Synthesis of Versatile Chiral N,P Ligands Derived from Pyridine and Quinoline von Drury III, William J., Zimmermann, Nicole, Keenan, Martine, Hayashi, Masahiko, Kaiser, Stefan, Goddard, Richard, Pfaltz, Andreas

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The Tethered Aminohydroxylation (TA) of Cyclic Allylic Carbamates von Donohoe, Timothy J, Johnson, Peter D, Cowley, Andrew, Keenan, Martine

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Enantioselective Heck reactions using chiral P,N-ligands von Loiseleur, Olivier, Hayashi, Masahiko, Keenan, Martine, Schmees, Norbert, Pfaltz, Andreas

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The regioselective aminohydroxylation of allylic carbamates von Donohoe, T J, Johnson, P D, Helliwell, M, Keenan, M

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Complexes of Trypanosoma cruzi sterol 14α-demethylase (CYP51) with two pyridine-based drug candidates for Chagas disease: structural basis for pathogen selectivity von Hargrove, Tatiana Y, Wawrzak, Zdzislaw, Alexander, Paul W, Chaplin, Jason H, Keenan, Martine, Charman, Susan A, Perez, Catherine J, Waterman, Michael R, Chatelain, Eric, Lepesheva, Galina I

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Short-course combination treatment for experimental chronic Chagas disease von González, Silvia, Wall, Richard J, Thomas, John, Braillard, Stephanie, Brunori, Gino, Camino Díaz, Isabel, Cantizani, Juan, Carvalho, Sandra, Castañeda Casado, Pablo, Chatelain, Eric, Cotillo, Ignacio, Fiandor, Jose M, Francisco, Amanda Fortes, Grimsditch, David, Keenan, Martine, Kelly, John M, Kessler, Albane, Luise, Chiara, Lyon, Jon J, MacLean, Lorna, Marco, Maria, Martin, J Julio, Martinez Martinez, Maria S, Paterson, Christy, Read, Kevin D, Santos-Villarejo, Angel, Zuccotto, Fabio, Wyllie, Susan, Miles, Tim J, De Rycker, Manu

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Boron-based drugs as antiprotozoals von Jacobs, Robert T, Plattner, Jacob J, Keenan, Martine

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DNDI-6174 is a preclinical candidate for visceral leishmaniasis that targets the cytochrome bc1 von Braillard, Stéphanie, Keenan, Martine, Breese, Karen J, Heppell, Jacob, Abbott, Michael, Islam, Rafiqul, Shackleford, David M, Katneni, Kasiram, Crighton, Elly, Chen, Gong, Patil, Rahul, Lee, Given, White, Karen L, Carvalho, Sandra, Wall, Richard J, Chemi, Giulia, Zuccotto, Fabio, González, Silvia, Marco, Maria, Deakyne, Julianna, Standing, David, Brunori, Gino, Lyon, Jonathan J, Castañeda-Casado, Pablo, Camino, Isabel, Martinez Martinez, Maria S, Zulfiqar, Bilal, Avery, Vicky M, Feijens, Pim-Bart, Van Pelt, Natascha, Matheeussen, An, Hendrickx, Sarah, Maes, Louis, Caljon, Guy, Yardley, Vanessa, Wyllie, Susan, Charman, Susan A, Chatelain, Eric

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Re-evaluating pretomanid analogues for Chagas disease: Hit-to-lead studies reveal both in vitro and in vivo trypanocidal efficacy von Thompson, Andrew M., O’Connor, Patrick D., Marshall, Andrew J., Francisco, Amanda F., Kelly, John M., Riley, Jennifer, Read, Kevin D., Perez, Catherine J., Cornwall, Scott, Thompson, R.C. Andrew, Keenan, Martine, White, Karen L., Charman, Susan A., Zulfiqar, Bilal, Sykes, Melissa L., Avery, Vicky M., Chatelain, Eric, Denny, William A.

