Synthesis of New 26,27-Difluoro- and 26,26,27,27-Tetrafluoro-25-hydroxyvitamin D3: Effects of Terminal Fluorine Atoms on Biological Activity and Half-life von Kawagoe, Fumihiro, Mototani, Sayuri, Yasuda, Kaori, Mano, Hiroki, Takeuchi, Akiko, Saitoh, Hiroshi, Sakaki, Toshiyuki, Kittaka, Atsushi

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The First Convergent Synthesis of 23,23-Difluoro-25-hydroxyvitamin D3 and Its 24-Hydroxy Derivatives: Preliminary Assessment of Biological Activities von Mototani, Sayuri, Kawagoe, Fumihiro, Yasuda, Kaori, Mano, Hiroki, Sakaki, Toshiyuki, Kittaka, Atsushi

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Efficient Stereo-Selective Fluorination on Vitamin D3 Side-Chain Using Electrophilic Fluorination von Kawagoe, Fumihiro, Mototani, Sayuri, Kittaka, Atsushi

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Introduction of fluorine atoms to vitamin D3 side-chain and synthesis of 24,24-difluoro-25-hydroxyvitamin D3 von Kawagoe, Fumihiro, Mototani, Sayuri, Yasuda, Kaori, Nagasawa, Kazuo, Uesugi, Motonari, Sakaki, Toshiyuki, Kittaka, Atsushi

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The Synthesis and Biological Evaluation of D-Ring-Modified Vitamin D Analogues von Kawagoe, Fumihiro, Mototani, Sayuri, Kittaka, Atsushi

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Elucidation of metabolic pathways of 25-hydroxyvitamin D3 mediated by CYP24A1 and CYP3A using Cyp24a1 knockout rats generated by CRISPR/Cas9 system von Yasuda, Kaori, Nishikawa, Miyu, Okamoto, Kairi, Horibe, Kyohei, Mano, Hiroki, Yamaguchi, Mana, Okon, Risa, Nakagawa, Kimie, Tsugawa, Naoko, Okano, Toshio, Kawagoe, Fumihiro, Kittaka, Atsushi, Ikushiro, Shinichi, Sakaki, Toshiyuki

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Concise synthesis of 23-hydroxylated vitamin D3 metabolites von Kawagoe, Fumihiro, Sugiyama, Toru, Yasuda, Kaori, Uesugi, Motonari, Sakaki, Toshiyuki, Kittaka, Atsushi

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Synthesis and CYP24A1-Dependent Metabolism of 23-Fluorinated Vitamin D3 Analogues von Kawagoe, Fumihiro, Yasuda, Kaori, Mototani, Sayuri, Sugiyama, Toru, Uesugi, Motonari, Sakaki, Toshiyuki, Kittaka, Atsushi

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Chemistry of fluorinated vitamin D derivatives von Kawagoe, Fumihiro, Kittaka, Atsushi

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Design and Synthesis of Fluoro Analogues of Vitamin D von Kawagoe, Fumihiro, Mototani, Sayuri, Kittaka, Atsushi

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An Efficient Route to Benzene and Phenol Derivatives via Ring-Closing Olefin Metathesis von Yoshida, Kazuhiro, Horiuchi, Shingo, Iwadate, Noriyuki, Kawagoe, Fumihiro, Imamoto, Tsuneo

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Efficient Stereo-Selective Fluorination on Vitamin D[sub.3] Side-Chain Using Electrophilic Fluorination von Kawagoe, Fumihiro, Mototani, Sayuri, Kittaka, Atsushi

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Ring-Closing Olefin Metathesis for the Synthesis of Benzene Derivatives von Yoshida, Kazuhiro, Kawagoe, Fumihiro, Iwadate, Noriyuki, Takahashi, Hidetoshi, Imamoto, Tsuneo

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An Improved and Scalable Synthesis of the Potent SREBP Inhibitor KK-052 via [3+2] Cycloaddition von Kawagoe, Fumihiro, Mototani, Sayuri, Takemoto, Yasushi, Uesugi, Motonari, Kittaka, Atsushi

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Efficient Stereo-Selective Fluorination on Vitamin D 3 Side-Chain Using Electrophilic Fluorination von Kawagoe, Fumihiro, Mototani, Sayuri, Kittaka, Atsushi

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Synthesis of (22R)‑, (22S)‑22-Fluoro‑, and 22,22-Difluoro-25-hydroxyvitamin D3 and Effects of Side-Chain Fluorination on Biological Activity and CYP24A1-Dependent Metabolism von Kawagoe, Fumihiro, Mototani, Sayuri, Yasuda, Kaori, Takeuchi, Akiko, Mano, Hiroki, Kakuda, Shinji, Saitoh, Hiroshi, Sakaki, Toshiyuki, Kittaka, Atsushi

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Recent developments for introducing a hexafluoroisopropanol unit into the Vitamin D side chain von Kawagoe, Fumihiro, Sugiyama, Toru, Uesugi, Motonari, Kittaka, Atsushi

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Synthesis of (22 R )-, (22 S )-22-Fluoro-, and 22,22-Difluoro-25-hydroxyvitamin D 3 and Effects of Side-Chain Fluorination on Biological Activity and CYP24A1-Dependent Metabolism von Kawagoe, Fumihiro, Mototani, Sayuri, Yasuda, Kaori, Takeuchi, Akiko, Mano, Hiroki, Kakuda, Shinji, Saitoh, Hiroshi, Sakaki, Toshiyuki, Kittaka, Atsushi

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Stereoselective Synthesis of 24-Fluoro-25-Hydroxyvitamin D3 Analogues and Their Stability to hCYP24A1-Dependent Catabolism von Kawagoe, Fumihiro, Mototani, Sayuri, Yasuda, Kaori, Mano, Hiroki, Sakaki, Toshiyuki, Kittaka, Atsushi

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Synthesis of new 26,27-difluoro- and 26,26,27,27-tetrafluoro-25-hydroxyvitamin D 3 : Effects of terminal fluorine atoms on biological activity and half-life von Kawagoe, Fumihiro, Mototani, Sayuri, Yasuda, Kaori, Mano, Hiroki, Takeuchi, Akiko, Saitoh, Hiroshi, Sakaki, Toshiyuki, Kittaka, Atsushi

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