Rational Design of Nanobody80 Loop Peptidomimetics: Towards Biased β2 Adrenergic Receptor Ligands von Martin, Charlotte, Moors, Samuel L. C., Danielsen, Mia, Betti, Cecilia, Fabris, Cecilia, Sejer Pedersen, Daniel, Pardon, Els, Peyressatre, Marion, Fehér, Krisztina, Martins, José C., Mosolff Mathiesen, Jesper, Morris, May C., Devoogdt, Nick, Caveliers, Vicky, De Proft, Frank, Steyaert, Jan, Ballet, Steven

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Glepaglutide, a novel glucagon-like peptide-2 agonist, has anti-inflammatory and mucosal regenerative effects in an experimental model of inflammatory bowel disease in rats von Skarbaliene, Jolanta, Mathiesen, Jesper Mosolff, Larsen, Bjarne Due, Thorkildsen, Christian, Petersen, Yvette Miata

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Bitopic Ligands Support the Presence of a Metastable Binding Site at the β2 Adrenergic Receptor von Gaiser, Birgit Isabel, Danielsen, Mia, Xu, Xinyu, Røpke Jørgensen, Kira, Fronik, Philipp, Märcher-Rørsted, Emil, Wróbel, Tomasz M., Liu, Xiangyu, Mosolff Mathiesen, Jesper, Sejer Pedersen, Daniel

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Real-time trafficking and signaling of the glucagon-like peptide-1 receptor von Roed, Sarah Noerklit, Wismann, Pernille, Underwood, Christina Rye, Kulahin, Nikolaj, Iversen, Helle, Cappelen, Karen Arevad, Schäffer, Lauge, Lehtonen, Janne, Hecksher-Soerensen, Jacob, Secher, Anna, Mathiesen, Jesper Mosolff, Bräuner-Osborne, Hans, Whistler, Jennifer L., Knudsen, Sanne Moeller, Waldhoer, Maria

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A cAMP Biosensor-Based High-Throughput Screening Assay for Identification of Gs-Coupled GPCR Ligands and Phosphodiesterase Inhibitors von Vedel, Line, Bräuner-Osborne, Hans, Mathiesen, Jesper Mosolff

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Antagonism of the prostaglandin D2 receptor CRTH2 attenuates asthma pathology in mouse eosinophilic airway inflammation von Uller, Lena, Mathiesen, Jesper Mosolff, Alenmyr, Lisa, Korsgren, Magnus, Ulven, Trond, Högberg, Thomas, Andersson, Gunnar, Persson, Carl G A, Kostenis, Evi

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Rational Design of Nanobody80 Loop Peptidomimetics: Towards Biased β 2 Adrenergic Receptor Ligands von Martin, Charlotte, Moors, Samuel L C, Danielsen, Mia, Betti, Cecilia, Fabris, Cecilia, Sejer Pedersen, Daniel, Pardon, Els, Peyressatre, Marion, Fehér, Krisztina, Martins, José C, Mosolff Mathiesen, Jesper, Morris, May C, Devoogdt, Nick, Caveliers, Vicky, De Proft, Frank, Steyaert, Jan, Ballet, Steven

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Molecular Pharmacology and Therapeutic Prospects of Metabotropic Glutamate Receptor Allosteric Modulators von Ritzén, Andreas, Mathiesen, Jesper Mosolff, Thomsen, Christian

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Positive allosteric modulation of the human metabotropic glutamate receptor 4 (hmGluR4) by SIB‐1893 and MPEP von Mathiesen, Jesper Mosolff, Svendsen, Nannette, Bräuner‐Osborne, Hans, Thomsen, Christian, Ramirez, M Teresa

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Glycine: a long-sought novel ligand for GPR158 von Rosenkilde, Mette Marie, Mathiesen, Jesper Mosolff

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Identification of Indole Derivatives Exclusively Interfering with a G Protein-Independent Signaling Pathway of the Prostaglandin D2 Receptor CRTH2 von Mathiesen, Jesper Mosolff, Ulven, Trond, Martini, Lene, Gerlach, Lars Ole, Heinemann, Akos, Kostenis, Evi

