Discovery, Synthesis, and Biological Evaluation of Thiazoloquin(az)olin(on)es as Potent CD38 Inhibitors von Haffner, Curt D, Becherer, J. David, Boros, Eric E, Cadilla, Rodolfo, Carpenter, Tiffany, Cowan, David, Deaton, David N, Guo, Yu, Harrington, Wallace, Henke, Brad R, Jeune, Michael R, Kaldor, Istvan, Milliken, Naphtali, Petrov, Kim G, Preugschat, Frank, Schulte, Christie, Shearer, Barry G, Shearer, Todd, Smalley, Terrence L, Stewart, Eugene L, Stuart, J. Darren, Ulrich, John C

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Discovery of 4‑Amino-8-quinoline Carboxamides as Novel, Submicromolar Inhibitors of NAD-Hydrolyzing Enzyme CD38 von Becherer, J. David, Boros, Eric E., Carpenter, Tiffany Y., Cowan, David J., Deaton, David N., Haffner, Curt D., Jeune, Michael R., Kaldor, Istvan W., Poole, J. Chuck, Preugschat, Frank, Rheault, Tara R., Schulte, Christie A., Shearer, Barry G., Shearer, Todd W., Shewchuk, Lisa M., Smalley, Terrence L., Stewart, Eugene L., Stuart, J. Darren, Ulrich, John C.

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2,4-Diamino-8-quinazoline carboxamides as novel, potent inhibitors of the NAD hydrolyzing enzyme CD38: Exploration of the 2-position structure-activity relationships von Deaton, David N., Haffner, Curt D., Henke, Brad R., Jeune, Michael R., Shearer, Barry G., Stewart, Eugene L., Stuart, J. Darren, Ulrich, John C.

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A knowledge-based, structural-aided discovery of a novel class of 2-phenylimidazo[1,2-a]pyridine-6-carboxamide H-PGDS inhibitors von Schulte, Christie A., Deaton, David N., Diaz, Elsie, Do, Young, Gampe, Robert T., Guss, Jeffrey H., Hancock, Ashley P., Hobbs, Heather, Hodgson, Simon T., Holt, Jason, Jeune, Michael R., Kahler, Kirsten M., Kramer, H. Fritz, Le, Joelle, Mortenson, Paul N., Musetti, Caterina, Nolte, Robert T., Orband-Miller, Lisa A., Peckham, Gregory E., Petrov, Kim G., Pietrak, Beth L., Poole, Chuck, Price, Daniel J., Saxty, Gordon, Shillings, Anthony, Smalley, Terrence L., Somers, Don O., Stewart, Eugene L., Stuart, J. Darren, Thomson, Stephen A.

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The discovery of quinoline-3-carboxamides as hematopoietic prostaglandin D synthase (H-PGDS) inhibitors von Deaton, David N., Do, Young, Holt, Jason, Jeune, Michael R., Kramer, H. Fritz, Larkin, Andrew L., Orband-Miller, Lisa A., Peckham, Gregory E., Poole, Chuck, Price, Daniel J., Schaller, Lee T., Shen, Ying, Shewchuk, Lisa M., Stewart, Eugene L., Stuart, J. Darren, Thomson, Stephen A., Ward, Paris, Wilson, Joseph W., Xu, Tianshun, Guss, Jeffrey H., Musetti, Caterina, Rendina, Alan R., Affleck, Karen, Anders, David, Hancock, Ashley P., Hobbs, Heather, Hodgson, Simon T., Hutchinson, Jonathan, Leveridge, Melanie V., Nicholls, Harry, Smith, Ian E.D., Somers, Don O., Sneddon, Helen F., Uddin, Sorif, Cleasby, Anne, Mortenson, Paul N., Richardson, Caroline, Saxty, Gordon

