Thrombospondin-1 Mimetic Peptide Inhibitors of Angiogenesis and Tumor Growth:  Design, Synthesis, and Optimization of Pharmacokinetics and Biological Activities von Haviv, Fortuna, Bradley, Michael F, Kalvin, Douglas M, Schneider, Andrew J, Davidson, Donald J, Majest, Sandra M, McKay, Laura M, Haskell, Catherine J, Bell, Randy L, Nguyen, Bach, Marsh, Kennan C, Surber, Bruce W, Uchic, John T, Ferrero, James, Wang, Yi-Chun, Leal, Juan, Record, Rae D, Hodde, Jason, Badylak, Stephen F, Lesniewski, Richard R, Henkin, Jack

Volltext

Structure−Activity Relationship Studies on N′-Aryl Carbohydrazide P2X7 Antagonists von Nelson, Derek W, Sarris, Kathy, Kalvin, Douglas M, Namovic, Marian T, Grayson, George, Donnelly-Roberts, Diana L, Harris, Richard, Honore, Prisca, Jarvis, Michael F, Faltynek, Connie R, Carroll, William A

Volltext

Novel and potent 3-(2,3-dichlorophenyl)-4-(benzyl)-4H-1,2,4-triazole P2X7 antagonists von CARROLL, William A, KALVIN, Douglas M, PEREZ MEDRANO, Arturo, FLORJANCIC, Alan S, YING WANG, DONNELLY-ROBERTS, Diana L, NAMOVIC, Marian T, GRAYSON, George, HONORE, Prisca, JARVIS, Michael F

Volltext

Discovery of a Series of Cyclohexylethylamine-Containing Protein Farnesyltransferase Inhibitors Exhibiting Potent Cellular Activity von Henry, Kenneth J, Wasicak, James, Tasker, Andrew S, Cohen, Jerome, Ewing, Patricia, Mitten, Michael, Larsen, John J, Kalvin, Douglas M, Swenson, Rolf, Ng, Shi-Chung, Saeed, Badr, Cherian, Sajeev, Sham, Hing, Rosenberg, Saul H

Volltext

Structure−Activity Relationship Studies on N ′-Aryl Carbohydrazide P2X 7 Antagonists von Nelson, Derek W., Sarris, Kathy, Kalvin, Douglas M., Namovic, Marian T., Grayson, George, Donnelly-Roberts, Diana L., Harris, Richard, Honore, Prisca, Jarvis, Michael F., Faltynek, Connie R., Carroll, William A.

Volltext

Novel and potent 3-(2,3-dichlorophenyl)-4-(benzyl)-4H-1,2,4-triazole P2X sub(7) antagonists von Carroll, William A, Kalvin, Douglas M, Medrano, Arturo Perez, Florjancic, Alan S, Wang, Ying, Donnelly-Roberts, Diana L, Namovic, Marian T, Grayson, George, Honore, Prisca, Jarvis, Michael F

Volltext

Novel and potent 3-(2,3-dichlorophenyl)-4-(benzyl)-4 H-1,2,4-triazole P2X 7 antagonists von Carroll, William A., Kalvin, Douglas M., Perez Medrano, Arturo, Florjancic, Alan S., Wang, Ying, Donnelly-Roberts, Diana L., Namovic, Marian T., Grayson, George, Honoré, Prisca, Jarvis, Michael F.

Volltext

Synthesis of (4R)-D,L-[4-2H]- and (4S)-D,L-[42H]homoserine lactones von Kalvin, Douglas M, Woodard, Ronald W

Volltext

Synthesis of (1S,2R)- and (1S,2S)-1-amino[2-2H]cyclopropane-1-carboxylic acids: The total 1H NMR assignment of cyclo[ACC-.alpha.-methyl-Phe] von Subramanian, Pullachipatti K, Kalvin, Douglas M, Ramalingam, Kondareddiar, Woodard, Ronald W

Volltext

Preparation of 1-deuterioaldehydes via tub use of diisobutylaluminum deuteride (DIBAL-D) von Kalvin, Douglas M., Woodard, Ronald W.

Volltext

A practical large scale chemical synthesis of chiral glycines von Ramalingam, Kondareddiar, Nanjappan, Palaniappagownder, Kalvin, Douglas M., Woodard, Ronald W.

