Preclinical Pharmacology of BMS-275183, an Orally Active Taxane von ROSE, William C, LONG, Byron H, FAIRCHILD, Craig R, LEE, Francis Y. F, KADOW, John F

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Synthesis and Antitumor Activity of Novel C-7 Paclitaxel Ethers:  Discovery of BMS-184476 von Altstadt, Thomas J, Fairchild, Craig R, Golik, Jerzy, Johnston, Kathy A, Kadow, John F, Lee, Francis Y, Long, Byron H, Rose, William C, Vyas, Dolatrai M, Wong, Henry, Wu, Mu-Jen, Wittman, Mark D

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Structure–activity relationships study at the 3′- N position of paclitaxel. part 2: synthesis and biological evaluation of 3′- N-thiourea- and 3′- N-thiocarbamate-bearing paclitaxe... von Xue, May, Long, Byron H, Fairchild, Craig, Johnston, Kathy, Rose, William C, Kadow, John F, Vyas, Dolatrai M, Chen, Shu-Hui

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Monoclonal antibody-.beta.-lactamase conjugates for the activation of a cephalosporin mustard prodrug von Svensson, Hakan P, Kadow, John F, Vrudhula, Vivekananda M, Wallace, Philip M, Senter, Peter D

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Phosphocholine conjugation: an unexpected in vivo conjugation pathway associated with hepatitis c ns5b inhibitors featuring a bicyclo[1.1.1]pentane von Zhuo, Xiaoliang, Cantone, Joseph L, Wang, Yingzi, Leet, John E, Drexler, Dieter M, Yeung, Kap-Sun, Huang, Xiaohua Stella, Eastman, Kyle J, Parcella, Kyle E, Mosure, Kathleen W, Soars, Matthew G, Kadow, John F, Johnson, Benjamin M

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Synthesis and antitumor activity of novel paclitaxel–chlorambucil hybrids von Wittman, Mark D., Kadow, John F., Vyas, Dolatrai M., Lee, Francis L., Rose, William C., Long, Byron H., Fairchild, Craig, Johnston, Kathy

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Synthesis of etoposide lactam via a mitsunobu reaction sequence von Kadow, J.F., Vyas, D.M., Doyle, T.W.

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Synthesis and bioactivity of 2,4-diacyl analogues of paclitaxel von Chordia, Mahendra D, Yuan, Haiqing, Jagtap, Prakash G, Kadow, John F, Long, Byron H, Fairchild, Craig R, Johnston, Kathy A, Kingston, David G.I

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Synthesis of a novel C-10 spiro-epoxide of paclitaxel von Walker, Michael A., Johnson, Timothy D., Huang, Stella, Vyas, Dolatorai M., Kadow, John F.

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Synthesis of metabolically blocked paclitaxel analogues von Wittman, Mark D., Altstadt, Thomas J., Fairchild, Craig, Hansel, Stephen, Johnston, Kathy, Kadow, John F., Long, Byron H., Rose, William C., Vyas, Dolatrai M., Wu, Mu-Jen, Zoeckler, Mary E.

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A base-catalyzed, direct synthesis of 3,5-disubstituted 1,2,4-triazoles from nitriles and hydrazides von Yeung, Kap-Sun, Farkas, Michelle E., Kadow, John F., Meanwell, Nicholas A.

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Structure-activity relationships of taxol®: synthesis and biological evaluation of C2 taxol analogs von Chen, Shu-Hui, Farina, Vittorio, Wei, Jian-Mei, Long, Bryon, Fairchild, Craig, Mamber, Stephen W., Kadow, John F., Vyas, Dolatrai, Doyle, Terrence W.

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Convergent approach to intermediates used for the synthesis of the enediyne structure of the esperamicins and calicheamicins von Kadow, J.F., Saulnier, M.G., Tun, M.M., Langley, D.R., Vyas, D.M.

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A chemoselective approach to functionalize the C-10 position of 10-deacetylbaccatin III. Synthesis and biological properties of novel C-10 Taxol® analogues von Kant, Joydeep, O'Keeffe, Wendy S., Chen, Shu-Hui, Farina, Vittorio, Fairchild, Craig, Johnston, Kathy, Kadow, John F., Long, Byron H., Vyas, Dolatrai

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New dual inhibitors of EGFR and HER2 protein tyrosine kinases von Fink, Brian E., Vite, Gregory D., Mastalerz, Harold, Kadow, John F., Kim, Soong-Hoon, Leavitt, Kenneth J., Du, Karen, Crews, Donald, Mitt, Toomas, Wong, Tai W., Hunt, John T., Vyas, Dolatrai M., Tokarski, John S.

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Structure-activity relationships study at the 3′-N position of paclitaxel-part 1: Synthesis and biological evaluation of the 3′-( t)-butylaminocarbonyloxy bearing paclitaxel analog... von Chen, Shu-Hui, Xue, May, Huang, Stella, Long, Byron H, Fairchild, Craig A, Rose, William C, Kadow, John F, Vyas, Dolatrai

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A Strategy for the Synthesis of Aryl α-Ketoamides Based upon the Acylation of Anions Derived from Cyanomethylamines Followed by Oxidative Cleavage von Yang, Zhong, Zhang, Zhongxing, Meanwell, Nicholas A, Kadow, John F, Wang, Tao

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An Effective Procedure for the Acylation of Azaindoles at C-3 von Zhang, Zhongxing, Yang, Zhong, Wong, Henry, Zhu, Juliang, Meanwell, Nicholas A, Kadow, John F, Wang, Tao

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Chemoselective synthesis of allyltrimethylsilanes by cross-coupling of vinyl triflates with tris((trimethylsilyl)methyl)aluminum catalyzed by palladium(0) von Saulnier, Mark G, Kadow, John F, Tun, Min Min, Langley, David R, Vyas, Dolatrai M

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A General Method for the Preparation of 4- and 6-Azaindoles von Zhang, Zhongxing, Yang, Zhong, Meanwell, Nicholas A, Kadow, John F, Wang, Tao

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