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The metabotropic glutamate receptor 4 is internalized and desensitized upon protein kinase C activation von Mathiesen, Jesper Mosolff, Ramirez, M Teresa

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On the Mechanism of Interaction of Potent Surmountable and Insurmountable Antagonists with the Prostaglandin D2 Receptor CRTH2 von Mathiesen, Jesper Mosolff, Christopoulos, Arthur, Ulven, Trond, Royer, Julia F., Campillo, Mercedes, Heinemann, Akos, Pardo, Leonardo, Kostenis, Evi

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Structural insights into differences in G protein activation by family A and family B GPCRs von Hilger, Daniel, Kumar, Kaavya Krishna, Hu, Hongli, Pedersen, Mie Fabricius, O'Brien, Evan S, Giehm, Lise, Jennings, Christine, Eskici, Gözde, Inoue, Asuka, Lerch, Michael, Mathiesen, Jesper Mosolff, Skiniotis, Georgios, Kobilka, Brian K

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A new metabotropic glutamate receptor agonist with in vivo anti-allodynic activity von Stanley, Nathan J., Hutchinson, Mark R., Kvist, Trine, Nielsen, Birgitte, Mathiesen, Jesper Mosolff, Bräuner-Osborne, Hans, Avery, Thomas D., Tiekink, Edward R.T., Pedersen, Daniel Sejer, Irvine, Rodney J., Abell, Andrew D., Taylor, Dennis K.

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Negative allosteric modulation of the glucagon receptor by RAMP2 von Krishna Kumar, Kaavya, O’Brien, Evan S., Habrian, Chris H., Latorraca, Naomi R., Wang, Haoqing, Tuneew, Inga, Montabana, Elizabeth, Marqusee, Susan, Hilger, Daniel, Isacoff, Ehud Y., Mathiesen, Jesper Mosolff, Kobilka, Brian K.

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Bitopic Ligands Support the Presence of a Metastable Binding Site at the β 2 Adrenergic Receptor von Gaiser, Birgit Isabel, Danielsen, Mia, Xu, Xinyu, Røpke Jørgensen, Kira, Fronik, Philipp, Märcher-Rørsted, Emil, Wróbel, Tomasz M, Liu, Xiangyu, Mosolff Mathiesen, Jesper, Sejer Pedersen, Daniel

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Probing the Existence of a Metastable Binding Site at the β 2 -Adrenergic Receptor with Homobivalent Bitopic Ligands von Gaiser, Birgit I, Danielsen, Mia, Marcher-Rørsted, Emil, Røpke Jørgensen, Kira, Wróbel, Tomasz M, Frykman, Mikael, Johansson, Henrik, Bräuner-Osborne, Hans, Gloriam, David E, Mathiesen, Jesper Mosolff, Sejer Pedersen, Daniel

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Probing the Existence of a Metastable Binding Site at the β2‑Adrenergic Receptor with Homobivalent Bitopic Ligands von Gaiser, Birgit I, Danielsen, Mia, Marcher-Rørsted, Emil, Røpke Jørgensen, Kira, Wróbel, Tomasz M, Frykman, Mikael, Johansson, Henrik, Bräuner-Osborne, Hans, Gloriam, David E, Mathiesen, Jesper Mosolff, Sejer Pedersen, Daniel

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The C-terminal Tail of CRTH2 Is a Key Molecular Determinant That Constrains Gαi and Downstream Signaling Cascade Activation von Schröder, Ralf, Merten, Nicole, Mathiesen, Jesper Mosolff, Martini, Lene, Kruljac-Letunic, Anamarija, Krop, Friederike, Blaukat, Andree, Fang, Ye, Tran, Elizabeth, Ulven, Trond, Drewke, Christel, Whistler, Jennifer, Pardo, Leonardo, Gomeza, Jesús, Kostenis, Evi

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