A general model for predicting the binding affinity of reversibly and irreversibly dimerized ligands von Foreman, Kenneth W

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Structural and functional profiling of the human histone methyltransferase SMYD3 von Foreman, Kenneth W, Brown, Mark, Park, Frances, Emtage, Spencer, Harriss, June, Das, Chhaya, Zhu, Li, Crew, Andy, Arnold, Lee, Shaaban, Salam, Tucker, Philip

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Binding of Inhibitors to Nuclear Localization Signal Peptide from Venezuelan Equine Encephalitis Virus Capsid Protein Explored with All-Atom Replica Exchange Molecular Dynamics von Delfing, Bryan M., Laracuente, Xavier E., Luo, Xingyu, Olson, Audrey, Jeffries, William, Foreman, Kenneth W., Paige, Mikell, Kehn-Hall, Kylene, Lockhart, Christopher, Klimov, Dmitri K.

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Reversible linkage of two distinct small molecule inhibitors of Myc generates a dimeric inhibitor with improved potency that is active in myc over-expressing cancer cell lines von Wanner, Jutta, Romashko, Darlene, Werner, Douglas S, May, Earl W, Peng, Yue, Schulz, Ryan, Foreman, Kenneth W, Russo, Suzanne, Arnold, Lee D, Pingle, Maneesh, Bergstrom, Donald E, Barany, Francis, Thomson, Stuart

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Small-molecule inhibition and activation-loop trans-phosphorylation of the IGF1 receptor von Wu, Jinhua, Li, Wanqing, Craddock, Barbara P, Foreman, Kenneth W, Mulvihill, Mark J, Ji, Qun-sheng, Miller, W Todd, Hubbard, Stevan R

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Binding of viral nuclear localization signal peptides to importin-α nuclear transport protein von Delfing, Bryan M, Laracuente, Xavier E, Olson, Audrey, Foreman, Kenneth W, Paige, Mikell, Kehn-Hall, Kylene, Lockhart, Christopher, Klimov, Dmitri K

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Binding of Venezuelan Equine Encephalitis Virus Inhibitors to Importin‑α Receptors Explored with All-Atom Replica Exchange Molecular Dynamics von Delfing, Bryan M., Olson, Audrey, Laracuente, Xavier E., Foreman, Kenneth W., Paige, Mikell, Kehn-Hall, Kylene, Lockhart, Christopher, Klimov, Dmitri K.

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Novel, Self-Assembling Dimeric Inhibitors of Human β Tryptase von Giardina, Sarah F, Werner, Douglas S, Pingle, Maneesh, Feinberg, Philip B, Foreman, Kenneth W, Bergstrom, Donald E, Arnold, Lee D, Barany, Francis

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Can Free Energy Perturbation Simulations Coupled with Replica-Exchange Molecular Dynamics Study Ligands with Distributed Binding Sites? von Lockhart, Christopher, Luo, Xingyu, Olson, Audrey, Delfing, Bryan M., Laracuente, Xavier E., Foreman, Kenneth W., Paige, Mikell, Kehn-Hall, Kylene, Klimov, Dmitri K.

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Competitive Binding of Viral Nuclear Localization Signal Peptide and Inhibitor Ligands to Importin‑α Nuclear Transport Protein von Delfing, Bryan M., Laracuente, Xavier E., Jeffries, William, Luo, Xingyu, Olson, Audrey, Foreman, Kenneth W., Petruncio, Greg, Lee, Kyung Hyeon, Paige, Mikell, Kehn-Hall, Kylene, Lockhart, Christopher, Klimov, Dmitri K.

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Substrate-dependent modulation of the leukotriene A4 hydrolase aminopeptidase activity and effect in a murine model of acute lung inflammation von Lee, Kyung Hyeon, Ali, Nadia Fazal, Lee, Soo Hyeon, Zhang, Zhimin, Burdick, Marie, Beaulac, Zachary J., Petruncio, Greg, Li, Linxia, Xiang, Jiangdong, Chung, Ezra M., Foreman, Kenneth W., Noble, Schroeder M., Shim, Yun M., Paige, Mikell

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Target-Directed Self-Assembly of Homodimeric Drugs Against β‑Tryptase von Giardina, Sarah F, Werner, Douglas S, Pingle, Maneesh, Foreman, Kenneth W, Bergstrom, Donald E, Arnold, Lee D, Barany, Francis

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Minimal Theoretical Description of Magnesium Halogen Exchanges von Pham, Anh D. H., Bui, Johnny, Foreman, Kenneth W.

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Combinatorial synthesis of substituted 3-(2-indolyl)piperidines and 2-phenyl indoles as inhibitors of ZipA–FtsZ interaction von Jennings, Lee D., Foreman, Kenneth W., Rush, Thomas S., Tsao, Desiree H.H., Mosyak, Lidia, Kincaid, Scott L., Sukhdeo, Mohani N., Sutherland, Alan G., Ding, Weidong, Kenny, Cynthia Hess, Sabus, Chantel L., Liu, Hanlan, Dushin, Elizabeth G., Moghazeh, Soraya L., Labthavikul, Pornpen, Petersen, Peter J., Tuckman, Margareta, Ruzin, Alexey V.

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Substrate-dependent modulation of the leukotriene A 4 hydrolase aminopeptidase activity and effect in a murine model of acute lung inflammation von Lee, Kyung Hyeon, Ali, Nadia Fazal, Lee, Soo Hyeon, Zhang, Zhimin, Burdick, Marie, Beaulac, Zachary J, Petruncio, Greg, Li, Linxia, Xiang, Jiangdong, Chung, Ezra M, Foreman, Kenneth W, Noble, Schroeder M, Shim, Yun M, Paige, Mikell

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Abstract B43: Reversible linkage of two distinct small molecule inhibitors of MYC generates a more potent and selective dimeric inhibitor that is active in cancer cell lines over-e... von Wanner, Jutta, Romashko, Darlene, Werner, Douglas S., May, Earl W., Peng, Yue, Schulz, Ryan, Foreman, Kenneth W., Russo, Suzanne, Arnold, Lee D., Pingle, Maneesh, Bergstrom, Donald E., Barany, Francis, Thomson, Stuart

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Silicon based drug conjugates and methods of using same von NGUYEN, Hanh Nho, OFORI, Leslie Odame, WANNER, Jutta, WERNER, Douglas S, FOREMAN, Kenneth W

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SILICON BASED DRUG CONJUGATES AND METHODS OF USING SAME von Wanner, Jutta, Werner, Douglas S, Foreman, Kenneth W, Nguyen, Hanh Nho, Ofori, Leslie Odame

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Silicon based drug conjugates and methods of using same von Wanner, Jutta, Werner, Douglas S, Foreman, Kenneth W, Nguyen, Hanh N, Ofori, Leslie O

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Corrigendum to “Combinatorial synthesis of substituted 3-(2-indolyl)piperidines and 2-phenyl indoles as inhibitors of ZipA–FtsZ interaction” [Bioorg. Med. Chem. 12 (2004) 5115–5131... von Jennings, Lee D., Foreman, Kenneth W., Rush, Thomas S., Tsao, Desiree H.H., Mosyak, Lidia, Kincaid, Scott L., Sukhdeo, Mohani N., Sutherland, Alan G., Ding, Weidong, Kenny, Cynthia Hess, Sabus, Chantel L., Liu, Hanlan, Dushin, Elizabeth G., Moghazeh, Soraya L., Labthavikul, Pornpen, Petersen, Peter J., Tuckman, Margareta, Haney, Steven A., Ruzin, Alexey V.

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