Discovery and binding mode of small molecule inhibitors of the apo form of human TDO2 von Lotz-Jenne, Carina, Lange, Roland, Cren, Sylvaine, Bourquin, Geoffroy, Goglia, Laksmei, Kimmerlin, Thierry, Wicki, Micha, Müller, Manon, Artico, Nadia, Ackerknecht, Sabine, Pfaff, Philippe, Joesch, Christoph, Mac Sweeney, Aengus

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The Screening Compound Collection: A Key Asset for Drug Discovery von Boss, Christoph, Hazemann, Julien, Kimmerlin, Thierry, von Korff, Modest, Lüthi, Urs, Peter, Oliver, Sander, Thomas, Siegrist, Romain

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Highly Potent and Cellularly Active β-Peptidic Inhibitor of the p53/hDM2 Interaction von Hintersteiner, Martin, Kimmerlin, Thierry, Garavel, Geraldine, Schindler, Thorsten, Bauer, Roman, Meisner, Nicole-Claudia, Seifert, Jan-Marcus, Uhl, Volker, Auer, Manfred

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Discovery and Optimization of Isoquinoline Ethyl Ureas as Antibacterial Agents von Panchaud, Philippe, Bruyère, Thierry, Blumstein, Anne-Catherine, Bur, Daniel, Chambovey, Alain, Ertel, Eric A, Gude, Markus, Hubschwerlen, Christian, Jacob, Loïc, Kimmerlin, Thierry, Pfeifer, Thomas, Prade, Lars, Seiler, Peter, Ritz, Daniel, Rueedi, Georg

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Identification of SARS-CoV-2 Mpro inhibitors through deep reinforcement learning for drug design and computational chemistry approaches von Hazemann, Julien, Kimmerlin, Thierry, Lange, Roland, Sweeney, Aengus Mac, Bourquin, Geoffroy, Ritz, Daniel, Czodrowski, Paul

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Identification of SARS-CoV-2 Mpro inhibitors through deep reinforcement learning for de novo drug design and computational chemistry approaches von Hazemann, Julien, Kimmerlin, Thierry, Lange, Roland, Sweeney, Aengus Mac, Bourquin, Geoffroy, Ritz, Daniel, Czodrowski, Paul

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Peptide Folding Induces High and Selective Affinity of a Linear and Small β-Peptide to the Human Somatostatin Receptor 4 von Gademann, Karl, Kimmerlin, Thierry, Hoyer, Daniel, Seebach, Dieter

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How we drifted into peptide chemistry and where we have arrived at von Seebach, Dieter, Kimmerlin, Thierry, Šebesta, Radovan, Campo, Marino A., Beck, Albert K.

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Covalent Fluorescence Labeling of His-Tagged Proteins on the Surface of Living Cells von Hintersteiner, Martin, Weidemann, Thomas, Kimmerlin, Thierry, Filiz, Nimet, Buehler, Christof, Auer, Manfred

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Investigation of the Interactions of β-Peptides with DNA Duplexes by Circular Dichroism Spectroscopy von Namoto, Kenji, Gardiner, James, Kimmerlin, Thierry, Seebach, Dieter

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Solid-Phase Synthesis of a β3-Icosapeptide Containing the Homologs of the Twenty Common Proteinaceous Amino Acids. Preliminary Communication von Kimmerlin, Thierry, Seebach, Dieter

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Solid‐Phase Synthesis of a β 3 ‐Icosapeptide Containing the Homologs of the Twenty Common Proteinaceous Amino Acids. Preliminary Communication von Kimmerlin, Thierry, Seebach, Dieter

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Investigation of the Interactions of b-Peptides with DNA Duplexes by Circular Dichroism Spectroscopy von Namoto, Kenji, Gardiner, James, Kimmerlin, Thierry, Seebach, Dieter

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Beta(2)/beta(3)-di- and alpha/beta(3)-tetrapeptide derivatives as potent agonists at somatostatin sst(4) receptors von Nunn, Caroline, Rueping, Magnus, Langenegger, Daniel, Schuepbach, Edi, Kimmerlin, Thierry, Micuch, Peter, Hurth, Konstanze, Seebach, Dieter, Hoyer, Daniel

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68 Targeting SH2-Domain Mediated Cell Signaling by Mixed α/β Peptide Ligands von Kalthoff, Frank S., Hintersteiner, Martin, Kimmerlin, Thierry, Buehler, Christoph, Garavel, Geraldine, Auer, Manfred

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Comparative Metabolism of α- and β-Peptides in the Insect Heliothis virescens and in Plant Cells of Black Mexican Sweet Maize von Lind, Rob, Greenhow, Daren, Perry, Simon, Kimmerlin, Thierry, Seebach, Dieter

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Preparation of β2-Amino Acid Derivatives (β2hThr, β2hTrp, β2hMet, β2hPro, β2hLys, Pyrrolidine-3-carboxylic Acid) by Using DIOZ as Chiral Auxiliary von Gessier, Francois, Schaeffer, Laurent, Kimmerlin, Thierry, Flögel, Oliver, Seebach, Dieter

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Evidence from Circular Dichroism and from Melting Behavior for Helix-Inducing Complexation of a Designed β3-Pentadecapeptide with DNA Duplexes. Preliminary Communication von Kimmerlin, Thierry, Namoto, Kenji, Seebach, Dieter

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Evidence from Circular Dichroism and from Melting Behavior for Helix‐Inducing Complexation of a Designed β 3 ‐Pentadecapeptide with DNA Duplexes. Preliminary Communication von Kimmerlin, Thierry, Namoto, Kenji, Seebach, Dieter

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Evidence from Circular Dichroism and from Melting Behavior for Helix-Inducing Complexation of a Designed b3-Pentadecapeptide with DNA Duplexes. Preliminary Communication von Kimmerlin, Thierry, Namoto, Kenji, Seebach, Dieter

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