Characterization of Prostaglandin G/H Synthase 1 and 2 in rat, dog, monkey, and human gastrointestinal tracts von Kargman, S, Charleson, S, Cartwright, M, Frank, J, Riendeau, D, Mancini, J, Evans, J, O'Neill, G

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Expression of prostaglandin G/H synthase-1 and -2 protein in human colon cancer von KARGMAN, S. L, O'NEILL, G. P, VICKERS, P. J, EVANS, J. F, MANCINI, J. A, JOTHY, S

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Expression of the cysteinyl leukotriene 1 receptor in normal human lung and peripheral blood leukocytes von FIGUEROA, David J, BREYER, Richard M, JONES, Thomas R, LYNCH, Kevin R, AUSTIN, Christopher P, EVANS, Jilly F, DEFOE, Stephanie K, KARGMAN, Stacia, DAUGHERTY, Bruce L, WALDBURGER, Kristine, QINGYUN LIU, CLEMENTS, Michelle, ZHIZEN ZENG, O'NEILL, Gary P

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Receptor for Motilin Identified in the Human Gastrointestinal System von Feighner, Scott D., Tan, Carina P., McKee, Karen Kulju, Palyha, Oksana C., Hreniuk, Donna L., Pong, Sheng-Shung, Austin, Christopher P., Figueroa, David, MacNeil, Douglas, Cascieri, Margaret A., Nargund, Ravi, Bakshi, Raman, Abramovitz, Mark, Stocco, Rino, Kargman, Stacia, O'Neill, Gary, Lex H. T. Van Der Ploeg, Evans, Jilly, Patchett, Arthur A., Smith, Roy G., Howard, Andrew D.

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The discovery of rofecoxib, [MK 966, VIOXX ®, 4-(4′-methylsulfonylphenyl)-3-phenyl-2(5 H)-furanone], an orally active cyclooxygenase-2 inhibitor von Prasit, P, Wang, Z, Brideau, C, Chan, C.-C, Charleson, S, Cromlish, W, Ethier, D, Evans, J.F, Ford-Hutchinson, A.W, Gauthier, J.Y, Gordon, R, Guay, J, Gresser, M, Kargman, S, Kennedy, B, Leblanc, Y, Léger, S, Mancini, J, O'Neill, G.P, Ouellet, M, Percival, M.D, Perrier, H, Riendeau, D, Rodger, I, Tagari, P, Thérien, M, Vickers, P, Wong, E, Xu, L.-J, Young, R.N, Zamboni, R, Boyce, S, Rupniak, N, Forrest, M, Visco, D, Patrick, D

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Biochemical and pharmacological profile of a tetrasubstituted furanone as a highly selective COX‐2 inhibitor von Riendeau, D, Percival, M D, Boyce, S, Brideau, C, Charleson, S, Cromlish, W, Ethier, D, Evans, J, Falgueyret, J ‐P, Ford‐Hutchinson, A W, Gordon, R, Greig, G, Gresser, M, Guay, J, Kargman, S, Léger, S, Mancini, J A, O'Neill, G, Ouellet, M, Rodger, I W, Thérien, M, Wang, Z, Webb, J K, Wong, E, Xu, L, Young, R N, Zamboni, R, Prasit, P, Chan, C ‐C

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A human whole blood assay for clinical evaluation of biochemical efficacy of cyclooxygenase inhibitors von Brideau, C, Kargman, S, Liu, S, Dallob, A L, Ehrich, E W, Rodger, I W, Chan, C C

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Translocation of 5-lipoxygenase to the membrane in human leukocytes challenged with ionophore A23187 von Rouzer, C A, Kargman, S

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Overexpression of human prostaglandin G/H synthase-1 and -2 by recombinant vaccinia virus: inhibition by nonsteroidal anti-inflammatory drugs and biosynthesis of 15-hydroxyeicosate... von O'Neill, G P, Mancini, J A, Kargman, S, Yergey, J, Kwan, M Y, Falgueyret, J P, Abramovitz, M, Kennedy, B P, Ouellet, M, Cromlish, W

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Cloning of the cDNA for Human 5-lipoxygenase von Richard A. F. Dixon, Jones, Raymond E., Diehl, Ronald E., Bennett, Carl D., Kargman, Stacia, Rouzer, Carol A.

