Dual Inhibitors of Human DNA Topoisomerase II and Other Cancer-Related Targets von Skok, Žiga, Zidar, Nace, Kikelj, Danijel, Ilaš, Janez

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3,4-Dihydro-2H-1,4-benzoxazine Derivatives Combining Thrombin Inhibitory and Glycoprotein IIb/IIIa Receptor Antagonistic Activity as a Novel Class of Antithrombotic Compounds with... von Ilaš, Janez, Jakopin, Žiga, Borštnar, Tina, Stegnar, Mojca, Kikelj, Danijel

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Exploring protein hotspots by optimized fragment pharmacophores von Bajusz, Dávid, Wade, Warren S., Satała, Grzegorz, Bojarski, Andrzej J., Ilaš, Janez, Ebner, Jessica, Grebien, Florian, Papp, Henrietta, Jakab, Ferenc, Douangamath, Alice, Fearon, Daren, von Delft, Frank, Schuller, Marion, Ahel, Ivan, Wakefield, Amanda, Vajda, Sándor, Gerencsér, János, Pallai, Péter, Keserű, György M.

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Discovery of Benzothiazole Scaffold-Based DNA Gyrase B Inhibitors von Gjorgjieva, Marina, Tomašič, Tihomir, Barančokova, Michaela, Katsamakas, Sotirios, Ilaš, Janez, Tammela, Päivi, Peterlin Mašič, Lucija, Kikelj, Danijel

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Targeted Cancer Therapy Using Compounds Activated by Light von Dunkel, Petra, Ilas, Janez

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Identification of a Novel Structural Class of HV1 Inhibitors by Structure-Based Virtual Screening von Piga, Martina, Varga, Zoltan, Feher, Adam, Papp, Ferenc, Korpos, Eva, Bangera, Kavya C., Frlan, Rok, Ilaš, Janez, Dernovšek, Jaka, Tomašič, Tihomir, Zidar, Nace

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A road map for prioritizing warheads for cysteine targeting covalent inhibitors von Ábrányi-Balogh, Péter, Petri, László, Imre, Tímea, Szijj, Péter, Scarpino, Andrea, Hrast, Martina, Mitrović, Ana, Fonovič, Urša Pečar, Németh, Krisztina, Barreteau, Hélène, Roper, David I., Horváti, Kata, Ferenczy, György G., Kos, Janko, Ilaš, Janez, Gobec, Stanislav, Keserű, György M.

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Discovery of 4,5,6,7-Tetrahydrobenzo[1,2‑d]thiazoles as Novel DNA Gyrase Inhibitors Targeting the ATP-Binding Site von Tomašič, Tihomir, Katsamakas, Sotirios, Hodnik, Žiga, Ilaš, Janez, Brvar, Matjaž, Solmajer, Tom, Montalvão, Sofia, Tammela, Päivi, Banjanac, Mihailo, Ergović, Gabrijela, Anderluh, Marko, Mašič, Lucija Peterlin, Kikelj, Danijel

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Biolayer interferometry and its applications in drug discovery and development von Jug, Ana, Bratkovič, Tomaž, Ilaš, Janez

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Novel Potent and Selective Thrombin Inhibitors Based on a Central 1,4-Benzoxazin-3(4H)-one Scaffold von Ilaš, Janez, Tomašić, Tihomir, Kikelj, Danijel

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Influence of different classes of crosslinkers on alginate polyelectrolyte nanoparticle formation, thermodynamics and characteristics von Mirtič, Janja, Ilaš, Janez, Kristl, Julijana

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Rational design of balanced dual-targeting antibiotics with limited resistance von Nyerges, Akos, Tomasic, Tihomir, Durcik, Martina, Revesz, Tamas, Szili, Petra, Draskovits, Gabor, Bogar, Ferenc, Skok, Ziga, Zidar, Nace, Ilas, Janez, Zega, Anamarija, Kikelj, Danijel, Daruka, Lejla, Kintses, Balint, Vasarhelyi, Balint, Foldesi, Imre, Kata, Diana, Welin, Martin, Kimbung, Raymond, Focht, Dorota, Masic, Lucija Peterlin, Pal, Csaba

