Characterization of a KDM5 small molecule inhibitor with antiviral activity against hepatitis B virus von Sarah A Gilmore, Danny Tam, Tara L Cheung, Chelsea Snyder, Julie Farand, Ryan Dick, Mike Matles, Joy Y Feng, Ricardo Ramirez, Li Li, Helen Yu, Yili Xu, Dwight Barnes, Gregg Czerwieniec, Katherine M Brendza, Todd C Appleby, Gabriel Birkus, Madeleine Willkom, Tetsuya Kobayashi, Eric Paoli, Marc Labelle, Thomas Boesen, Chin H Tay, William E Delaney, Gregory T Notte, Uli Schmitz, Becket Feierbach

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Sequence Confirmation of Modified Oligonucleotides Using Chemical Degradation, Electrospray Ionization, Time-of-Flight, and Tandem Mass Spectrometry von Farand, Julie, Beverly, Michael

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Selectivity switch between FAK and Pyk2: Macrocyclization of FAK inhibitors improves Pyk2 potency von Farand, Julie, Mai, Nicholas, Chandrasekhar, Jayaraman, Newby, Zachary E., Van Veldhuizen, Josh, Loyer-Drew, Jennifer, Venkataramani, Chandrasekar, Guerrero, Juan, Kwok, Amy, Li, Ning, Zherebina, Yelena, Wilbert, Sibylle, Zablocki, Jeff, Phillips, Gary, Watkins, William J., Mourey, Robert, Notte, Gregory T.

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Progress toward the Total Synthesis of (±)-Havellockate von Beingessner, Rachel L, Farand, Julie A, Barriault, Louis

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De Novo Sequence Determination of Modified Oligonucleotides von Farand, Julie, Gosselin, Francis

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Discovery of GS-2278, a Potent and Selective LPAR1 Antagonist for the Treatment of Idiopathic Pulmonary Fibrosis von Tang, Doris T, Du, Zhimin, Yang, Kin S, Bestvater, Brian P, Kaplan, Joshua, Neubig, Megan E, Olen, Casey L, Phillips, Bart, Wang, Peiyuan, Hudson, Thomas, Marchand, Bruno, Chan, Julie, Sharma, Monika, Hu, Yiding, Matles, Mike, Nejati, Elham, Chojnacka, Maja, Adams, Clifton, Pong, Cassie, Holsapple, Kevin, Budas, Grant, Tsui, Vickie, Venkataramani, Chandrasekar, Lazerwith, Scott E, Notte, Gregory T, Watkins, William J, McGlinchey, Ellen, Zagorska, Anna, Farand, Julie

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Characterization of a KDM5 small molecule inhibitor with antiviral activity against hepatitis B virus von Gilmore, Sarah A, Tam, Danny, Cheung, Tara L, Snyder, Chelsea, Farand, Julie, Dick, Ryan, Matles, Mike, Feng, Joy Y, Ramirez, Ricardo, Li, Li, Yu, Helen, Xu, Yili, Barnes, Dwight, Czerwieniec, Gregg, Brendza, Katherine M, Appleby, Todd C, Birkus, Gabriel, Willkom, Madeleine, Kobayashi, Tetsuya, Paoli, Eric, Labelle, Marc, Boesen, Thomas, Tay, Chin H, Delaney, 4th, William E, Notte, Gregory T, Schmitz, Uli, Feierbach, Becket

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Sequence Confirmation of Modified Oligonucleotides Using Chemical Degradation, Electrospray lonization, Time-of-Flight, and Tandem Mass Spectrometry von FARAND, Julie, BEVERLY, Michael

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Discovery of Potent and Selective MTH1 Inhibitors for Oncology: Enabling Rapid Target (In)Validation von Farand, Julie, Kropf, Jeffrey E, Blomgren, Peter, Xu, Jianjun, Schmitt, Aaron C, Newby, Zachary E, Wang, Ting, Murakami, Eisuke, Barauskas, Ona, Sudhamsu, Jawahar, Feng, Joy Y, Niedziela-Majka, Anita, Schultz, Brian E, Schwartz, Karen, Viatchenko-Karpinski, Serge, Kornyeyev, Dmytro, Kashishian, Adam, Fan, Peidong, Chen, Xiaowu, Lansdon, Eric B, Ports, Michael O, Currie, Kevin S, Watkins, William J, Notte, Gregory T

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Progress toward the Total Synthesis of (±)-Havelloekate von BEINGESSNER, Rachel L, FARAND, Julie A, BARRIAULT, Louis

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Improving the In Vivo Therapeutic Index of siRNA Polymer Conjugates through Increasing pH Responsiveness von Guidry, Erin N, Farand, Julie, Soheili, Arash, Parish, Craig A, Kevin, Nancy J, Pipik, Brenda, Calati, Kathleen B, Ikemoto, Nori, Waldman, Jacob H, Latham, Andrew H, Howell, Bonnie J, Leone, Anthony, Garbaccio, Robert M, Barrett, Stephanie E, Parmar, Rubina Giare, Truong, Quang T, Mao, Bing, Davies, Ian W, Colletti, Steven L, Sepp-Lorenzino, Laura