Volltext

PEPTIDE ANTIANGIOGENIC DRUGS von HENKIN, JACK, SCHNEIDER, ANDREW J, HAVIV, FORTUNA, BRADLEY, MICHAEL F, KALVIN, DOUGLAS M

Volltext bestellen

5-HETEROARYL SUBSTITUTED INDAZOLES AS KINASE INHIBITORS von BAKKER MARGARETHA, LI BIQIN, ST JOHN MOORE NIGEL, PATEL JYOTI R, MACK HELMUT, KALVIN DOUGLAS M, AKRITOPOULOU-ZANZE IRINI, LONG ANDREW J, FRANK KRISTINE, JOHNSON ERIC T, GRACIAS VIJAYA J, WAKEFIELD BRIAN D, SARRIS KATHY, HOBSON ADRIAN D, TURNER SEAN C, WANG LU, TEUSCH NICOLE, GASIECKI ALAN F, VASUDEVAN ANIL, SHUAI QI, MICHMERHUIZEN MELISSA J, GEORGE DAWN, KOVAR PETER J, DJURIC STEVAN W

Volltext bestellen

5-substituted indazoles as kinase inhibitors von BAKKER MARGARETHA H. M, PENNING THOMAS D, LI BIQIN, MACK HELMUT, KALVIN DOUGLAS M, GRACIAS VIJAYA J, HOBSON ADRIAN D, TEUSCH NICOLE, GASIECKI ALAN F, SHUAI QI, VASUDEVAN ANIL, GEORGE DAWN M, SARRIS KATHY A, PATEL JYOTI R, JOHNSON ERIC F, AKRITOPOULOU-ZANZE IRINI, LONG ANDREW J, WOODS KEITH W, WAKEFIELD BRIAN D, TURNER SEAN C, WANG LU, MOORE NIGEL S, SWANN, JR. STEVEN L, MICHMERHUIZEN MELISSA J, MIYASHIRO JULIE M, KOVAR PETER J, DJURIC STEVAN W

Volltext bestellen

Novel and Potent 3‐(2,3‐Dichlorophenyl)‐4‐(benzyl)‐4H‐1,2,4‐triazole P2X 7 Antagonists von Carroll, William A., Kalvin, Douglas M., Perez‐Medrano, Arturo, Florjancic, Alan S., Wang, Ying, Donnelly‐Roberts, Diana L., Namovic, Marian T., Grayson, George, Honore, Prisca, Jarvis, Michael F.

Volltext

PEPTIDE ANTIANGIOGENIC DRUGS von HAVIV FORTUNA, KALVIN DOUGLAS M, HENKIN JACK, SCHNEIDER ANDREW J, BRADLEY MICHAEL F

Volltext bestellen

INDAZÓIS 5-HETEROARIL SUBSTITUÍDOS COMO INIBIDORES DE QUINASE von ALAN F GASIECKI, MELISSA J. MICHMERHUIZEN, ERIC F. JOHNSON, BIQIN LI, NIGEL ST. JOHN MOORE, NICOLE TEUSCH, PETER J KOVAR, ANIL VASUDEVAN, DAWN GEORGE, KATHY SARRIS, JYOTI R. PATEL, LU WANG, VIJAVA J GRACIAS, HELMUT MACK, DOUGLAS M KALVIN, BRIAN D. WAKEFIELD, ADRIAN HOBSON, SEAN C. TURNER, MARGARETHA BAKKER, IRINI AKRITOPOULOU-ZANZE, ANDREW J LONG, QI SHUAI, KRISTINE FRANK, STEVAN W DJURIC

Volltext bestellen

Peptide antiangiogenic drugs, pharmaceutical composition containing the same, and their use von HAVIV FORTUNA, KALVIN DOUGLAS M, HENKIN JACK, SCHNEIDER ANDREW J, BRADLEY MICHAEL F

Volltext bestellen

BENZOYL AMINO ACID DERIVATIVES USEFUL AS INHIBITORS OF PROTEIN ISOPRENYL TRANFERASES von AUGERI, DAVID J, SULLIVAN, GERARD M, WINN, MARTIN, SHEN, WANG, ROSENBERG, SAUL H, LARSEN, JOHN J, FAKHOURY, STEPHEN A, DONNER, BERNARD G, LIU, GANG, WASICK, JAMES I, O'CONNOR, STEPHEN J, SZCZEPANKIEWICZ, BRUCE G, BARR, KENNETH J, SWENSON, ROLF E, TASKER, ANDREW S, SEBTI, SAID M, SORENSEN, BRYAN K, JANOWICK, DAVID A, HAMILTON, ANDREW D, KALVIN, DOUGLAS M

Volltext bestellen

PEPTIDE ANTIANGIOGENIC DRUGS von HAVIV FORTUNA, KALVIN DOUGLAS M, HENKIN JACK, SCHNEIDER ANDREW J, BRADLEY MICHAEL F

Volltext bestellen