Structures of Kibdelomycin Bound to Staphylococcus aureus GyrB and ParE Showed a Novel U‑Shaped Binding Mode von Lu, Jun, Patel, Sangita, Sharma, Nandini, Soisson, Stephen M, Kishii, Ryuta, Takei, Masaya, Fukuda, Yasumichi, Lumb, Kevin J, Singh, Sheo B

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Contribution of Topoisomerase IV Mutation to Quinolone Resistance in Mycoplasma genitalium von YAMAGUCHI, Yuko, TAKEI, Masaya, KISHII, Ryuta, YASUDA, Mitsuru, DEGUCHI, Takashi

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Relationship between the expression of ompF and quinolone resistance in Escherichia coli von Kishii, Ryuta, Takei, Masaya

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Kibdelomycin is a bactericidal broad-spectrum aerobic antibacterial agent von Singh, Sheo B, Dayananth, Priya, Balibar, Carl J, Garlisi, Charles G, Lu, Jun, Kishii, Ryuta, Takei, Masaya, Fukuda, Yasumichi, Ha, Sookhee, Young, Katherine

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Target Preference of 15 Quinolones against Staphylococcus aureus, Based on Antibacterial Activities and Target Inhibition von TAKEI, Masaya, FUKUDA, Hideyuki, KISHII, Ryuta, HOSAKA, Masaki

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In Vitro Activities and Spectrum of the Novel Fluoroquinolone Lascufloxacin (KRP-AM1977) von Kishii, Ryuta, Yamaguchi, Yuko, Takei, Masaya

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Structural and Functional Studies of the HAMP Domain of EnvZ, an Osmosensing Transmembrane Histidine Kinase in Escherichia coli von Kishii, Ryuta, Falzon, Liliana, Yoshida, Takeshi, Kobayashi, Hiroshi, Inouye, Masayori

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Serum/glucocorticoid-regulated kinase 1 contributes to the proliferation of varicella-zoster virus and induction of cyclin B1 expression von Oda, Shinya, Yokoyama, Akinobu, Kishii, Ryuta, Nagasawa, Michiaki

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Contributions of the 8-Methoxy Group of Gatifloxacin to Resistance Selectivity, Target Preference, and Antibacterial Activity against Streptococcus pneumoniae von FUKUDA, Hideyuki, KISHII, Ryuta, TAKEI, Masaya, HOSAKA, Masaki

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Contribution of the 8-Methoxy Group to the Activity of Gatifloxacin against Type II Topoisomerases of Streptococcus pneumoniae von KISHII, Ryuta, TAKEI, Masaya, FUKUDA, Hideyuki, HAYASHI, Katsuhiko, HOSAKA, Masaki

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Sulfonamide-based non-alkyne LpxC inhibitors as Gram-negative antibacterial agents von Kawai, Tetsuya, Kazuhiko, Iwase, Takaya, Noriko, Yamaguchi, Yuko, Kishii, Ryuta, Kohno, Yasushi, Kurasaki, Haruaki

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Structure activity relationship of N-1 substituted 1,5-naphthyrid-2-one analogs of oxabicyclooctane-linked novel bacterial topoisomerase inhibitors as broad-spectrum antibacterial... von Singh, Sheo B., Tan, Christopher M., Kaelin, David, Meinke, Peter T., Miesel, Lynn, Olsen, David B., Fukuda, Hideyuki, Kishii, Ryuta, Takei, Masaya, Ohata, Kohei, Takeuchi, Tomoko, Shibue, Taku, Takano, Hisashi, Nishimura, Akinori, Fukuda, Yasumichi

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LpxC Inhibitors: Design, Synthesis, and Biological Evaluation of Oxazolidinones as Gram-negative Antibacterial Agents von Kurasaki, Haruaki, Tsuda, Kosuke, Shinoyama, Mariko, Takaya, Noriko, Yamaguchi, Yuko, Kishii, Ryuta, Iwase, Kazuhiko, Ando, Naoki, Nomura, Masahiro, Kohno, Yasushi

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The effect of pharmacokinetic/pharmacodynamic (PK/PD) parameters of gatifloxacin on its bactericidal activity and resistance selectivity against clinical isolates of Streptococcus... von Ebisu, Hiroyuki, Kishii, Ryuta, Takei, Masaya, Fukuda, Hideyuki