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From indomethacin to a selective COX-2 inhibitor: Development of indolalkanoic acids as potent and selective cyclooxygenase-2 inhibitors von Black, W.C., Bayly, C., Belley, M., Chan, C.-C., Charleson, S., Denis, D., Gauthier, J.Y., Gordon, R., Guay, D., Kargman, S., Lau, C.K., Leblanc, Y., Mancini, J., Ouellet, M., Percival, D., Roy, P., Skorey, K., Tagari, P., Vickers, P., Wong, E., Xu, L., Prasit, P.

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Characterization of the human cysteinyl leukotriene CysLT1 receptor von LYNCH, K. R, O'NEILL, G. P, CONNOLLY, B. M, CHANG BAI, AUSTIN, C. P, CHATEAUNEUF, A, STOCCO, R, GREIG, G. M, KARGMAN, S, HOOKS, S. B, HOSFIELD, E, WILLIAMS, D. L, QINGYUN LIU, FORD-HUTCHINSON, A. W, CASKEY, C. T, EVANS, J. F, IM, D.-S, SAWYER, N, METTERS, K. M, COULOMBE, N, ABRAMOVITZ, M, FIGUEROA, D. J, ZHIZHEN ZENG

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Correlation between expression of 5-lipoxygenase-activating protein, 5-lipoxygenase, and cellular leukotriene synthesis von Reid, G K, Kargman, S, Vickers, P J, Mancini, J A, Léveillé, C, Ethier, D, Miller, D K, Gillard, J W, Dixon, R A, Evans, J F

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Inhibition of cyclooxygenase-2 by rofecoxib attenuates the growth and metastatic potential of colorectal carcinoma in mice von MIN YAO, KARGMAN, Stacia, LAM, Eugene C, KELLY, Colleen R, YAXIN ZHENG, LUK, Pauline, KWONG, Elizabeth, EVANS, Jilly F, WOLFE, M. Michael

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Cytosolic phospholipase A2, cyclo-oxygenases and arachidonate in human stomach tumours von Soydan, A.S., Gaffen, J.D., Weech, P.K., Tremblay, N.M., Kargman, S., O'Neill, G., Bennett, A., Tavares, I.A.

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Translocation of HL-60 cell 5-lipoxygenase. Inhibition of A23187- or N-formyl-methionyl-leucyl-phenylalanine-induced translocation by indole and quinoline leukotriene synthesis inh... von KARGMAN, S, PRASIT, P, EVANS, J. F

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Studies on the Regulation, Biosynthesis, and Activation of 5-Lipoxygenase in Differentiated HL60 Cells von Kargman, S, Rouzer, C A

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Maintenance of Caspase-3 Proenzyme Dormancy by an Intrinsic "Safety Catch" Regulatory Tripeptide von Roy, Sophie, Bayly, Christopher I., Gareau, Yves, Houtzager, Vicky M., Kargman, Stacia, Sabina L. C. Keen, Rowland, Kathleen, Seiden, Isolde M., Thornberry, Nancy A., Nicholson, Donald W.

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A new series of selective COX-2 inhibitors: 5,6-diarylthiazolo[3,2-b][1,2,4]triazoles von Roy, P., Leblanc, Y., Ball, R.G., Brideau, C., Chan, C.C., Chauret, N., Cromlish, W., Ethier, D., Gauthier, J.Y., Gordon, R., Greig, G., Guay, J., Kargman, S., Lau, C.K., O'Neill, G., Silva, J., Thérien, M., van Staden, C., Wong, E., Xu, L., Prasit, P.

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Synthesis and biological evaluation of both enantiomers of L-761,000 as inhibitors of cyclooxygenase 1 and 2 von Leblanc, Y., Black, W.C., Chan, C.C., Charleson, S., Delorme, D., Denis, D., Gauthier, J.Y., Grimm, E.L., Gordon, R., Guay, D., Hamel, P., Kargman, S., Lau, C.K., Mancini, J., Ouellet, M., Percival, D., Roy, P., Skorey, K., Tagari, P., Vickers, P., Wong, E., Xu, L., Prasit, P.

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