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N‑Phenyl-4,5-dibromopyrrolamides and N‑Phenylindolamides as ATP Competitive DNA Gyrase B Inhibitors: Design, Synthesis, and Evaluation von Zidar, Nace, Macut, Helena, Tomašič, Tihomir, Brvar, Matjaž, Montalvão, Sofia, Tammela, Päivi, Solmajer, Tom, Peterlin Mašič, Lucija, Ilaš, Janez, Kikelj, Danijel

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Recent progress in the discovery and development of DNA gyrase B inhibitors von Baran oková, Michaela, Kikelj, Danijel, Ilaš, Janez

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Exploring the Chemical Space of Benzothiazole-Based DNA Gyrase B Inhibitors von Skok, Žiga, Barančoková, Michaela, Benek, Ondřej, Cruz, Cristina Durante, Tammela, Päivi, Tomašič, Tihomir, Zidar, Nace, Mašič, Lucija Peterlin, Zega, Anamarija, Stevenson, Clare E. M, Mundy, Julia E. A, Lawson, David M, Maxwell, Anthony, Kikelj, Danijel, Ilaš, Janez

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Synthesis and Evaluation of Spumigin Analogues Library with Thrombin Inhibitory Activity von Žula, Aleš, Będziak, Izabela, Kikelj, Danijel, Ilaš, Janez

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On the Stability and Degradation Pathways of Venetoclax under Stress Conditions von Zigart, Nina, Crnugelj, Martin, Ilas, Janez, Casar, Zdenko

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Next-Generation Heterocyclic Electrophiles as Small-Molecule Covalent MurA Inhibitors von Ábrányi-Balogh, Péter, Keeley, Aaron, Ferenczy, György G, Petri, László, Imre, Tímea, Grabrijan, Katarina, Hrast, Martina, Knez, Damijan, Ilaš, Janez, Gobec, Stanislav, Keserű, György M

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Development of narrow-spectrum topoisomerase-targeting antibacterials against mycobacteria von Sterle, Maša, Habjan, Eva, Piga, Martina, Peršolja, Peter, Durcik, Martina, Dernovšek, Jaka, Szili, Petra, Czikkely, Marton Simon, Zidar, Nace, Janez, Ilaš, Pal, Csaba, Accetto, Tomaž, Pardo, Luis A., Kikelj, Danijel, Peterlin Mašič, Lucija, Tomašič, Tihomir, Bitter, Wilbert, Cotman, Andrej Emanuel, Speer, Alexander, Zega, Anamarija

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Discovery and Hit-to-Lead Optimization of Benzothiazole Scaffold-Based DNA Gyrase Inhibitors with Potent Activity against Acinetobacter baumannii and Pseudomonas aeruginosa von Cotman, Andrej Emanuel, Durcik, Martina, Benedetto Tiz, Davide, Fulgheri, Federica, Secci, Daniela, Sterle, Maša, Možina, Štefan, Skok, Žiga, Zidar, Nace, Zega, Anamarija, Ilaš, Janez, Peterlin Mašič, Lucija, Tomašič, Tihomir, Hughes, Diarmaid, Huseby, Douglas L., Cao, Sha, Garoff, Linnéa, Berruga Fernández, Talía, Giachou, Paraskevi, Crone, Lisa, Simoff, Ivailo, Svensson, Richard, Birnir, Bryndis, Korol, Sergiy V., Jin, Zhe, Vicente, Francisca, Ramos, Maria C., de la Cruz, Mercedes, Glinghammar, Björn, Lenhammar, Lena, Henderson, Sara R., Mundy, Julia E. A., Maxwell, Anthony, Stevenson, Clare E. M., Lawson, David M., Janssen, Guido V., Sterk, Geert Jan, Kikelj, Danijel

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