Enantioselective Synthesis of 4′-Ethynyl-2-fluoro-2′-deoxyadenosine (EFdA) via Enzymatic Desymmetrization von McLaughlin, Mark, Kong, Jongrock, Belyk, Kevin M, Chen, Billy, Gibson, Andrew W, Keen, Stephen P, Lieberman, David R, Milczek, Erika M, Moore, Jeffrey C, Murray, David, Peng, Feng, Qi, Ji, Reamer, Robert A, Song, Zhiguo J, Tan, Lushi, Wang, Lin, Williams, Michael J

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Enantioselective Synthesis of β‑Aryloxycarboxylic Esters via Asymmetric Hydrogenation of β‑Aryloxy-α,β-Unsaturated Esters von Stewart, Gavin W, Shevlin, Michael, Yamagata, Adam D. Gammack, Gibson, Andrew W, Keen, Stephen P, Scott, Jeremy P

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Process Development of the HCV NS5B Site D Inhibitor MK-8876 von Williams, Michael J, Chen, Qinghao, Codan, Lorenzo, Dermenjian, Renee K, Dreher, Spencer, Gibson, Andrew W, He, Xianliang, Jin, Yan, Keen, Stephen P, Lee, Alfred Y, Lieberman, David R, Lin, Wei, Liu, Guiquan, McLaughlin, Mark, Reibarkh, Mikhail, Scott, Jeremy P, Strickfuss, Sophie, Tan, Lushi, Varsolona, Richard J, Wen, Feng

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Development of a Fit-for-Purpose Large-Scale Synthesis of an Oral PARP Inhibitor von Wallace, Debra J, Baxter, Carl A, Brands, Karel J. M, Bremeyer, Nadine, Brewer, Sarah E, Desmond, Richard, Emerson, Khateeta M, Foley, Jennifer, Fernandez, Paul, Hu, Weifeng, Keen, Stephen P, Mullens, Peter, Muzzio, Daniel, Sajonz, Peter, Tan, Lushi, Wilson, Robert D, Zhou, George, Zhou, Guoyue

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Process Development and Large-Scale Synthesis of a c-Met Kinase Inhibitor von Stewart, Gavin W, Brands, Karel M. J, Brewer, Sarah E, Cowden, Cameron J, Davies, Antony J, Edwards, John S, Gibson, Andrew W, Hamilton, Simon E, Katz, Jason D, Keen, Stephen P, Mullens, Peter R, Scott, Jeremy P, Wallace, Debra J, Wise, Christopher S

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Practical Asymmetric Synthesis of a γ-Secretase Inhibitor Exploiting Substrate-Controlled Intramolecular Nitrile Oxide−Olefin Cycloaddition von Scott, Jeremy P, Oliver, Steven F, Brands, Karel M. J, Brewer, Sarah E, Davies, Antony J, Gibb, Andrew D, Hands, David, Keen, Stephen P, Sheen, Faye J, Reamer, Robert A, Wilson, Robert D, Dolling, Ulf-H

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Stereoselective Total Syntheses and Reassignment of Stereochemistry of the Freshwater Cyanobacterial Hepatotoxins Cylindrospermopsin and 7-Epicylindrospermopsin von Heintzelman, Geoffrey R, Fang, Wen-Kui, Keen, Stephen P, Wallace, Grier A, Weinreb, Steven M

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Stereoselective Total Synthesis of the Cyanobacterial Hepatotoxin 7-Epicylindrospermopsin:  Revision of the Stereochemistry of Cylindrospermopsin von Heintzelman, Geoffrey R, Fang, Wen-Kui, Keen, Stephen P, Wallace, Grier A, Weinreb, Steven M

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Process Development of a Tricyclic Diazepine-Based IDH1 Mutant Inhibitor von Maddess, Matthew L., Cleator, Ed, Morimoto, Mariko, Goodyear, Adrian, Dieguez-Vazquez, Alejandro, Gibb, Andrew, Kirtley, Andy, Christensen, Melodie, Song, Chaohui, Peng, Feng, Alam, Mahbub, Keen, Stephen P., Oliver, Steven F.

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Studies on total synthesis of cylindrospermopsin: new constructions of uracils from α,β-unsaturated esters von Keen, Stephen P, Weinreb, Steven M

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Studies on the Synthesis of Pinnaic Acid and Halichlorine. Stereoselective Preparation of a (Z)-δ-Chloro-γ,δ-unsaturated-β-keto Phosphonate as a Side Chain Synthon von Keen, Stephen P, Weinreb, Steven M

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Practical Asymmetric Synthesis of a Non-Peptidic αvβ3 Antagonist von Keen, Stephen P, Cowden, Cameron J, Bishop, Brian C, Brands, Karel M. J, Davies, Antony J, Dolling, Ulf H, Lieberman, David R, Stewart, Gavin W

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Cross metathesis of the amino acid homoallylglycine von Gibson (née Thomas), Susan E., Gibson, Vernon C., Keen, Stephen P.

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Practical Asymmetric Synthesis of a Non-Peptidic α v β 3 Antagonist von Keen, Stephen P., Cowden, Cameron J., Bishop, Brian C., Brands, Karel M. J., Davies, Antony J., Dolling, Ulf H., Lieberman, David R., Stewart, Gavin W.

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Practical asymmetric synthesis of a non-peptidic alphavbeta3 antagonist von Keen, Stephen P, Cowden, Cameron J, Bishop, Brian C, Brands, Karel M J, Davies, Antony J, Dolling, Ulf H, Lieberman, David R, Stewart, Gavin W

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Cross-metathesis of unsaturated α-amino acid derivatives von Biagini, Stefano C. G., GibsonéThomas, Susan E., Keen, Stephen P.

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ChemInform Abstract: Enantioselective Synthesis of β-Aryloxycarboxylic Esters via Asymmetric Hydrogenation of β-Aryloxy-α,β-unsaturated Esters von Stewart, Gavin W., Shevlin, Michael, Yamagata, Adam D. Gammack, Gibson, Andrew W., Keen, Stephen P., Scott, Jeremy P.

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ChemInform Abstract: Enantioselective Synthesis of [beta]-Aryloxycarboxylic Esters via Asymmetric Hydrogenation of [beta]-Aryloxy-[alpha],[beta]-unsaturated Esters von Stewart, Gavin W, Shevlin, Michael, Yamagata, Adam D. Gammack, Gibson, Andrew W, Keen, Stephen P, Scott, Jeremy P

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ChemInform Abstract: Total Synthesis of Cylindrospermopsin: New Constructions of Uracils from α,β-Unsaturated Esters von Keen, Stephen P., Weinreb, Steven M.

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Enantioselective Synthesis of 13-Oxotricyclo[8.2.1.0. 3,8] Trideca-3(8),4,6-Triene-5-Carboxylates von STEWART GAVIN W, KEEN STEPHEN P, OLIVER STEVEN F

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