FRI0002 Inhibition of chemokine receptors ccr1 and ccr6 as promising therapies for rheumatoid arthritis von Jaen, J. C., Dairaghi, D., Leleti, M., Powers, J. P., Wang, Y., Zhang, P., Schall, T. J.

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OP0204 Characterization of the novel C5AR antagonist CCX168, a potential therapeutic for ANCA-vasculitis, rheumatoid arthritis, and other autoimmune disorders von Powers, J.P., Bekker, P.J., Dairaghi, D.J., Jennette, J.C., Johnson, D.A., Leleti, M., Miao, S., Seitz, L.C., Wang, Y., Xiao, H., Schall, T.J., Jaen, J.C.

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PD-90780, a Nonpeptide Inhibitor of Nerve Growth Factor′s Binding to the P75 NGF Receptor von Spiegel, K., Agrafiotis, D., Caprathe, B., Davis, R.E., Dickerson, M.R., Fergus, J.H., Hepburn, T.W., Marks, J.S., Vandorf, M., Wieland, D.M., Jaen, J.C.

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Pharmacological characterization of PD102807: An m4 subtype selective muscarinic antagonist von Schwarz, R.D., Nelson, C.B., Augelli-Szafran, C.E., Penvose, J.R., Jaen, J.C., Wiley, J., Frey, K.A.

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Identification and characterization of m4 selective muscarinic antagonists von Augelli-Szafran, C.E., Moreland, D.W., Nelson, C.B., Penvose-Yi, J.R., Schwarz, R.D., Jaen, J.C.

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Development of M1 subtype selective muscarinic agonists for Alzheimer's disease: Translation of in vitro selectivity into in vivo efficacy von Schwarz, R.D., Callahan, M.J., Davis, R.E., Jaen, J.C., Tecle, H.

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Functional characterisation of PD102807: A novel M4-selective muscarinic antagonist von Gross, J., Augelli-Szafran, C.E., Czeche, S., Friebe, T., Jaen, J.C., Penvose-Yi, J.R., Schwarz, R.D., Mutschier, E., Lambrecht, G.

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Functional characterisation of PD102807: A novel M 4-selective muscarinic antagonist von Gross, J., Augelli-Szafran, C.E., Czeche, S., Friebe, T., Jaen, J.C., Penvose-Yi, J.R., Schwarz, R.D., Mutschier, E., Lambrecht, G.

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Identification and characterization of m1 selective muscarinic antagonists von Augelli-Szafran, C.E., Blankley, C.J., Jaen, J.C., Moreland, D.W., Nelson, C.B., Penvose, J.R., Schwarz, R.D., Thomas, A.J.

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Aryleneyne 1-azabicyclo[2.2.1]heptan-3-one oximes: Potent muscarinic agonists von Tecle, H., Lauffer, D.J., Davis, R.E., Mirzadegan, T., Moreland, D.W., Schwarz, R.D., Thomas, A.J., Raby, C., Jaen, J.C.

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CI-1017, a functionally M1-selective muscarinic agonist: design, synthesis, and preclinical pharmacology von Tecle, H, Schwarz, R.D, Barrett, S.D, Callahan, M.J, Caprathe, B.W, Davis, R.E, Doyle, P, Emmerling, M, Lauffer, D.J, Mirzadegan, T, Moreland, D.W, Lipiniski, W, Nelson, C, Raby, C, Spencer, C, Spiegel, K, Thomas, A.J, Jaen, J.C

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(±)-1-Azabicyclo[2.2.1]heptan-3-one, O-(3-methyl-5-aryl-2-penten-4-ynyl) oximes: Potent muscarinic agonists von Tecle, H., Lauffer, D.J., Davis, R.E., Mirzadegan, T., Moreland, D.W., Schwan, R.D., Thomas, A.J., Raby, C., Eubanks, D., Brann, M.R., Jaen, J.C.

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Pharmacological characterization of PD150714: An m1 selective muscarinic antagonist von Nelson, C.B., Augelli-Szafran, C.E., Callahan, M.J., Christoffersen, C., Jaen, J.C., Meltzer, L.T., Penvose, J.R., Schwarz, R.D., Thomas, A.J., Wiley, J.

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Z-(±)-1-azabicyclo[2.2.1]heptan-3-one, O-(3-aryl-2-propynyl) oximes as potential m1-subtype selective muscarinic agonists von Tecle, H., Jaen, J.C., Augelli-Szafran, C., Barrett, S.D., Caprathe, B.W., Lauffer, D.J., Mirzadegan, T., Moos, W.H., Moreland, D.W., Pavia, M.R., Schwarz, R.D., Thomas, A.J., Davis, R.E.

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4H-1-BENZOPYRAN-4-ONE DERIVATIVES, SULPHUR ANALOGUES AND PHARMACEUTICAL COMPOSITIONS von WISE, L.D, JAEN, J.C

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Chemical purity and mutagenicity: Case study of a drug in development von Kropko, M.L., Jaen, J.C., Theiss, J.C., Wold, S., Caprathe, B.W., Wise, L.D.

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Anti-viral pyrimidine derivs von T.D. CUSHING, H.L. MELLON, J.C. JAEN

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(R)-(2)-1-azabicyclo [2,2,1]heptan-3-one, o-[3-(3-methoxyphenyl)2-propynyl] oxime maleate as a pharmaceuticals von H.Y. UNDO, J.C. JAEN, S.D. BARRETT

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Exceptional Activity for Methane Combustion over Modular Pd@CeO2 Subunits on Functionalized Al2O3 von CARGNELLO, M, DELGADO JAEN, J. J, HERNANDEZ GARRIDO, J. C, BAKHMUTSKY, K, MONTINI, T, CALVINO GAMEZ, J. J, GORTE, R. J, FORNASIERO, P

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Monkeypox virus case with maculopapular exanthem and proctitis during the Spanish outbreak in 2022 von Nicolas‐Ruanes, B., Vivancos, M.J., Azcarraga‐Llobet, C., Moreno, A.M., Rodriguez‐Dominguez, M., Berna‐Rico, E.D., Garcia‐Mouronte, E., Carron‐Herrero, A., McGee, A., Galan, J.C., Moreno, S., Jaen‐Olasolo, P., Fernandez‐Gonzalez, P.

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