M1 agonists for the treatment of Alzheimer's disease. Novel properties and clinical update von Fisher, A, Heldman, E, Gurwitz, D, Haring, R, Karton, Y, Meshulam, H, Pittel, Z, Marciano, D, Brandeis, R, Sadot, E, Barg, Y, Pinkas-Kramarski, R, Vogel, Z, Ginzburg, I, Treves, T A, Verchovsky, R, Klimowsky, S, Korczyn, A D

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Amyloid Precursor Protein Secretion via Muscarinic Receptors: Reduced Desensitization Using the M1-Selective Agonist AF102B von Haring, R., Gurwitz, D., Barg, J., Pinkaskramarski, R., Heldman, E., Pittel, Z., Wengier, A., Meshulam, H., Marciano, D., Karton, Y., Fisher, A.

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NGF Promotes Amyloid Precursor Protein Secretion via Muscarinic Receptor Activation von Haring, R., Gurwitz, D., Barg, J., Pinkaskramarski, R., Heldman, E., Pittel, Z., Danenberg, H.D., Wengier, A., Meshulam, H., Marciano, D., Karton, Y., Fisher, A.

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Selective site controlled nucleophilic attacks in 5-membered ring phosphate esters: unusual C-O vs. common P-O bond cleavage von Ashkenazi, Nissan, Zade, Sanjio S, Segall, Yoffi, Karton, Yishai, Bendikov, Michael

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Nucleophilic transformations of cyclic phosphate triesters von Ashkenazi, Nissan, Karton, Yishai, Segall, Yoffi

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Stereoselectivity toward VX Is Determined by Interactions with Residues of the Acyl Pocket as Well as of the Peripheral Anionic Site of AChE von Ordentlich, Arie, Barak, Dov, Sod-Moriah, Gali, Kaplan, Dana, Mizrahi, Dana, Segall, Yoffi, Kronman, Chanoch, Karton, Yishai, Lazar, Arie, Marcus, Dino, Velan, Baruch, Shafferman, Avigdor

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The role of AChE active site gorge in determining stereoselectivity of charged and noncharged VX enantiomers von Ordentlich, Arie, Barak, Dov, Sod-Moriah, Gali, Kaplan, Dana, Mizrahi, Dana, Segall, Yoffi, Kronman, Chanoch, Karton, Yishai, Lazar, Arie, Marcus, Dino, Velan, Baruch, Shafferman, Avigdor

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Synthesis and Biological Activities of Flavonoid Derivatives as A3 Adenosine Receptor Antagonists von Karton, Yishai, Jiang, Ji-long, Ji, Xiao-duo, Melman, Neli, Olah, Mark E, Stiles, Gary L, Jacobson, Kenneth A

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M1 Agonists for the Treatment of Alzheimer's Disease: Novel Properties and Clinical Updatea von Fisher, A, Heldman, E, Gurwitz, D, Haring, R, KARTON, Y, Meshulam, H, Pittel, Z, Marciano, D, Brandeis, R, SADOT, E, Barg, Y, Pinkas-Kramarski, R, Vogel, Z, Ginzburg, I, Treves, T A, Verchovsky, R, KLIMOWSKY, S, Korczyn, Ad

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Structure-activity relationships of 8-styrylxanthines as A2-selective adenosine antagonists von Jacobson, Kenneth A, Gallo-Rodriguez, Carola, Melman, Neli, Fischer, Bilha, Maillard, Michel, van Bergen, Andrew, van Galen, Philip J. M, Karton, Yishai

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NGF-dependent neurotrophic-like effects of AF102B, an M1 muscarinic agonist, in PC12M1 cells von GURWITZ, D, HARING, R, PINKAS-KRAMARSKI, R, STEIN, R, HELDMAN, E, KARTON, Y, FISHER, A

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Novel m1 muscarinic agonists in treatment and delaying the progression of Alzheimer's disease: An unifying hypothesis von Fisher, Abraham, Brandeis, Rachel, Haring, Rachel, Eshhar, Naomi, Heldman, Eliahu, Karton, Yishai, Eisenberg, Orli, Meshulam, Haim, Marciano, Daniele, Bar-Ner, Nira, Pittel, Zipora

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NGF-dependent neurotrophic-like effects of AF102B, an M1 muscarinic agonist, in PC12M1 cells von Gurwitz, D, Haring, R, Pinkas-Kramarski, R, Stein, R, Heldman, E, Karton, Y, Fisher, A

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Selective signaling via unique M1 muscarinic agonists von Fisher, A, Heldman, E, Gurwitz, D, Haring, R, Barak, D, Meshulam, H, Marciano, D, Brandeis, R, Pittel, Z, Segal, M

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Functionalized congener approach to muscarinic antagonists: analogs of pirenzepine von Karton, Yishai, Bradbury, Barton J, Baumgold, Jesse, Paek, Robert, Jacobson, Kenneth A

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Acyl-hydrazide derivatives of a xanthine carboxylic congener (XCC) as selective antagonists at human A2B adenosine receptors von Kim, Yong-Chul, Karton, Yishai, Ji, Xiao-duo, Melman, Neli, Linden, Joel, Jacobson, Kenneth A.

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Synthesis and biological activities of flavonoid derivatives as A sub(3) adenosine receptor antagonists von Karton, Y, Jiang, J, Ji, X, Melman, N, Olah, ME, Stiles, G L, Jacobson, KA

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192 Novel m1 muscarinic agonists: From symptomatic treatment to delaying the progression of Alzheimer's disease (AD) von Fisher, A., Haring, R., Ginzburg, I., Sadot, E., Pittel, Z., Barg, Y., Behar, L., Gunwitz, D., Karton, Y., Meshulam, H., Marciano, D., Brandeis, R., Heldman, E.

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Molecular probes for muscarinic receptors: derivatives of the M1-antagonist telenzepine von Karton, Yishai, Baumgold, Jesse, Handen, Jeffrey S, Jacobson, Kenneth A

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High affinity acylating antagonists for muscarinic receptors von Baumgold, Jesse, Karton, Yishai, Malka, Naftali, Jacobson, Kenneth A.

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