2-aminobenzimidazoles for leishmaniasis: From initial hit discovery to in vivo profiling von Ferreira, Rafael Augusto Alves, Junior, Celso de Oliveira Rezende, Martinez, Pablo David Grigol, Koovits, Paul John, Soares, Bruna Miranda, Ferreira, Leonardo L G, Michelan-Duarte, Simone, Chelucci, Rafael Consolin, Andricopulo, Adriano D, Galuppo, Mariana K, Uliana, Silvia R B, Matheeussen, An, Caljon, Guy, Maes, Louis, Campbell, Simon, Kratz, Jadel M, Mowbray, Charles E, Dias, Luiz Carlos

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Synthetic Studies toward the Total Synthesis of Tautomycetin von Pereira de Sant’Ana, Danilo, de Oliveira Rezende Júnior, Celso, Campagne, Jean-Marc, Dias, Luiz Carlos, Marcia de Figueiredo, Renata

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Chemoinformatics Studies on a Series of Imidazoles as Cruzain Inhibitors von Medeiros, Alex R, Ferreira, Leonardo L G, de Souza, Mariana L, de Oliveira Rezende Junior, Celso, Espinoza-Chávez, Rocío Marisol, Dias, Luiz Carlos, Andricopulo, Adriano D

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Discovery of Potent, Reversible, and Competitive Cruzain Inhibitors with Trypanocidal Activity: A Structure-Based Drug Design Approach von de Souza, Mariana L, de Oliveira Rezende Junior, Celso, Ferreira, Rafaela S, Espinoza Chávez, Rocio Marisol, Ferreira, Leonardo L. G, Slafer, Brian W, Magalhães, Luma G, Krogh, Renata, Oliva, Glaucius, Cruz, Fabio Cardoso, Dias, Luiz Carlos, Andricopulo, Adriano D

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Structure‐Metabolism Relationships of Benzimidazole Derivatives with anti‐Trypanosoma cruzi Activity for Chagas Disease von Espinoza‐Chávez, Rocío Marisol, Oliveira Rezende Júnior, Celso, Laureano de Souza, Mariana, Consolin Chelucci, Rafael, Michelan‐Duarte, Simone, Krogh, Renata, Gomes Ferreira, Leonardo Luiz, Valli, Marilia, Sena de Oliveira, Aldo, Andricopulo, Adriano D., Carlos Dias, Luiz

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A Novel Compound from the Phenylsulfonylpiperazine Class: Evaluation of In Vitro Activity on Luminal Breast Cancer Cells von da Silva, Fernanda Cardoso, Martinho, Ana Clara Cassiano, Ferreira, Helen Soares Valença, Siqueira, Raoni Pais, Arruda, Vinicius Marques, Guerra, Joyce Ferreira da Costa, de Souza, Maria Laura Dos Reis, Landin, Emanuelly Silva, Rezende Júnior, Celso de Oliveira, de Araújo, Thaise Gonçalves

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Synthesis, Design, and Structure‐Activity Relationship of a Benzenesulfonylpiperazine Series against Trypanosoma cruzi von Cassiano Martinho, Ana Clara, Melo Resende, Daniela, Landin, Emanuelly Silva, Dit Lapierre, Thibault Joseph William Jacques, Bernardes, Talita Cristina Diniz, Martins, Luan Carvalho, Ferreira, Rafaela Salgado, Murta, Silvane Maria Fonseca, Oliveira Rezende Júnior, Celso

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Evaluation and discovery of novel benzothiazole derivatives as promising hits against Leishmania infantum von Lapierre, Thibault Joseph William Jacques Dit, Farago, Danilo Nascimento, de Moura Lodi Cruz, Mariza Gabriela Faleiro, de Melo Resende, Daniela, de Oliveira, Adriane Cristina Rosa, Dos Santos, Brenda Rosa Macedo, de Oliveira Souza, Felipe, Michelan-Duarte, Simone, Chelucci, Rafael C, Andricopulo, Adriano D, Ferreira, Leonardo L G, Pilau, Eduardo Jorge, Murta, Silvane Maria Fonseca, de Oliveira Rezende Júnior, Celso