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The exploration of aza-quinolines as hematopoietic prostaglandin D synthase (H-PGDS) inhibitors with low brain exposure von Cadilla, Rodolfo, Deaton, David N., Do, Young, Elkins, Patricia A., Ennulat, Daniela, Guss, Jeffrey H., Holt, Jason, Jeune, Michael R., King, Andrew G., Klapwijk, Jan C., Kramer, H. Fritz, Kramer, Nicholas J., Laffan, Susan B., Masuria, Paresh I., McDougal, Alan V., Mortenson, Paul N., Musetti, Caterina, Peckham, Gregory E., Pietrak, Beth L., Poole, Chuck, Price, Daniel J., Rendina, Alan R., Sati, Girish, Saxty, Gordon, Shearer, Barry G., Shewchuk, Lisa M., Sneddon, Helen F., Stewart, Eugene L., Stuart, J. Darren, Thomas, Dean N., Thomson, Stephen A., Ward, Paris, Wilson, Joseph W., Xu, Tiahshun, Youngman, Mark A.

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Discovery of 3-Aryl-4-isoxazolecarboxamides as TGR5 Receptor Agonists von Evans, Karen A, Budzik, Brian W, Ross, Sean A, Wisnoski, David D, Jin, Jian, Rivero, Ralph A, Vimal, Mythily, Szewczyk, George R, Jayawickreme, Channa, Moncol, David L, Rimele, Thomas J, Armour, Susan L, Weaver, Susan P, Griffin, Robert J, Tadepalli, Sarva M, Jeune, Michael R, Shearer, Todd W, Chen, Zibin B, Chen, Lihong, Anderson, Donald L, Becherer, J. David, De Los Frailes, Maite, Colilla, Francisco Javier

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Identification and Characterization of 4-Chloro-N-(2-{[5-trifluoromethyl)-2-pyridyl]sulfonyl}ethyl)benzamide (GSK3787), a Selective and Irreversible Peroxisome Proliferator-Activat... von Shearer, Barry G, Wiethe, Robert W, Ashe, Adam, Billin, Andrew N, Way, James M, Stanley, Thomas B, Wagner, Craig D, Xu, Robert X, Leesnitzer, Lisa M, Merrihew, Raymond V, Shearer, Todd W, Jeune, Michael R, Ulrich, John C, Willson, Timothy M

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Effect of Matrix Metalloproteinase Inhibition on Progression of Atherosclerosis and Aneurysm in LDL Receptor-Deficient Mice Overexpressing MMP-3, MMP-12, and MMP-13 and on Restenos... von PRESCOTT, MARGARET FORNEY, SAWYER, WILBUR K., VON LINDEN-REED, JEAN, JEUNE, MICHAEL, CHOU, MARY, CAPLAN, SHARI L., JENG, ARCO Y.

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A knowledge-based, structural-aided discovery of a novel class of 2-phe-nylimidazo[1,2-a]pyridine-6-carboxamide H-PGDS inhibitors von Schulte, Christie A., Deaton, David N., Diaz, Elsie, Do, Young, Gampe, Robert T., Guss, Jeffrey H., Hancock, Ashley P., Hobbs, Heather, Hodgson, Simon T., Holt, Jason, Jeune, Michael R., Kahler, Kirsten M., Kramer, H. Fritz, Le, Joelle, Mortenson, Paul N., Musetti, Caterina, Nolte, Robert T., Orband-Miller, Lisa A., Peckham, Gregory E., Petrov, Kim G., Pietrak, Beth L., Poole, Chuck, Price, Daniel J., Saxty, Gordon, Shillings, Anthony, Smalley, Terrence L., Somers, Don O., Stewart, Eugene L., Stuart, J. Darren, Thomson, Stephen A.