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Re-evaluating pretomanid analogues for Chagas disease: Hit-to-lead studies reveal both in vitro and in vivo trypanocidal efficacy von Thompson, Andrew M, O'Connor, Patrick D, Marshall, Andrew J, Francisco, Amanda F, Kelly, John M, Riley, Jennifer, Read, Kevin D, Perez, Catherine J, Cornwall, Scott, Thompson, RC Andrew, Keenan, Martine, White, Karen L, Charman, Susan A, Zulfiqar, Bilal, Sykes, Melissa L, Avery, Vicky M, Chatelain, Eric, Denny, William A

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Analogues of Fenarimol Are Potent Inhibitors of Trypanosoma cruzi and Are Efficacious in a Murine Model of Chagas Disease von Keenan, Martine, Abbott, Michael J, Alexander, Paul W, Armstrong, Tanya, Best, Wayne M, Berven, Bradley, Botero, Adriana, Chaplin, Jason H, Charman, Susan A, Chatelain, Eric, von Geldern, Thomas W, Kerfoot, Maria, Khong, Andrea, Nguyen, Tien, McManus, Joshua D, Morizzi, Julia, Ryan, Eileen, Scandale, Ivan, Thompson, R. Andrew, Wang, Sen Z, White, Karen L

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Two Analogues of Fenarimol Show Curative Activity in an Experimental Model of Chagas Disease von Keenan, Martine, Chaplin, Jason H, Alexander, Paul W, Abbott, Michael J, Best, Wayne M, Khong, Andrea, Botero, Adriana, Perez, Catherine, Cornwall, Scott, Thompson, R. Andrew, White, Karen L, Shackleford, David M, Koltun, Maria, Chiu, Francis C. K, Morizzi, Julia, Ryan, Eileen, Campbell, Michael, von Geldern, Thomas W, Scandale, Ivan, Chatelain, Eric, Charman, Susan A

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Highly efficient and flexible total synthesis of coelenterazine von Keenan, Martine, Jones, Keith, Hibbert, Frank

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New facile and mild synthesis of 2-substituted oxazolopyridines von Heuser, Stefan, Keenan, Martine, Weichert, Andreas G.

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Complexes of Trypanosoma cruzi Sterol 14α-Demethylase (CYP51) with Two Pyridine-based Drug Candidates for Chagas Disease von Hargrove, Tatiana Y., Wawrzak, Zdzislaw, Alexander, Paul W., Chaplin, Jason H., Keenan, Martine, Charman, Susan A., Perez, Catherine J., Waterman, Michael R., Chatelain, Eric, Lepesheva, Galina I.

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Design, structure–activity relationship and in vivo efficacy of piperazine analogues of fenarimol as inhibitors of Trypanosoma cruzi von Keenan, Martine, Alexander, Paul W., Diao, Hugo, Best, Wayne M., Khong, Andrea, Kerfoot, Maria, Thompson, R. C. Andrew, White, Karen L., Shackleford, David M., Ryan, Eileen, Gregg, Alison D., Charman, Susan A., von Geldern, Thomas W., Scandale, Ivan, Chatelain, Eric

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Contra-Friedel-Crafts tert-butylation of substituted aromatic rings via directed metallation and sulfinylation von Clayden, Jonathan, Stimson, Christopher C, Keenan, Martine

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Asymmetric Ortholithiation of Amides by Conformationally Mediated Chiral Memory: An Enantioselective Route to Naphtho- and Benzofuranones von Clayden, Jonathan, Stimson, Christopher C., Keenan, Martine

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Efficient Acyclic Stereocontrol Using the Tethered Aminohydroxylation Reaction von Donohoe, Timothy J, Johnson, Peter D, Pye, Richard J, Keenan, Martine

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Concise and Enantioselective Synthesis of the Aminocyclitol Core of Hygromycin A von Donohoe, Timothy J, Johnson, Peter D, Pye, Richard J, Keenan, Martine

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