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New Palladium(II) Complexes Containing Methyl Gallate and Octyl Gallate: Effect against Mycobacterium tuberculosis and Campylobacter jejuni von Silva, Raphael Tristão Cruvinel, Guidotti-Takeuchi, Micaela, Peixoto, Jéssica Laura Miranda, Demarqui, Fernanda Manaia, Mori, Ananda Paula, Dumont, Carolyne Ferreira, Ferreira, Gabriella Rayane Aparecida, Pereira, Gabriele de Menezes, Rossi, Daise Aparecida, Corbi, Pedro Paulo, Pavan, Fernando Rogério, Rezende Júnior, Celso de Oliveira, Melo, Roberta Torres de, Guerra, Wendell

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Quinic acid derivatives inhibit dengue virus replication in vitro von Zanello, Paula Rodrigues, Koishi, Andrea Cristine, Rezende Júnior, Celso de Oliveira, Oliveira, Larissa Albuquerque, Pereira, Adriane Antonia, de Almeida, Mauro Vieira, Duarte dos Santos, Claudia Nunes, Bordignon, Juliano

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Structure-based discovery of thiosemicarbazones as SARS-CoV-2 main protease inhibitors von Maltarollo, Vinícius Gonçalves, da Silva, Elany Barbosa, Kronenberger, Thales, Sena Andrade, Marina Mol, de Lima Marques, Gabriel V, Cândido Oliveira, Nereu J, Santos, Lucianna H, Oliveira Rezende Júnior, Celso de, Cassiano Martinho, Ana C, Skinner, Danielle, Fajtová, Pavla, M Fernandes, Thaís H, Silveira Dos Santos, Eduardo da, Rodrigues Gazolla, Poliana A, Martins de Souza, Ana P, da Silva, Milene Lopes, Dos Santos, Fabíola S, Lavorato, Stefânia N, Oliveira Bretas, Ana C, Carvalho, Diogo Teixeira, Franco, Lucas Lopardi, Luedtke, Stephanie, Giardini, Miriam A, Poso, Antti, Dias, Luiz C, Podust, Larissa M, Alves, Ricardo J, McKerrow, James, Andrade, Saulo F, Teixeira, Róbson R, Siqueira-Neto, Jair L, O'Donoghue, Anthony, de Oliveira, Renata B, Ferreira, Rafaela S

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Synthesis, design, and optimization of a potent and selective series of pyridylpiperazines as promising antimalarial agents von da Silva Oliveira, Douglas Davison, Paz, Franciarli, Brito, Nícolas Peterson Ferreira, Krüger, Arne, Martinho, Ana Clara Cassiano, Lapierre, Thibault Joseph William Jacques Dit, de Oliveira Souza, Felipe, Maltarollo, Vinícius G., Kronenberger, Thales, Mendes, Marina Sena, Nonato, Maria Cristina, Pilau, Eduardo Jorge, Wrenger, Carsten, Wunderlich, Gerhard, Rezende Júnior, Celso de Oliveira

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Hit-to-lead optimization of a pyrazinylpiperazine series against Leishmania infantum and Leishmania braziliensis von Jacques Dit Lapierre, Thibault Joseph William, Cruz, Mariza Gabriela Faleiro de Moura Lodi, Brito, Nícolas Peterson Ferreira, Resende, Daniela de Melo, Souza, Felipe de Oliveira, Pilau, Eduardo Jorge, da Silva, Meryck Felipe Brito, Neves, Bruno Junior, Murta, Silvane Maria Fonseca, Rezende Júnior, Celso de Oliveira

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Optimization of benzenesulfonyl derivatives as anti-Trypanosomatidae agents: Structural design, synthesis, and pharmacological assessment against Trypanosoma cruzi and Leishmania i... von Freitas de Lima Hercos, Guilherme, Gabriela Faleiro de Moura Lodi Cruz, Mariza, Clara Cassiano Martinho, Ana, de Melo Resende, Daniela, Farago Nascimento, Danilo, Derksen Macruz, Paula, Jorge Pilau, Eduardo, Maria Fonseca Murta, Silvane, de Oliveira Rezende Júnior, Celso