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In Vitro and In Vivo Characterization of the Novel Oxabicyclooctane-Linked Bacterial Topoisomerase Inhibitor AM-8722, a Selective, Potent Inhibitor of Bacterial DNA Gyrase von Tan, Christopher M, Gill, Charles J, Wu, Jin, Toussaint, Nathalie, Yin, Jingjun, Tsuchiya, Takayuki, Garlisi, Charles G, Kaelin, David, Meinke, Peter T, Miesel, Lynn, Olsen, David B, Lagrutta, Armando, Fukuda, Hideyuki, Kishii, Ryuta, Takei, Masaya, Oohata, Kouhei, Takeuchi, Tomoko, Shibue, Taku, Takano, Hisashi, Nishimura, Akinori, Fukuda, Yasumichi, Singh, Sheo B

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Oxabicyclooctane-Linked Novel Bacterial Topoisomerase Inhibitors as Broad Spectrum Antibacterial Agents von Singh, Sheo B, Kaelin, David E, Wu, Jin, Miesel, Lynn, Tan, Christopher M, Meinke, Peter T, Olsen, David, Lagrutta, Armando, Bradley, Prudence, Lu, Jun, Patel, Sangita, Rickert, Keith W, Smith, Robert F, Soisson, Stephen, Wei, Changqing, Fukuda, Hideyuki, Kishii, Ryuta, Takei, Masaya, Fukuda, Yasumichi

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Tricyclic 1,5-naphthyridinone oxabicyclooctane-linked novel bacterial topoisomerase inhibitors as broad-spectrum antibacterial agents-SAR of left-hand-side moiety (Part-2) von Singh, Sheo B, Kaelin, David E, Wu, Jin, Miesel, Lynn, Tan, Christopher M, Black, Todd, Nargund, Ravi, Meinke, Peter T, Olsen, David B, Lagrutta, Armando, Lu, Jun, Patel, Sangita, Rickert, Keith W, Smith, Robert F, Soisson, Stephen, Sherer, Edward, Joyce, Leo A, Wei, Changqing, Peng, Xuanjia, Wang, Xiu, Fukuda, Hideyuki, Kishii, Ryuta, Takei, Masaya, Takano, Hisashi, Shibasaki, Mitsuhito, Yajima, Masanobu, Nishimura, Akinori, Shibata, Takeshi, Fukuda, Yasumichi

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Hydroxy tricyclic 1,5-naphthyridinone oxabicyclooctane-linked novel bacterial topoisomerase inhibitors as broad-spectrum antibacterial agents-SAR of RHS moiety (Part-3) von Singh, Sheo B., Kaelin, David E., Wu, Jin, Miesel, Lynn, Tan, Christopher M., Gill, Charles, Black, Todd, Nargund, Ravi, Meinke, Peter T., Olsen, David B., Lagrutta, Armando, Wei, Changqing, Peng, Xuanjia, Wang, Xiu, Fukuda, Hideyuki, Kishii, Ryuta, Takei, Masaya, Takeuchi, Tomoko, Shibue, Taku, Ohata, Kohei, Takano, Hisashi, Ban, Shizuka, Nishimura, Akinori, Fukuda, Yasumichi

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Structure activity relationship of pyridoxazinone substituted RHS analogs of oxabicyclooctane-linked 1,5-naphthyridinyl novel bacterial topoisomerase inhibitors as broad-spectrum a... von Singh, Sheo B., Kaelin, David E., Wu, Jin, Miesel, Lynn, Tan, Christopher M., Meinke, Peter T., Olsen, David B., Lagrutta, Armando, Wei, Changqing, Liao, Yonggang, Peng, Xuanjia, Wang, Xiu, Fukuda, Hideyuki, Kishii, Ryuta, Takei, Masaya, Yajima, Masanobu, Shibue, Taku, Shibata, Takeshi, Ohata, Kohei, Nishimura, Akinori, Fukuda, Yasumichi

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Structure activity relationship of C-2 ether substituted 1,5-naphthyridine analogs of oxabicyclooctane-linked novel bacterial topoisomerase inhibitors as broad-spectrum antibacteri... von Singh, Sheo B., Kaelin, David E., Meinke, Peter T., Wu, Jin, Miesel, Lynn, Tan, Christopher M., Olsen, David B., Lagrutta, Armando, Fukuda, Hideyuki, Kishii, Ryuta, Takei, Masaya, Takeuchi, Tomoko, Takano, Hisashi, Ohata, Kohei, Kurasaki, Haruaki, Nishimura, Akinori, Shibata, Takeshi, Fukuda, Yasumichi

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