Perspectives on the Designation of Oligonucleotide Starting Materials von Kiesman, William F., McPherson, Andrew K., Diorazio, Louis J., Van den Bergh, Leo, Smith, Peter D., Northall, John M., Fettes, Alec, Wang, Tiejun, Mehlmann, Martin, Raza, Syed, Held, Gary

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Development of Kilogram-Scale Convergent Liquid-Phase Synthesis of Oligonucleotides von Zhou, Xuan, Kiesman, William F, Yan, Wuming, Jiang, Hong, Antia, Firoz D, Yang, Jing, Fillon, Yannick A, Xiao, Li, Shi, Xianglin

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The Chelate Effect Rationalizes Observed Rate Acceleration and Enantioselectivity in BINOL‐Catalyzed Petasis Reactions von Haeffner, Fredrik, Pickel, Thomas C., Hou, April, Walker, Donald G., Kiesman, William F., Shi, Xianglin

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Solid-Phase Synthesis of Phosphorothioate Oligonucleotides Using Sulfurization Byproducts for in Situ Capping von Yang, Jimin, Stolee, Jessica A, Jiang, Hong, Xiao, Li, Kiesman, William F, Antia, Firoz D, Fillon, Yannick A, Ng, Austen, Shi, Xianglin

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Catalytic Asymmetric Petasis Reactions of Vinylboronates von Shi, Xianglin, Kiesman, William F, Levina, Anna, Xin, Zhili

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Synthesis of Vixotrigine, a Voltage- and Use-Dependent Sodium Channel Blocker. Part 2: Development of a Late-Stage Process von Chen, Robbie, Couming, Vincent, Guzowski, John, Irdam, Erwin, Kiesman, William F, Kwok, Daw-Iong Albert, Liang, Wenli, Mack, Tamera, O’Brien, Erin M, Opalka, Suzanne M, Patience, Daniel, Sahli, Stefan, Walker, Donald G, Osei-Yeboah, Frederick, Gu, Chaozhan, Zhang, Xin, Stöckli, Markus, Stucki, Thiemo, Matzinger, Hanspeter, Kuhn, Roman, Thut, Michael, Grohmann, Markus, Haefner, Benjamin, Lotz, Joerg, Nonnenmacher, Michael, Cerea, Paolangelo

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Acceleration of Petasis Reactions of Salicylaldehyde Derivatives with Molecular Sieves von Shi, Xianglin, Hebrault, Dominique, Humora, Michael, Kiesman, William F, Peng, Hairuo, Talreja, Tina, Wang, Zezhou, Xin, Zhili

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Process Development of an N‑Benzylated Chloropurine at the Kilogram Scale von Shi, Xianglin, Chang, Hexi, Grohmann, Markus, Kiesman, William F, Kwok, Daw-Iong Albert

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Part 2: Designation and Justification of API Starting Materials: Current Practices across Member Companies of the IQ Consortium von Faul, Margaret M, Busacca, Carl A, Eriksson, Magnus C, Hicks, Fred, Kiesman, William F, Smulkowski, Maciej, Orr, John D, Pfeiffer, Steven

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Part 3: Designation and Justification of API Starting Materials: Proposed Framework for Alignment from an Industry Perspective von Faul, Margaret M, Argentine, Mark D, Egan, Marjorie, Eriksson, Magnus C, Ge, Zhihong, Hicks, Fred, Kiesman, William F, Mergelsberg, Ingrid, Orr, John D, Smulkowski, Maciej, Wächter, Gerald A

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Understanding and Control of Dimethyl Sulfate in a Manufacturing Process: Kinetic Modeling of a Fischer Esterification Catalyzed by H2SO4 von Guzowski, John P, Delaney, Edward J, Humora, Michael J, Irdam, Erwin, Kiesman, William F, Kwok, Albert, Moran, Amy D

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Detection of Aryl Radicals in Hydrodediazoniations von Wassmundt, Frederick W, Kiesman, William F

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Soluble Catalysts for Improved Pschorr Cyclizations von Wassmundt, Frederick W, Kiesman, William F

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Highly Regio- and Enantioselective Catalytic Hydrogenation of Enamides in Conjugated Diene Systems:  Synthesis and Application of γ,δ-Unsaturated Amino Acids von Burk, Mark J, Allen, John G, Kiesman, William F

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Development of an Early Phase Process for a Potent Oligodendrocyte Precursor Cell Differentiator von Walker, Donald G., Ferguson, Steven, Humora, Michael J., Irdam, Erwin, Kiesman, William F., Kwok, Daw-Iong Albert, Liang, Wenli, Opalka, Suzanne M.

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Norbornyllactone-substituted xanthines as adenosine A1 receptor antagonists von KIESMAN, William F, JIN ZHAO, CONLON, Patrick R, PETTER, Russell C, XIAOWEI JIN, SMITS, Glenn, LUTTERODT, Frank, SULLIVAN, Gail W, LINDEN, Joel

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Lewis-acid catalysis of the asymmetric Diels–Alder reaction of dimenthyl fumarate and cyclopentadiene von Kiesman, William F, Petter, Russell C

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Efficient Catalysis of Hydrodediazoniations in Dimethylformamide von Wassmundt, Frederick W, Kiesman, William F

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Synthesis of alkyne derivatives of a novel triazolopyrazine as A 2A adenosine receptor antagonists von Yao, Gang, Haque, Serajul, Sha, Li, Kumaravel, Gnanasambandam, Wang, Joy, Engber, Thomas M., Whalley, Eric T., Conlon, Patrick R., Chang, Hexi, Kiesman, William F., Petter, Russell C.

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Synthesis of alkyne derivatives of a novel triazolopyrazine as A(2A) adenosine receptor antagonists von Yao, Gang, Haque, Serajul, Sha, Li, Kumaravel, Gnanasambandam, Wang, Joy, Engber, Thomas M, Whalley, Eric T, Conlon, Patrick R, Chang, Hexi, Kiesman, William F, Petter, Russell C

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