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Discovery of Arylpiperazines with Broad-Spectrum Antimicrobial Activity and Favorable Pharmacokinetic Profiles von da Silva Oliveira, Douglas Davison, Sousa Silva, Nagela Bernadelli, Jacques Dit Lapierre, Thibault Joseph William, Lemes de Souza, Sara, Ferreira Brito, Nícolas Peterson, Cassiano Martinho, Ana Clara, Clemente Dias, Renieidy Flávia, Nascimento Farago, Danilo, Michelan-Duarte, Simone, Consolin Chelucci, Rafael, de Moura Lodi Cruz, Mariza Gabriela Faleiro, de Melo Resende, Daniela, Andricopulo, Adriano D, Fonseca Murta, Silvane Maria, Ferreira, Leonardo L G, Gomes Martins, Carlos Henrique, de Oliveira Rezende Júnior, Celso

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Discovery and structural optimization of a new series of N-acyl-2-aminobenzothiazole as inhibitors of Zika virus von Flávia Clemente Dias, Renieidy, Murta Rezende Moraes Ribeiro, Beatriz, Marques Cassani, Natasha, Nascimento Farago, Danilo, André Antoniucci, Giovanna, Eduardo de Oliveira Rocha, Rafael, de Oliveira Souza, Felipe, Jorge Pilau, Eduardo, Carolina Gomes Jardim, Ana, Salgado Ferreira, Rafaela, de Oliveira Rezende Júnior, Celso

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Crystal structure and in vitro biological studies of a Pt(II) complex based on gallic acid and triphenylphosphine von Tristão Cruvinel Silva, Raphael, Pereira Silva-Caldeira, Priscila, Manaia Demarqui, Fernanda, Duque Lopes, Carla, de Albuquerque, Sérgio, Rogério Pavan, Fernando, Cristina Pereira-Maia, Elene, Diniz, Renata, de Oliveira, Alberto, de Oliveira Rezende Júnior, Celso, Guerra, Wendell

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Hit-to-lead optimization of a 2-aminobenzimidazole series as new candidates for chagas disease von de Oliveira Rezende Júnior, Celso, Martinez, Pablo David Grigol, Ferreira, Rafael Augusto Alves, Koovits, Paul John, Miranda Soares, Bruna, Ferreira, Leonardo L.G., Michelan-Duarte, Simone, Chelucci, Rafael Consolin, Andricopulo, Adriano D., Matheeussen, An, Van Pelt, Natascha, Caljon, Guy, Maes, Louis, Campbell, Simon, Kratz, Jadel M., Mowbray, Charles E., Dias, Luiz Carlos

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New Palladium Complexes Containing Methyl Gallate and Octyl Gallate: Effect against IMycobacterium tuberculosis/I and ICampylobacter jejuni/I von Silva, Raphael Tristão Cruvinel, Guidotti-Takeuchi, Micaela, Peixoto, Jéssica Laura Miranda, Demarqui, Fernanda Manaia, Mori, Ananda Paula, Dumont, Carolyne Ferreira, Ferreira, Gabriella Rayane Aparecida, Pereira, Gabriele de Menezes, Rossi, Daise Aparecida, Corbi, Pedro Paulo, Pavan, Fernando Rogério, Rezende Júnior, Celso de Oliveira, Melo, Roberta Torres de, Guerra, Wendell

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Structure–activity relationships of novel N-imidazoylpiperazines with potent anti-Trypanosoma cruzi activity von Marisol Espinoza-Chavez, Rocio, de Oliveira Rezende Junior, Celso, de Souza, Mariana Laureano, Pauli, Ivani, Valli, Marilia, Ferreira, Leonardo Luiz Gomes, Chelucci, Rafael Consolin, Michelan-Duarte, Simone, Krogh, Renata, Bezerra Romualdo da Silva, Fernando, Cruz, Fabio Cardoso, Sena de Oliveira, Aldo, Andricopulo, Adriano Defini, Dias, Luiz Carlos

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