Discovery of New Quinolone-Based Diarylamides as Potent B-RAFV600E/C-RAF Kinase Inhibitors Endowed with Promising In Vitro Anticancer Activity von Hyun Ji Kim, Jung Woo Park, Seo, Sangjae, Cho, Kwang-Hwi, Alanazi, Mohammed M, Bang, Eun-Kyoung, Gyochang Keum, El-Damasy, Ashraf K

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Metal/catalyst-free sequential C-N bond forming cascades at room temperature: environment-friendly one-pot synthesis of 5-aminoimidazoles from aryl glyoxals, anilines, and amidines von Jalani, Hitesh B, Sivaraman, Aneesh, Min, Kyoung ho, Lee, Hwa Young, Oh, Na Kyoung, Kang, Hyeseul, Keum, Gyochang, Choi, Yongseok, Lee, Kyeong

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Immunogenicity and protection of a triple repeat domain III mRNA vaccine against Zika virus von Lee, Yu-Sun, Cheong, Mi Sun, Lee, Jisun, Bang, Eun-Kyoung, Park, Sang In, Park, Hyo-Jung, Bae, Seo-Hyeon, Yoon, Subin, Roh, Gahyun, Lee, Seonghyun, Cho, Youngran, Ha, Dahyeon, Oh, Ayoung, Lee, Soo-Yeon, Choi, Eun-Jin, Choi, Huijeong, Jo, Sohee, Lee, Yeeun, Kim, Jungmin, Kwak, Hye Won, Bang, Yoo-Jin, Lee, Dabin, Shim, Heeyoun, Park, Young Kun, Keum, Gyochang, Nam, Jae-Hwan, Kim, Wonil

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Discovery of new 6-ureido/amidocoumarins as highly potent and selective inhibitors for the tumour-relevant carbonic anhydrases IX and XII von El-Damasy, Ashraf K., Kim, Hyun Ji, Nocentini, Alessio, Seo, Seon Hee, Eldehna, Wagdy M., Bang, Eun-Kyoung, Supuran, Claudiu T., Keum, Gyochang

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Overcoming the imatinib-resistant BCR-ABL mutants with new ureidobenzothiazole chemotypes endowed with potent and broad-spectrum anticancer activity von El-Damasy, Ashraf K, Jin, Heewon, Park, Jung Woo, Kim, Hyun Ji, Khojah, Hanan, Seo, Seon Hee, Lee, Ju-Hyeon, Bang, Eun-Kyoung, Keum, Gyochang

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Discovery of New Quinoline-Based Diarylamides as Potent B-RAFV600E/C-RAF Kinase Inhibitors Endowed with Promising In Vitro Anticancer Activity von Kim, Hyun, Park, Jung, Seo, Sangjae, Cho, Kwang-Hwi, Alanazi, Mohammed, Bang, Eun-Kyoung, Keum, Gyochang, El-Damasy, Ashraf

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Discovery of 3-((3-amino-1H-indazol-4-yl)ethynyl)-N-(4-((4-ethylpiperazin-1-yl)methyl)-3-(trifluoromethyl)phenyl)benzamide (AKE-72), a potent Pan-BCR-ABL inhibitor including the T3... von El-Damasy, Ashraf K., Kim, Hyun Ji, Park, Jung Woo, Nam, Yunju, Hur, Wooyoung, Bang, Eun-Kyoung, Keum, Gyochang

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mRNA‐HPV vaccine encoding E6 and E7 improves therapeutic potential for HPV‐mediated cancers via subcutaneous immunization von Lee, Seonghyun, Yoon, Hyunho, Hong, Seol Hee, Kwon, Sung Pil, Hong, Jung Joo, Kwak, Hye Won, Park, Hyeong‐Jun, Yoo, Soyeon, Bae, Seo‐Hyeon, Park, Hyo‐Jung, Lee, Jisun, Bang, Yoo‐Jin, Lee, Yu‐Sun, Kim, Jae‐Yong, Yoon, Subin, Roh, Gahyun, Cho, Youngran, Kim, Yongkwan, Kim, Daegeun, Park, Sang‐In, Kim, Do‐Hyung, Lee, Sowon, Oh, Ayoung, Ha, Dahyeon, Lee, Soo‐Yeon, Park, Misung, Hwang, Eun‐Ha, Bae, Gyuseo, Jeon, Eunsu, Park, Sung Hyun, Choi, Won Seok, Oh, Ho Rim, Kim, In Woo, Youn, Hyewon, Keum, Gyochang, Bang, Eun‐Kyoung, Rhee, Joon Haeng, Lee, Shee Eun, Nam, Jae‐Hwan

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Identification of New N -methyl-piperazine Chalcones as Dual MAO-B/AChE Inhibitors von El-Damasy, Ashraf K, Park, Jong Eun, Kim, Hyun Ji, Lee, Jinhyuk, Bang, Eun-Kyoung, Kim, Hoon, Keum, Gyochang

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Identification of Ureidocoumarin-Based Selective Discoidin Domain Receptor 1 (DDR1) Inhibitors via Drug Repurposing Approach, Biological Evaluation, and In Silico Studies von El-Damasy, Ashraf K, Kim, Hyun Ji, Al-Karmalawy, Ahmed A, Alnajjar, Radwan, Khalifa, Mohamed M, Bang, Eun-Kyoung, Keum, Gyochang

