

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Copper-Catalyzed Domino Halide Exchange-Cyanation of Aryl Bromides von Zanon, Jacopo, Klapars, Artis, Buchwald, Stephen L

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Biocatalytic oxidation of alcohols using galactose oxidase and a manganese() activator for the synthesis of islatravir von Johnson, Heather C, Zhang, Shaoguang, Fryszkowska, Anna, Ruccolo, Serge, Robaire, Sandra A, Klapars, Artis, Patel, Niki R, Whittaker, Aaron M, Huffman, Mark A, Strotman, Neil A

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The Copper-Catalyzed N-Arylation of Indoles von Antilla, Jon C, Klapars, Artis, Buchwald, Stephen L

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A General and Efficient Copper Catalyst for the Amidation of Aryl Halides and the N-Arylation of Nitrogen Heterocycles von Klapars, Artis, Antilla, Jon C, Huang, Xiaohua, Buchwald, Stephen L

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Supercritical fluid chromatography-photodiode array detection-electrospray ionization mass spectrometry as a framework for impurity fate mapping in the development and manufacture... von Pirrone, Gregory F., Mathew, Rose M., Makarov, Alexey A., Bernardoni, Frank, Klapars, Artis, Hartman, Robert, Limanto, John, Regalado, Erik L.

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Efficient synthesis of antiviral agent uprifosbuvir enabled by new synthetic methods von Klapars, Artis, Chung, John Y. L, Limanto, John, Calabria, Ralph, Campeau, Louis-Charles, Campos, Kevin R, Chen, Wenyong, Dalby, Stephen M, Davis, Tyler A, DiRocco, Daniel A, Hyde, Alan M, Kassim, Amude M, Larsen, Mona Utne, Liu, Guiquan, Maligres, Peter E, Moment, Aaron, Peng, Feng, Ruck, Rebecca T, Shevlin, Michael, Simmons, Bryon L, Song, Zhiguo Jake, Tan, Lushi, Wright, Timothy J, Zultanski, Susan L

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Preparation of Enamides via Palladium-Catalyzed Amidation of Enol Tosylates von Klapars, Artis, Campos, Kevin R, Chen, Cheng-yi, Volante, Ralph P

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Metallfreie, elektrochemische Synthese von Sulfonamiden direkt aus (Hetero)arenen, SO2 und Aminen von Blum, Stephan P., Karakaya, Tarik, Schollmeyer, Dieter, Klapars, Artis, Waldvogel, Siegfried R.

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Engineered Ribosyl-1-Kinase Enables Concise Synthesis of Molnupiravir, an Antiviral for COVID-19 von McIntosh, John A, Benkovics, Tamas, Silverman, Steven M, Huffman, Mark A, Kong, Jongrock, Maligres, Peter E, Itoh, Tetsuji, Yang, Hao, Verma, Deeptak, Pan, Weilan, Ho, Hsing-I, Vroom, Jonathan, Knight, Anders M, Hurtak, Jessica A, Klapars, Artis, Fryszkowska, Anna, Morris, William J, Strotman, Neil A, Murphy, Grant S, Maloney, Kevin M, Fier, Patrick S

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Enantioselective, Biocatalytic Reduction of 3-Substituted Cyclopentenones: Application to the Asymmetric Synthesis of an hNK-1 Receptor Antagonist von Campos, Kevin R, Klapars, Artis, Kohmura, Yoshinori, Pollard, David, Ishibashi, Hideaki, Kato, Shinji, Takezawa, Akihiro, Waldman, Jacob H, Wallace, Debra J, Chen, Cheng-yi, Yasuda, Nobuyoshi

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Electrochemical Activation of Galactose Oxidase: Mechanistic Studies and Synthetic Applications von Zhang, Shaoguang, Ruccolo, Serge, Fryszkowska, Anna, Klapars, Artis, Marshall, Nicholas, Strotman, Neil A

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Synthetic Enantiopure Aziridinomitosenes:  Preparation, Reactivity, and DNA Alkylation Studies von Vedejs, Edwin, Naidu, B. N, Klapars, Artis, Warner, Don L, Li, Ven-shun, Na, Younghwa, Kohn, Harold

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