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The Discovery of 4-{1-[({2,5-Dimethyl-4-[4-(trifluoromethyl)benzyl]-3-thienyl}carbonyl)amino]cyclopropyl}benzoic Acid (MK-2894), A Potent and Selective Prostaglandin E 2 Subtype 4... von Blouin, Marc, Han, Yongxin, Burch, Jason, Farand, Julie, Mellon, Christophe, Gaudreault, Mireille, Wrona, Mark, Lévesque, Jean-François, Denis, Danielle, Mathieu, Marie-Claude, Stocco, Rino, Vigneault, Erika, Therien, Alex, Clark, Patsy, Rowland, Steve, Xu, Daigen, O’Neill, Gary, Ducharme, Yves, Friesen, Rick

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The Discovery of 4-{1-[({2,5-Dimethyl-4-[4-(trifluoromethyl)benzyl]-3-thienyl}carbonyl)amino]cyclopropyl}benzoic Acid (MK-2894), A Potent and Selective Prostaglandin E2 Subtype 4 R... von Blouin, Marc, Han, Yongxin, Burch, Jason, Farand, Julie, Mellon, Christophe, Gaudreault, Mireille, Wrona, Mark, Lévesque, Jean-François, Denis, Danielle, Mathieu, Marie-Claude, Stocco, Rino, Vigneault, Erika, Therien, Alex, Clark, Patsy, Rowland, Steve, Xu, Daigen, O’Neill, Gary, Ducharme, Yves, Friesen, Rick

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Naphthalene/quinoline amides and sulfonylureas as potent and selective antagonists of the EP₄ receptor von Burch, Jason D, Farand, Julie, Colucci, John, Sturino, Claudio, Ducharme, Yves, Friesen, Richard W, Lévesque, Jean-François, Gagné, Sébastien, Wrona, Mark, Therien, Alex G, Mathieu, Marie-Claude, Denis, Danielle, Vigneault, Erika, Xu, Daigen, Clark, Patsy, Rowland, Steve, Han, Yongxin

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Naphthalene/quinoline amides and sulfonylureas as potent and selective antagonists of the EP sub(4) receptor von Burch, Jason D, Farand, Julie, Colucci, John, Sturino, Claudio, Ducharme, Yves, Friesen, Richard W, Levesque, Jean-Francois, Gagne, Sebastien, Wrona, Mark, Therien, Alex G, Mathieu, Marie-Claude, Denis, Danielle, Vigneault, Erika, Xu, Daigen, Clark, Patsy, Rowland, Steve, Han, Yongxin

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Naphthalene/quinoline amides and sulfonylureas as potent and selective antagonists of the EP 4 receptor von Burch, Jason D., Farand, Julie, Colucci, John, Sturino, Claudio, Ducharme, Yves, Friesen, Richard W., Lévesque, Jean-François, Gagné, Sébastien, Wrona, Mark, Therien, Alex G., Mathieu, Marie-Claude, Denis, Danielle, Vigneault, Erika, Xu, Daigen, Clark, Patsy, Rowland, Steve, Han, Yongxin

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Structure-activity relationships and pharmacokinetic parameters of quinoline acylsulfonamides as potent and selective antagonists of the EP4 receptor von BURCH, Jason D, BELLEY, Michel, VIGNEAULT, Erika, LEVESQUE, Jean-Francois, GAGNE, Sébastien, WRONA, Mark, DAIGEN XU, CLARK, Patsy, ROWLAND, Steve, YONGXIN HAN, FORTIN, Réjean, DESCHENES, Denis, GIRARD, Mario, COLUCCI, John, FARAND, Julie, THERIEN, Alex G, MATHIEU, Marie-Claude, DENIS, Danielle

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Structure-activity relationships and pharmacokinetic parameters of quinoline acylsulfonamides as potent and selective antagonists of the EP sub(4) receptor von Burch, Jason D, Belley, Michel, tin, Rejean, Deschenes, Denis, Girard, Mario, Colucci, John, Farand, Julie, Therien, Alex G, Mathieu, Marie-Claude, Denis, Danielle, Vigneault, Erika, Levesque, Jean-Francois, Gagne, Sebastien, Wrona, Mark, Xu, Daigen, Clark, Patsy, Rowland, Steve, Han, Yongxin

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Structure–activity relationships and pharmacokinetic parameters of quinoline acylsulfonamides as potent and selective antagonists of the EP 4 receptor von Burch, Jason D., Belley, Michel, Fortin, Réjean, Deschênes, Denis, Girard, Mario, Colucci, John, Farand, Julie, Therien, Alex G., Mathieu, Marie-Claude, Denis, Danielle, Vigneault, Erika, Lévesque, Jean-François, Gagné, Sébastien, Wrona, Mark, Xu, Daigen, Clark, Patsy, Rowland, Steve, Han, Yongxin

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Sulfinylaminobenzamide and sulfonylaminobenzamide derivatives von Sangi, Michael, Sperandio, David, Notte, Gregory, Farand, Julie, Kaplan, Joshua A, Olen, Casey Lockwood

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