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Coordinative Amphiphiles as Tunable siRNA Transporters von Kim, Jin Bum, Lee, Yeong Mi, Ryu, Jooyeon, Lee, Eunji, Kim, Won Jong, Keum, Gyochang, Bang, Eun-Kyoung

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Nanoformulated Single‐Stranded RNA‐Based Adjuvant with a Coordinative Amphiphile as an Effective Stabilizer: Inducing Humoral Immune Response by Activation of Antigen‐Presenting Ce... von Park, Hyo‐Jung, Bang, Eun‐Kyoung, Hong, Jung Joo, Lee, Sang‐Myeong, Ko, Hae Li, Kwak, Hye Won, Park, Hyelim, Kang, Kyung Won, Kim, Rhoon‐Ho, Ryu, Seung Rok, Kim, Green, Oh, Hanseul, Kim, Hye‐Jung, Lee, Kyuri, Kim, Minjeong, Kim, Soo Young, Kim, Jae‐Ouk, El‐Baz, Karim, Lee, Hyukjin, Song, Manki, Jeong, Dae Gwin, Keum, Gyochang, Nam, Jae‐Hwan

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Structural Basis for Design of New Purine-Based Inhibitors Targeting the Hydrophobic Binding Pocket of Hsp90 von Shin, Sang Chul, El-Damasy, Ashraf K, Lee, Ju Hyeon, Seo, Seon Hee, Kim, Ji Hyun, Seo, Young Ho, Lee, Yuri, Yu, Ji Hoon, Bang, Eun Kyoung, Kim, Eunice EunKyeong, Keum, Gyochang

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Design and Synthesis of New 4-(3,4,5-Trimethoxyphenyl)Thiazole-Pyrimidine Derivatives as Potential Antiproliferative Agents von El-Damasy, Ashraf K, Jin, Heewon, Sabry, Mohamed A, Kim, Hyun Ji, Alanazi, Mohammed M, Seo, Seon Hee, Bang, Eun-Kyoung, Keum, Gyochang

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Sulfur(vi) fluoride exchange as a key reaction for synthesizing biaryl sulfate core derivatives as potent hepatitis C virus NS5A inhibitors and their structure-activity relationshi... von You, Youngsu, Kim, Hee Sun, Park, Jung Woo, Keum, Gyochang, Jang, Sung Key, Kim, B Moon

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A novel tropomyosin-related kinase A inhibitor, KK5101 to treat pancreatic cancer von Fang, Zhenghuan, Han, Boreum, Jung, Kyung Hee, Lee, Ju-Hyeon, El-Damasy, Ashraf Kareem, Gadhe, Changdev G., Kim, Soo Jung, Yan, Hong Hua, Park, Jung Hee, Lee, Ji Eun, Kang, Yeo Wool, Pae, Ae Nim, Keum, Gyochang, Hong, Soon-Sun

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Analyzing immune responses to varied mRNA and protein vaccine sequences von Park, Hyeong-Jun, Bang, Yoo-Jin, Kwon, Sung Pil, Kwak, Woori, Park, Sang-In, Roh, Gahyun, Bae, Seo-Hyeon, Kim, Jae-Yong, Kwak, Hye Won, Kim, Yongkwan, Yoo, Soyeon, Kim, Daegeun, Keum, Gyochang, Bang, Eun-Kyoung, Hong, So-Hee, Nam, Jae-Hwan

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Synthesis and in Vitro Evaluation of the Antitubercular and Antibacterial Activity of Novel Oxazolidinones Bearing Octahydrocyclopenta[c]pyrrol-2-yl Moieties von Bhattarai, Deepak, Lee, Ju-hyeon, Seo, Seon Hee, Nam, Ghilsoo, Choo, Hyunah, Kang, Soon Bang, Kwak, Jin-Hwan, Oh, Taegwon, Cho, Sang-Nae, Pae, Ae Nim, Kim, Eunice Eunkyeong, Jeong, Nakcheol, Keum, Gyochang

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A lipid nanoparticle platform incorporating trehalose glycolipid for exceptional mRNA vaccine safety von Bae, Seo-Hyeon, Yoo, Soyeon, Lee, Jisun, Park, Hyo-Jung, Kwon, Sung Pil, Jin, Harin, Park, Sang-In, Lee, Yu-Sun, Bang, Yoo-Jin, Roh, Gahyun, Lee, Seonghyun, Youn, Sue Bean, Kim, In Woo, Oh, Ho Rim, El-Damasy, Ashraf K., Keum, Gyochang, Kim, Hojun, Youn, Hyewon, Nam, Jae-Hwan, Bang, Eun-Kyoung

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Oxazolopyridines and thiazolopyridines as monoamine oxidase B inhibitors for the treatment of Parkinson’s disease von Park, Hye Ri, Kim, Jiyoon, Kim, Taekeun, Jo, Seonmi, Yeom, Miyoung, Moon, Bongjin, Choo, Il Han, Lee, Jaeick, Lim, Eun Jeong, Park, Ki Duk, Min, Sun-Joon, Nam, Ghilsoo, Keum, Gyochang, Lee, C. Justin, Choo, Hyunah

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