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CGP 43371 paradoxically inhibits development of rabbit atherosclerotic lesions while inducing extra-arterial foam cell formation von Feldman, David L, Sawyer, Wilbur K, Jeune, Michael R, Mogelesky, Therese C, Von Linden-Reed, Jean, Forney Prescott, Margaret

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Identification and Characterization of 4-Chloro-N-(2-{[5-trifluoromethyl)-2-pyridyl]sulfonyl}ethylbenzamide (GSK3787), a Selective and Irreversible Peroxisome Proliferator-Activate... von SHEARER, Barry G, WIETHE, Robert W, SHEARER, Todd W, JEUNE, Michael R, ULRICH, John C, WILLSON, Timothy M, ASHE, Adam, BILLIN, Andrew N, WAY, James M, STANLEY, Thomas B, WAGNER, Craig D, XU, Robert X, LEESNITZER, Lisa M, MERRIHEW, Raymond V

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Diaminoindanes as Microsomal Triglyceride Transfer Protein Inhibitors von Ksander, Gary M, deJesus, Reynalda, Yuan, Andrew, Fink, Cynthia, Moskal, Michael, Carlson, Eric, Kukkola, Paivi, Bilci, Natalie, Wallace, Eli, Neubert, Alan, Feldman, David, Mogelesky, Therese, Poirier, Kevin, Jeune, Michael, Steele, Ronald, Wasvery, Jong, Stephan, Zouhair, Cahill, Edna, Webb, Randy, Navarrete, Aida, Lee, Warren, Gibson, Joyce, Alexander, Natalya, Sharif, Haamid, Hospattankar, Ashok

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Enhanced Expression of Matrix Metalloproteinase-3, -12, and -13 mRNAs in the Aortas of Apolipoprotein E-deficient Mice with Advanced Atherosclerosis von JENG, ARCO, CHOU, MARY, SAWYER, WILBUR K., CAPLAN, SHARI L., LINDEN-REED, JEAN VON, JEUNE, MICHAEL, PRESCOTT, MARGARET FORNEY

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The in vitro and ex vivo antioxidant properties, and hypolipidemic activity of CGP 2881 von Feldman, David L, Mogelesky, Therese C, Sharif, Robin, Sawyer, W.Kit, Jeune, Michael, Hu, Chii-Whei, Leonards, Kenneth S, Forney Prescott, Margaret

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Dissertatio juridica De eo, quod justum est, circa pabulatorias militum excursiones, vulgo Fouragiren / quam... praeside Dn. Michaele Grasso... eruditorum examini subjicit Caspar C... von Corswant, Caspar. Auteur du texte

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HIV risk perception, risk behavior, and seroprevalence among female commercial sex workers in Georgetown, Guyana von Carter, K H, Harry, B P, Jeune, M, Nicholson, D

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Percepción del riesgo, comportamientos riesgosos y seroprevalencia del VIH en trabajadoras sexuales de Georgetown, Guyana von Carter, Keith H., Harry, Bhiro P., Jeune, Michael, Nicholson, Devian

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Restrictive versus liberal blood transfusion for acute upper gastrointestinal bleeding (TRIGGER): a pragmatic, open-label, cluster randomised feasibility trial von Jairath, Vipul, Dr, Kahan, Brennan C, MSc, Gray, Alasdair, FCEM, Doré, Caroline J, BSc, Mora, Ana, PhD, James, Martin W, MRCP, Stanley, Adrian J, FRCP, Everett, Simon M, MRCP, Bailey, Adam A, FRACP, Dallal, Helen, FRCP, Greenaway, John, FRCP, Le Jeune, Ivan, MRCP, Darwent, Melanie, FCEM, Church, Nicholas, MRCP, Reckless, Ian, MRCP, Hodge, Renate, MSc, Dyer, Claire, BSc, Meredith, Sarah, MFPHM, Llewelyn, Charlotte, PhD, Palmer, Kelvin R, FRCP, Logan, Richard F, Prof, Travis, Simon P, FRCP, Walsh, Timothy S, Prof, Murphy, Michael F, Prof

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Charpente en cloisonnage composée d'éléments croisés en forme de planches von ZENZ JOHANN, GROBL FRANZ, JEUNE MICHAEL MOSER

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